公开(公告)号：EP2598506A1

公开(公告)日：2013-06-05

申请号：EP11745862.0

申请日：2011-07-29

申请人： OSI Pharmaceuticals, LLC

发明人： CASTELHANO, Arlindo, L. ,  CUTTING, Gary, A. ,  LOCKE, Andrew, J. ,  MAO, Yunyu ,  MULVIHILL, Kristen, Michelle ,  NORRIE, Robert ,  O'BRIEN, Andrew, J. ,  PARK, Stuart, R. ,  RECHKA, Josef, A. ,  STEVENS, Andrew, Michael ,  THOMAS, Christopher, I.

IPC分类号： C07D487/04

CPC分类号： C07D487/04

摘要： Process for preparing the tyrosine kinase inhibitor OSI-906 comprises coupling Compound (2) with Compound (6) under specified conditions.