PROCESS FOR THE PREPARATION OF ENANTIOMERS OF AMIDOACETONITRILE COMPOUNDS FROM THEIR RACEMATES
    1.
    发明授权
    PROCESS FOR THE PREPARATION OF ENANTIOMERS OF AMIDOACETONITRILE COMPOUNDS FROM THEIR RACEMATES 有权
    用于从AMIDOACETONITRILVERBINDUNGEN的外消旋体PRODUCING对映体

    公开(公告)号:EP1812385B1

    公开(公告)日:2012-07-18

    申请号:EP05803815.9

    申请日:2005-11-07

    申请人: Novartis AG

    摘要: The invention is directed at a new process for the preparation of pure enantiomers from the racemate of amidoacetonitrile compounds of formula (I) wherein R1, R2 and R3, independently of each other, signify hydrogen, halogen, nitro, cyano, C1-C6­-alkyl, halogen-C1-C6-alkyl, C1-C6-alkoxy, halogen-C1-C6-alkoxy, C2-C6-alkenyl, halogen-C2­-C6-alkenyl, C2-C6-alkinyl, halogen-C2-C6-alkinyl, C2-C6-alkenyloxy, halogen-C2-C6-alkenyloxy, C1-C6-alkylthio, halogen-C1-C6-alkylthio, C1-C6-alkylsulfonyloxy, halogen-C1-C6-alkylsulfonyloxy, C1-C6-alkylsulfinyl, halogen-C1-C6-alkylsulfinyl, C1-C6-alkylsulfonyl, halogen-C1-C6­alkylsulfonyl, C1-C6-alkenylthio, halogen-C1-C6-alkenylthio, C1-C6-alkenylsulfinyl, halogen-C1­-C6-alkenylsulfinyl, C1-C6-alkenylsulfonyl, halogen-C1-C6-alkenylsulfonyl, C1-C6-alkylamino, di-(C1-C6-alkyl)amino, C1-C6-alkylaminocarbonyl, di-(C1-C6-alkyl)aminocarbonyl, C1-C6-alkylsulfonylamino, halogen-C1-C6-alkylsulfonylamino, C1-C6-alkylcarbonyl, halogen-C1-C6-alkylcarbonyl, C1-C6-alkoxycarbonyl, unsubstituted or one- to five-fold substituted phenyl, unsubstituted or one- to five-fold substituted phenoxy, unsubstituted or one- to five-fold substituted phenylacetylenyl, unsubstituted or one- to four-fold substituted pyridyloxy, unsubstituted or one- to four-fold substituted pyridyl or unsubstituted or one- to seven-fold substituted naphthyl, the substituents in each case being selected from the group consisting of halogen, nitro, cyano, C1-C6-alkyl, halogen-C1-C6-alkyl, C1-C6-alkoxy and halogen-C1-C6-alkoxy, which are useful in the control of endo- and ectoparasites in and on warm-blooded animals, especially productive livestock and domestic animals, as well as on plants.

    AMENOACETONITRILE COMPOUNDS FOR CONTROLLING ENDOPARASITES
    4.
    发明授权
    AMENOACETONITRILE COMPOUNDS FOR CONTROLLING ENDOPARASITES 有权
    用于控制体内寄生虫氨基乙腈CONNECTIONS

    公开(公告)号:EP1401277B1

    公开(公告)日:2007-06-27

    申请号:EP02743200.4

    申请日:2002-06-14

    发明人: DUCRAY, Pierre

    IPC分类号: A01N37/40

    CPC分类号: A01N37/40

    摘要: The invention relates to the use of aminoacetonitrile compounds of formula wherein R1, R2 and m have the significances given in claim 1, in the control of endoparasites, especially helminths, in warm-blooded productive productive livestock and domestic animals.

    CYANOACETYL COMPOUNDS
    8.
    发明公开
    CYANOACETYL COMPOUNDS 审中-公开
    氰基乙CONNECTIONS

    公开(公告)号:EP1436250A1

    公开(公告)日:2004-07-14

    申请号:EP02779457.7

    申请日:2002-10-02

    IPC分类号: C07C255/40

    CPC分类号: A01N37/38 C07C255/20

    摘要: The invention relates to compounds of the general formula (I), wherein Ar1, Ar2, R4, R5, R6, R7, R8, R9, R10, W, X, a, b and c have the significances given in claim 1, and optionally the enantiomers thereof. The active ingredients have advantageous pesticidal properties. They are especially suitable for controlling parasites on warm-blooded animals.

    COMPOSITION FOR REPELLING AND DETERRING VERMIN
    9.
    发明公开
    COMPOSITION FOR REPELLING AND DETERRING VERMIN 有权
    组合物技术远的位置,而且跳蚤和壁虱防御

    公开(公告)号:EP2094079A1

    公开(公告)日:2009-09-02

    申请号:EP07847248.7

    申请日:2007-11-21

    申请人: Novartis AG

    摘要: The invention describes essentially a non-therapeutical process for deterring vermin, which is based on the usage of the largely known beta amino-alcohol derivatives of formula (I), as defined herein before. Furthermore, it describes the corresponding vermin-deterring compositions which contain these substances as the active ingredient, compounds of the formula (I) for the preparation of vermin-deterring compositions, and the use of compounds of formula (I) in the defense against vermin. Thus, the invention describes how and in which form the compounds of the formula (I) or their acid addition salts are used to deter vermin from materials, places or warm-blooded animals.