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公开(公告)号:EP1112998A1
公开(公告)日:2001-07-04
申请号:EP98936729.7
申请日:1998-08-11
发明人: YUASA, Masayuki Pola Chemical Industries, Inc. , KAWAZU, Yukio Pola Chemical Industries, Inc. , SUZUKI, Toshimitsu Pola Chemical Ind., Inc. , MAJIMA, Toshiro Pola Chemical Industries, Inc. , ITOH, Takao Pola Chemical Industries, Inc. , NAKASHIMA, Takuji Pola Chemical Industries, Inc. , NOZAWA, Akira Pola Chemical Industries, Inc. , TAKIMOTO, Hiroyuki Pola Chemical Industries, Inc. , YOKOYAMA, Kouji Pola Chemical Industries, Inc.
IPC分类号: C07C211/27 , C07C211/29 , C07C211/35 , C07C215/28 , C07C225/16 , A61K31/135
CPC分类号: C07C215/28 , C07C17/14 , C07C17/16 , C07C45/004 , C07C45/565 , C07C45/63 , C07C211/21 , C07C211/27 , C07C211/28 , C07C211/29 , C07C211/35 , C07C215/30 , C07C223/02 , C07C225/16 , C07C225/26 , C07C2601/02 , C07C25/02 , C07C49/76 , C07C47/546 , C07C49/80
摘要: The present invention relates to amine derivatives represented by formula (1) or salts thereof.
(wherein R 1 is C1-C4 alkyl; R 2 is
or
R 3 represents C1-C3 alkyl, hydroxylated C1-C5 alkyl, C1-C5 acyl; C2-C5 alkenyl, or a halogen atom; and k, l, and m are each an integer of 1 to 4.)
Exhibiting excellent antifungal effect, these compounds are highly useful as antifungal agents, antifungal compositions, drugs, etc.-
公开(公告)号:EP1112998B1
公开(公告)日:2004-12-08
申请号:EP98936729.7
申请日:1998-08-11
发明人: YUASA, Masayuki Pola Chemical Industries, Inc. , KAWAZU, Yukio Pola Chemical Industries, Inc. , SUZUKI, Toshimitsu Pola Chemical Ind., Inc. , MAJIMA, Toshiro Pola Chemical Industries, Inc. , ITOH, Takao Pola Chemical Industries, Inc. , NAKASHIMA, Takuji Pola Chemical Industries, Inc. , NOZAWA, Akira Pola Chemical Industries, Inc. , TAKIMOTO, Hiroyuki Pola Chemical Industries, Inc. , YOKOYAMA, Kouji Pola Chemical Industries, Inc.
IPC分类号: C07C211/27 , C07C211/29 , C07C211/35 , C07C215/28 , C07C225/16 , A61K31/135
CPC分类号: C07C215/28 , C07C17/14 , C07C17/16 , C07C45/004 , C07C45/565 , C07C45/63 , C07C211/21 , C07C211/27 , C07C211/28 , C07C211/29 , C07C211/35 , C07C215/30 , C07C223/02 , C07C225/16 , C07C225/26 , C07C2601/02 , C07C25/02 , C07C49/76 , C07C47/546 , C07C49/80
摘要: Amine derivatives represented by general formula (1) or their salts, wherein R1 represents C¿1-4? alkyl; R?2¿ represents (i), or (ii), (iii); R3 represents C¿1-3? alkyl, hydroxylated C1-5 alkyl, C1-5 acyl, C2-5 alkenyl or halogeno; and k, l and m are each an integer of 1 to 4. Because of being excellent in antifungal effect, these compounds are highly useful as antifungal agents, antifungal compositions, drugs, etc.
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