Thiapentanamide derivatives
    1.
    发明公开
    Thiapentanamide derivatives 失效
    硫代戊酰胺衍生物

    公开(公告)号:EP0298543A2

    公开(公告)日:1989-01-11

    申请号:EP88201304.8

    申请日:1988-06-23

    IPC分类号: C07C323/00 C07D333/38

    CPC分类号: C07D333/38

    摘要: A compound of the general formula
    in which X represents a chlorine or bromine atom, R¹ represents a hydrogen atom, a C(1-6) alkyl group, a benzyl group or a phenyl group optionally substituted by a C(1-6) alkyl group, and R² represents the group CN or the group COOR³ in which R³ represents a C(1-6) alkyl group, a process for the preparation of a compound of formula (I), and the use of a compound of formula (I) in the preparation of a compound of the general formula.
    in which R¹ is as defined above and R⁴ represents an amino group or a hydroxyl group.

    摘要翻译: 其中X代表氯或溴原子,R 1代表氢原子,C(1-6)烷基,苄基或任选被C(1-6)烷基取代的苯基的通式 并且R 2表示基团CN或其中R 3表示C(1-6)烷基的基团COOR 3,制备式(I)化合物的方法以及式(I)化合物的用途, )在制备通式化合物中的用途。 其中R 1如上定义,R 4代表氨基或羟基。

    Process for preparing thiophene derivatives
    3.
    发明公开
    Process for preparing thiophene derivatives 失效
    Verfahren zur Herstellung von Thiophenderivaten。

    公开(公告)号:EP0298542A1

    公开(公告)日:1989-01-11

    申请号:EP88201303.0

    申请日:1988-06-23

    IPC分类号: C07D333/36 C07D333/38

    CPC分类号: C07D333/38 C07D333/36

    摘要: A process for the preparation of 3-amino­thiophenes or acid-addition salts thereof, which comprises reacting the corresponding 3-oxotetra­hydrothiophenes with an acid-addition salt of hydroxylamine in the presence of a polar inert solvent and in the absence of a base at a temperature in the range of from 0 to 200°C.

    摘要翻译: 一种制备3-氨基噻吩或其酸加成盐的方法,该方法包括在极性惰性溶剂存在下,在不存在碱的情况下,使相应的3-氧代四氢噻吩与羟胺的酸加成盐反应, 在0至200℃的范围内。

    Thiapentanamide derivatives
    4.
    发明公开
    Thiapentanamide derivatives 失效
    三苯甲酰胺衍生物

    公开(公告)号:EP0298543A3

    公开(公告)日:1991-02-13

    申请号:EP88201304.8

    申请日:1988-06-23

    IPC分类号: C07C323/00 C07D333/38

    CPC分类号: C07D333/38

    摘要: A compound of the general formula
    in which X represents a chlorine or bromine atom, R¹ represents a hydrogen atom, a C(1-6) alkyl group, a benzyl group or a phenyl group optionally substituted by a C(1-6) alkyl group, and R² represents the group CN or the group COOR³ in which R³ represents a C(1-6) alkyl group, a process for the preparation of a compound of formula (I), and the use of a compound of formula (I) in the preparation of a compound of the general formula.
    in which R¹ is as defined above and R⁴ represents an amino group or a hydroxyl group.