专利检索 ap:("Merck Sharp & Dohme Corp.") AND inv:"SARKAR, Sujit Kumar" 第 1 页

1.

发明公开
BICYCLIC HETEROCYCLES AS INHIBITORS OF CHOLESTEROL ESTER TRANSFER PROTEIN 审中-公开

公开(公告)号：EP3322420A1

公开(公告)日：2018-05-23

申请号：EP16824927.4

申请日：2016-07-08

申请人： Merck Sharp & Dohme Corp.

发明人： SHAO, Pengcheng Patrick , KATIPALLY, Revathi Reddy , VACHAL, Petr , THATAI, Jayanth Thiruvellore , SARKAR, Sujit Kumar

IPC分类号： A61K31/4439 , C07D498/04

CPC分类号： C07D513/04 , A61K31/407 , A61K31/429 , A61K31/4439 , A61K31/444 , A61K31/455 , A61K31/519 , A61K31/714 , A61K45/06 , C07D487/04 , C07D498/04 , A61K2300/00

摘要： The invention provides compounds having the structure of Formula I, including pharmaceutically acceptable salts of the compounds, wherein D1, D2, D3, X, Y, A1, A2, R1, R5 and the subscript a are as described herein. The compounds are CETP inhibitors and are useful for raising FIDL-cholesterol, reducing LDL-cholesterol, and for treating or preventing atherosclerosis:

2.

发明授权
NOVEL PYRROLIDINE DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS 有权

公开(公告)号：EP3052099B1

公开(公告)日：2019-08-21

申请号：EP14850990.4

申请日：2014-09-29

申请人： Merck Sharp & Dohme Corp.

发明人： BARR, Kenneth Jay , SCOTT, Mark E. , THOMPSON, Christopher F. , ANTHONY, Neville , CAMMARANO, Carolyn Michelle , BAKSHI, Raman Kumar , MOHANTY, Subhendu Kumar , KORAPALA, Chandra Sekhar , LATTHE, Prashant R. , KAMBAM, Vyjayanthi N. , SARKAR, Sujit Kumar , THATAI, Jayanth Thiruvellore

IPC分类号： A61K31/435 , A61K31/4439

3.

发明公开
NOVEL PYRROLIDINE DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS 审中-公开
标题翻译：中性粒细胞白血病抑制剂

公开(公告)号：EP3052099A1

公开(公告)日：2016-08-10

申请号：EP14850990.4

申请日：2014-09-29

申请人： Merck Sharp & Dohme Corp.

发明人： BARR, Kenneth Jay , SCOTT, Mark E. , THOMPSON, Christopher F. , ANTHONY, Neville , CAMMARANO, Carolyn Michelle , BAKSHI, Raman Kumar , MOHANTY, Subhendu Kumar , KORAPALA, Chandra Sekhar , LATTHE, Prashant R. , KAMBAM, Vyjayanthi N. , SARKAR, Sujit Kumar , THATAI, Jayanth Thiruvellore

IPC分类号： A61K31/435 , A61K31/4439

CPC分类号： A61K31/4439 , A61K31/437 , A61K31/444 , A61K31/497 , A61K31/501 , A61K31/506 , A61K31/517 , A61K31/519 , A61K45/06 , C07B2200/07 , C07C53/06 , C07C53/18 , C07D207/08 , C07D207/09 , C07D401/06 , C07D401/12 , C07D401/14 , C07D403/12 , C07D413/14 , C07D471/04 , C07D495/04 , A61K2300/00

摘要： The present invention provides compounds of Formula (I), pharmaceutical compositions thereof, and method of using the same in the treatment or prevention of diseases mediated by the activation of β3-adrenoceptor.

摘要翻译： 本发明提供式（I）化合物，其药物组合物及其用于治疗或预防β3肾上腺素受体激活介导的疾病的方法。