中科微点-全球专利检索

  1. Login
  2. Sign Up

Search Results

92 records (took 0.049 seconds)

    PROCESS FOR PREPARING N-SUBSTITUTED 1H-PYRAZOLE-5-CARBOXYLIC ACID COMPOUNDS AND DERIVATIVES THEREOF
    4.
    发明公开
    PROCESS FOR PREPARING N-SUBSTITUTED 1H-PYRAZOLE-5-CARBOXYLIC ACID COMPOUNDS AND DERIVATIVES THEREOF 审中-公开
    PROCESS FOR制备N-取代的 - 吡唑1H-5-羧酸及其衍生物

    公开(公告)号：EP2997020A1

    公开(公告)日：2016-03-23

    申请号：EP14727749.5

    申请日：2014-05-16

    Applicant: BASF SE

    Inventor： KORADIN, Christopher ,  ZIERKE, Thomas ,  HOOCK, Ralf ,  KÖRBER, Karsten

    IPC: C07D401/04

    CPC classification number: C07D401/04

    Abstract: The present invention relates to a process for preparing N-substituted 1 H-pyrazole-5-carboxylic acid compounds of the formula l-A and derivatives thereof, in particular the corresponding carbonylchloride compounds (acid chlorides). It also relates to the use of these acid chlorides for preparing anthranilamide derivatives that are useful pesticides. in which the variables are as defined in the claims and the specification comprising the steps of i) reacting a compound of the formula (II) with a base selected from combinations of a magnesium-organic compound having a carbon bound magnesium and a secondary amine and magnesium amides of secondary amines in the presence of a lithium halide, where the base is used in an amount sufficient to achieve at least 80 % deprotonation of the compound of formula (II); and subjecting the product obtained in step (i) to a carboxylation by reacting it with carbon dioxide or a carbon dioxide equivalent, to obtain a magnesium salt of the compound of formula (l-A) and optionally aqueous workup to obtain the compound of the formula (l-A) as a free acid.

    ANILINE TYPE COMPOUNDS
    8.
    发明公开
    ANILINE TYPE COMPOUNDS 审中-公开
    苯胺类化合物

    公开(公告)号：EP2742021A1

    公开(公告)日：2014-06-18

    申请号：EP12745699.4

    申请日：2012-08-10

    Applicant: BASF SE

    Inventor： KÖRBER, Karsten ,  DESHMUKH, Prashant ,  KAISER, Florian ,  RACK, Michael ,  FRASSETTO, Timo ,  VEITCH, Gemma ,  KORDES, Markus ,  NAUJOK, Marco

    IPC: C07C381/10 ,  C07D401/04 ,  A01N37/28 ,  A01N43/56

    CPC classification number: A01N43/56 ,  A01N37/28 ,  A01N41/12 ,  A01N43/50 ,  A01N43/80 ,  C07B2200/13 ,  C07C381/10 ,  C07D401/04 ,  C07D401/14 ,  C07D409/14 ,  C07D413/14

    Abstract: The present invention relates to compounds of the formula (I) wherein R
    1 and R
    2 independently of one another are hydrogen, C
    1 -C
    10 -alkyl, C
    1 -C
    10 -haloalkyl, C
    3 -C
    10 -cycloalkyl, C
    3 -C
    10 -halocycloalkyl, C
    2 -C
    10 -alkenyl, C
    2 -C
    10 -haloalkenyl or together represent an aliphatic chain, or the like; R
    3 is halogen, cyano, C
    1 -C
    8 -alkyl, C
    1 -C
    8 - haloalkyl, C
    3 -C
    8 -cycloalkyl, C
    3 -C
    8 -halocycloalkyl, C
    2 -C
    8 -alkenyl, C
    2 -C
    8 -haloalkenyl, C
    1 -C
    8 -alkoxy, phenyl, or the like; R
    4 is hydrogen, C
    1 -C
    10 -alkyl, C
    1 -C
    10 -haloalkyl, C
    3 -C
    8 - cycloalkyl, C
    3 -C
    8 -halocycloalkyl, C
    2 -C
    10 -alkenyl, C
    2 -C
    10 -haloalkenyl, phenyl, or the like; t is 0 or 1; p is 0, 1, 2, 3 or 4. The present invention also relates to a process for preparing a compound of the formula (I) which comprises reacting a compound of the formula (II) with a compound of the formulae (III) or (IV): where t, p, R
    1 R
    3 , R
    3 and R
    4 are as defined in any of claims 1 to 6 and where A- is an equivalent of an anion having a pΚ
    B of at least 10 (determined under standard conditions in water).

Patent Agency Ranking