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公开(公告)号：EP1874772A1
公开(公告)日：2008-01-09
申请号：EP06740614.0
申请日：2006-04-05
申请人： PHARMACOPEIA, INC.
发明人： OHLMEYER, Michael , BOHNSTEDT, Adolph , KINGSBURY, Celia , HO, Koc-Kan , QUINTERO, Jorge , YOU, Ming , PARK, Haengsoon , LU, Yingchun
IPC分类号： C07D471/04 , C07D487/04 , C07D519/00 , A61K31/52 , A61P37/06
CPC分类号： C07D473/00 , C07D471/04 , C07D473/32 , C07D487/04
摘要： The present invention provides novel purine and imidazopyridine derivatives useful for the prevention and treatment of autoimmune diseases, inflammatory disease, mast cell mediated disease and transplant rejection. The compounds are of the general formulas ( I ) and ( II ).
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2.发明公开PYRAZOLO[1,5-A]PYRIMIDINE COMPOUNDS AS CYCLIN DEPENDENT KINASE INHIBITORS 有权并[1,5-A]嘧啶类作为抑制剂细胞周期蛋白依赖性激酶
公开(公告)号：EP1534712A2
公开(公告)日：2005-06-01
申请号：EP03796321.2
申请日：2003-09-03
发明人： GUZI, Timothy, J. , PARUCH, Kamil , DWYER, Michael, P. , DOLL, Ronald, J. , GIRIJAVALLABHAN, Viyyoor, Moopil , ALVAREZ, Carmen, S. , CHAN, Tin-Yau , KNUTSON, Chad , MADISON, Vincent , FISCHMANN, Thierry, O. , DILLARD, Lawrence, W. , TRAN, Vinh, D. , HE, Zhen Min , JAMES, Ray, Anthony , PARK, Haengsoon
IPC分类号： C07D487/04 , A61K31/519 , A61P25/00 , A61P35/00
CPC分类号： C07D487/04
摘要： In its many embodiments, the present invention provides a novel class of pyrazolo[1,5-a]pyrimidine compounds as inhibitors of cyclin dependent kinases, methods of preparing such compounds, pharmaceutical compositions containing one or more such compounds, methods of preparing pharmaceutical formulations comprising one or more such compounds, and methods of treatment, prevention, inhibition, or amelioration of one or more diseases associated with the CDKs using such compounds or pharmaceutical compositions.
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公开(公告)号：EP1534710A1
公开(公告)日：2005-06-01
申请号：EP03749347.5
申请日：2003-09-03
发明人： GUZI, Timothy, J. , PARUCH, Kamil , DWYER, Michael, P. , DOLL, Ronald, J. , GIRIJAVALLABHAN, Viyyoor, Moopil , DILLARD, Lawrence, W. , TRAN, Vinh, D. , HE, Zhen Min , JAMES, Ray, Anthony , PARK, Haengsoon
IPC分类号： C07D487/04 , A61K31/519 , A61P25/00 , A61P35/00
CPC分类号： C07D487/04 , A61K31/519 , A61K31/52 , A61K31/704 , A61K31/7072 , A61K45/06 , A61K2300/00
摘要： In its many embodiments, the present invention provides a novel class of pyrazolo[1,5-a]pyrimidine compounds as inhibitors of cyclin dependent kinases, methods of preparing such compounds, pharmaceutical compositions containing one or more such compounds, methods of preparing pharmaceutical formulations comprising one or more such compounds, and methods of treatment, prevention, inhibition, or amelioration of one or more diseases associated with the CDKs using such compounds or pharmaceutical compositions.
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公开(公告)号：EP1534710B1
公开(公告)日：2007-10-24
申请号：EP03749347.5
申请日：2003-09-03
发明人： GUZI, Timothy, J. , PARUCH, Kamil , DWYER, Michael, P. , DOLL, Ronald, J. , GIRIJAVALLABHAN, Viyyoor, Moopil , DILLARD, Lawrence, W. , TRAN, Vinh, D. , HE, Zhen Min , JAMES, Ray, Anthony , PARK, Haengsoon
IPC分类号： C07D487/04 , A61K31/519 , A61P25/00 , A61P35/00
CPC分类号： C07D487/04 , A61K31/519 , A61K31/52 , A61K31/704 , A61K31/7072 , A61K45/06 , A61K2300/00
摘要： In its many embodiments, the present invention provides a novel class of pyrazolo[1,5-a]pyrimidine compounds as inhibitors of cyclin dependent kinases, methods of preparing such compounds, pharmaceutical compositions containing one or more such compounds, methods of preparing pharmaceutical formulations comprising one or more such compounds, and methods of treatment, prevention, inhibition, or amelioration of one or more diseases associated with the CDKs using such compounds or pharmaceutical compositions.
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