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    SUBSTANCE FA-70D, PROCESS FOR PRODUCING THE SAME, AND USES THEREOF
    2.
    发明公开
    SUBSTANCE FA-70D, PROCESS FOR PRODUCING THE SAME, AND USES THEREOF 失效
    SUBSTANZ FA-70D，HERSTELLUNGSVERFAHREN UND VERWENDUNGEN

    公开(公告)号：EP0822260A1

    公开(公告)日：1998-02-04

    申请号：EP97904590.3

    申请日：1997-02-20

    申请人： TAIHO PHARMACEUTICAL CO., LTD.

    发明人： KITANO, Shizuo ,  SASAKI, Toru ,  YOSHIDA, Kenichiro ,  OTANI, Toshio ,  YU, Lei ,  WU, Yun ,  KATSUNUMA, Nobuhiko

    IPC分类号： C12P21/02 ,  C07K5/068 ,  A61K38/05

    CPC分类号： C07K5/06095 ,  A61K38/00 ,  C12P21/02

    摘要： Substance FA-70D which has the following formula (1) or its salt, a method for its production, a pharmaceutical composition comprising the compound as an active ingredient, a method of treating osteoporosis which comprises administering the compound, use of the compound as a drug, and a microorganism capable of producing Substance FA-70D.

    This compound has specific inhibitory activity against cathepsin series proteases and is of value as a therapeutic drug for various diseases with which these enzymes are associated, particularly osteoporosis.

    摘要翻译： 具有下式（1）的物质FA-70D或其盐，其制备方法，包含该化合物作为活性成分的药物组合物，治疗骨质疏松症的方法，其包括施用该化合物，使用该化合物作为 药物和能够产生物质FA-70D的微生物。 该化合物对组织蛋白酶系列蛋白酶具有特异性抑制活性，作为与这些酶相关的各种疾病，特别是骨质疏松症的治疗药物是有价值的。