-
公开(公告)号：EP2495236A1
公开(公告)日：2012-09-05
申请号：EP10826651.1
申请日：2010-10-25
发明人： KAN, Keizo , OHTANI, Tadaaki
IPC分类号： C07D223/16 , A61K31/55 , A61P9/12
CPC分类号： C07D223/16 , A61K31/55 , A61K45/06 , A61K2300/00
摘要： An object of the present invention is to provide a novel benzazepine compound or a salt thereof, which has excellent vasopressin antagonistic activity.
The benzazepine compound or a salt thereof of the present invention is represented by Formula (1):
wherein R 1 , R 2 and R 5 may be the same or different and each represents H or D; and R 3 and R 4 each represents a C 1-6 alkyl group, a C 1-6 deuteroalkyl group, or a C 1-6 perdeuteroalkyl group.摘要翻译： 本发明的目的是提供一种具有优异的加压素拮抗活性的新的苯并氮杂化合物或其盐。 本发明的苯并氮杂化合物或其盐由式（1）表示：其中R 1，R 2和R 5可以相同或不同，各自表示H或D; R 3和R 4各自表示C 1-6烷基，C 1-6氘代烷基或C 1-6芳基烷基。
-
公开(公告)号：EP2228441A1
公开(公告)日：2010-09-15
申请号：EP08867315.7
申请日：2008-12-25
发明人： SHIMADA, Yoshikazu , YASUDA, Setsuko , TAKAHASHI, Masayuki , HAYASHI, Takashi , MIYAZAWA, Norihiro , ABIRU, Yasuhiro , OHTANI, Tadaaki , SATO, Ikutaro
CPC分类号： C12P17/06 , C12N9/00 , C12N9/0073 , C12N9/93
摘要： An object of the present invention is to provide enzymes associated with equol synthesis, genes coding such enzymes, and a process for producing equol and its intermediates using the enzymes and genes.
The present invention provides a dihydrodaidzein synthesizing enzyme, tetrahydrodaidzein synthesizing enzyme, equol synthesizing enzyme, and genes coding these enzymes. The present invention also provides a process for synthesizing dihydrodaidzein, tetrahydrodaidzein, and/or equol using these enzymes.摘要翻译： 本发明的目的是提供与雌马酚合成相关的酶，编码这些酶的基因，以及使用酶和基因产生雌马酚及其中间体的方法。 本发明提供二氢黄豆苷元合成酶，四氢黄豆苷元合成酶，雌马酚合成酶，以及编码这些酶的基因。 本发明还提供了使用这些酶合成二氢黄豆苷元，四氢黄豆苷元和/或雌马酚的方法。
-
公开(公告)号：EP2228441B1
公开(公告)日：2013-06-19
申请号：EP08867315.7
申请日：2008-12-25
发明人： SHIMADA, Yoshikazu , YASUDA, Setsuko , TAKAHASHI, Masayuki , HAYASHI, Takashi , MIYAZAWA, Norihiro , ABIRU, Yasuhiro , OHTANI, Tadaaki , SATO, Ikutaro
CPC分类号： C12P17/06 , C12N9/00 , C12N9/0073 , C12N9/93
-
-
搜索结果
3 条记录 (耗时 0.013 秒)
