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1.发明授权4-(Aminomethyl)benzoic acids as intermediates for the preparation of chymase inhibiting 1,4-diazepan-2,5-dione compounds 有权4-（氨基甲基）苯甲酸作为中间体用于胃促胰酶抑制1,4-二氮杂环庚烷-2,5-二酮化合物的制备
公开(公告)号：EP2463268B1
公开(公告)日：2013-08-28
申请号：EP12156735.8
申请日：2005-12-01
IPC分类号： C07C229/38 , C07C229/56 , C07D307/68 , C07D333/40 , C07D213/79 , C07D213/80
CPC分类号： C07D243/08 , C07C233/47 , C07C271/22 , C07D213/79 , C07D213/80 , C07D243/10 , C07D307/68 , C07D333/40 , C07D401/06 , C07D401/12 , C07D403/12 , C07D405/06 , C07D405/12 , C07D409/12 , C07D413/12
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2.发明公开Aminomethyl-substituted aromatic acids as intermediates for the preparation of chymase inhibiting 1,4-diazepan-2,5-dione compounds 有权4-（Aminomethyl）benzoesäurenals Z chen chen ver b
公开(公告)号：EP2463268A1
公开(公告)日：2012-06-13
申请号：EP12156735.8
申请日：2005-12-01
IPC分类号： C07C229/38 , C07C229/56 , C07D307/68 , C07D333/40 , C07D213/79 , C07D213/80
CPC分类号： C07D243/08 , C07C233/47 , C07C271/22 , C07D213/79 , C07D213/80 , C07D243/10 , C07D307/68 , C07D333/40 , C07D401/06 , C07D401/12 , C07D403/12 , C07D405/06 , C07D405/12 , C07D409/12 , C07D413/12
摘要： A compound, or its salt or a solvate thereof, having the formula (Va):
for producing a 7-membered heterocyclic compound, or its salt or a solvate thereof having formula (I):
the compound of formula (I) having a chymase inhibitory action and useful for the prevention or treatment of various diseases in which chymase is involved and a method of producing a compound of formula (I) from a compound of formula (Va) are provided.摘要翻译： 具有式（Va）的化合物或其盐或其溶剂合物：用于制备具有式（I）的7-元杂环化合物或其盐或其溶剂化物：具有糜酶的式（I）化合物 提供抑制作用，并且可用于预防或治疗涉及胃促胰酶的各种疾病，以及由式（Va）化合物制备式（I）化合物的方法。
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