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1.发明公开DEPSIPEPTIDE DERIVATIVE, PROCESS FOR PRODUCTION THEREOF, AND NOVEL INTERMEDIATE THEREFOR 失效DEPSIPEPTID-DERIVAT，VERFAHREN ZU DESSEN HERSTELLUNG UND ZWISCHENPRODUKTDAFÜR
公开(公告)号：EP0872481A1
公开(公告)日：1998-10-21
申请号：EP96918897.8
申请日：1996-06-24
IPC分类号： C07D273/00 , C07C237/20 , A61K31/395
CPC分类号： C07D273/00
摘要： A novel industrial process for producing an anthelmintic depsipeptide derivative represented by structural formula (I), which is excellent in the yield etc.
摘要翻译： 一种用于生产由结构式（I）表示的驱虫剂去三肽衍生物的新型工业方法，其产率等优异
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公开(公告)号：EP0718293B1
公开(公告)日：2002-03-13
申请号：EP94925614.3
申请日：1994-08-31
IPC分类号： C07D273/00 , A61K31/395
CPC分类号： C07D273/00
摘要： A compound represented by general formula (I) or a salt thereof, having an excellent helminthicidal activity as a vermicide for humans and animals, wherein A represents appropriately substituted benzyl; Aa, B and D represent each lower alkyl; and C represents hydrogen or lower alkyl.
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3.发明公开PROCESS FOR PRODUCING DEPSIPEPTIDE DERIVATIVES AND NOVEL INTERMEDIATES THEREFOR 失效ZWISCHENPRODUKTEN DAVON VERFAHREN ZUR HERSTELLUNG VON DEPSIPEPTIDEN
公开(公告)号：EP0953563A1
公开(公告)日：1999-11-03
申请号：EP97941241.8
申请日：1997-09-24
发明人： YAMANISHI, Ryo , OHGAKI, Masaru
IPC分类号： C07C235/12 , C07D273/00 , A61K31/395
CPC分类号： C07D273/00 , C07C235/12 , C07D295/155 , Y02P20/55
摘要： An industrially excellent alternative process for producing cyclodepsipeptide derivatives, as represented in formula (1), having an excellent vermicidal activity as an animal and human anthelmintic, wherein R 1 represents hydrogen or a hydroxyl-protective group; R 2 represents a carboxyl group optionally protected; R 3 , R 4 , R 7 and R 8 represent each a lower alkyl, aryl or (un)substituted aralkyl; and R 5 , R 6 , R 9 and R 10 represent each a lower alkyl.
摘要翻译： 如式（1）所示的用于生产环糊精肽衍生物的工业上优异的替代方法，其具有优异的杀虫活性作为动物和人类驱虫剂，其中R1表示氢或羟基保护基; R2表示任选保护的羧基; R 3，R 4，R 7和R 8各自代表低级烷基，芳基或（取代）取代的芳烷基; 并且R 5，R 6，R 9和R 10各自表示低级烷基。
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公开(公告)号：EP0718293A1
公开(公告)日：1996-06-26
申请号：EP94925614.3
申请日：1994-08-31
IPC分类号： C07D273/00 , A61K31/395
CPC分类号： C07D273/00
摘要： A compound of the formula :
wherein
A is benzyl group which has suitable substituent (s),
A a , B and D are each lower alkyl,
C is hydrogen or lower alkyl,
or a salt thereof.
The compound or its salt of the present invention has excellent parasiticidal activities as parasiticides (anthelmintics) for animals and human bodies.摘要翻译： 具有下式的化合物：其中A为具有合适取代基的苄基，A a，B和D各自为低级烷基，C为氢或低级烷基或其盐。 本发明的化合物或其盐具有优异的杀虫活性，作为动物和人体的杀寄生虫剂（驱肠虫剂）。
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公开(公告)号：EP0634408B1
公开(公告)日：2002-01-02
申请号：EP93905622.2
申请日：1993-03-08
IPC分类号： C07D273/00 , C07D413/10 , C07D417/10 , C07D487/04 , C07D487/08 , A61K31/395 , C07K11/02
CPC分类号： C07D273/00
摘要： A compound represented by general formula (I) or a salt thereof, excellent in parasiticidal activity as an enthelmintic for animal and man, wherein A represents benzyl which is appropriately substituted or phenyl which may be appropriately substituted; A represents benzyl or phenyl each of which may be appropriately substituted; B and D represent each lower alkyl; and C represents hydrogen or lower alkyl.
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6.发明授权
公开(公告)号：EP0953563B1
公开(公告)日：2003-04-16
申请号：EP97941241.8
申请日：1997-09-24
发明人： YAMANISHI, Ryo , OHGAKI, Masaru
IPC分类号： C07C235/12 , C07D273/00 , A61K31/395
CPC分类号： C07D273/00 , C07C235/12 , C07D295/155 , Y02P20/55
摘要： An industrially excellent alternative process for producing cyclodepsipeptide derivatives, as represented in formula (1), having an excellent vermicidal activity as an animal and human anthelmintic, wherein R1 represents hydrogen or a hydroxyl-protective group; R2 represents a carboxyl group optionally protected; R3, R4, R7 and R8 represent each a lower alkyl, aryl or (un)substituted aralkyl; and R5, R6, R9 and R10 represent each a lower alkyl.
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公开(公告)号：EP0634408A1
公开(公告)日：1995-01-18
申请号：EP93905622.2
申请日：1993-03-08
IPC分类号： C07D273/00 , C07D413/10 , C07D417/10 , C07D487/04 , C07D487/08 , A61K31/395 , C07K11/02
CPC分类号： C07D273/00
摘要： A compound represented by general formula (I) or a salt thereof, excellent in parasiticidal activity as an enthelmintic for animal and man, wherein A represents benzyl which is appropriately substituted or phenyl which may be appropriately substituted; A a represents benzyl or phenyl each of which may be appropriately substituted; B and D represent each lower alkyl; and C represents hydrogen or lower alkyl.
摘要翻译： 由通式（I）表示的化合物或其盐作为动物和人的寄生虫具有优异的杀
虫活性，其中A代表被适当取代的苄基或可被适当取代的苯基; Aa代表各自可被适当取代的苄基或苯基; B和D代表每个低级烷基; C代表氢或低级烷基。
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