-
1.发明公开SUNITINIB HEMI-L-MALATE, POLYMORPHS AND PREPARATION THEREOF, POLYMORPHS OF RACEMIC SUNITINIB MALATE, COMPOSITINS CONTAINING SUNITINIB BASE AND MALIC ACID AND PREPARATION THEREOF 审中-公开舒尼替尼半L-苍鹭，多晶型物及其生产多晶型外消旋舒尼替尼苍鹭，舒尼替尼碱和苹果酸组合物及其制备
公开(公告)号：EP2220071A2
公开(公告)日：2010-08-25
申请号：EP08851719.8
申请日：2008-11-21
发明人： JEGOROV, Alexandr , VRASPIR, Pavel , ARONHIME, Judith , GAVENDA, Ales , ANGIOLETTI, Paolo , MACDONALD,Peter, Lindsay , SCARPITTA, Francesca , VILLA, Marco , BIGATTI, Ettore , CANAVESI, Augusto
IPC分类号： C07D403/06 , A61K31/404 , A61P35/00
CPC分类号： C07D403/06
摘要： The invention provides Sunitinib hemi-L-malate, polymorphs thereof, polymorphs of racemic sunitinib malate, compositions containing sunitinib base and either L or racemic malic acid, processes for the preparation thereof, and pharmaceutical compositions thereof.
-
2.发明公开PROCESS FOR THE PREPARATION OF SUNITINIB MALATE VIA SUNITINIB ACETATE AND THEIR POLYMORPHS 审中-公开用于生产舒尼替尼关于SUNITINIBACETAT和其多晶型
公开(公告)号：EP2373642A2
公开(公告)日：2011-10-12
申请号：EP09790764.6
申请日：2009-07-23
IPC分类号： C07D403/06
CPC分类号： C07D403/06 , C07D209/12
摘要： Polymorphs of sunitinib acetate and sunitinib base and sunitinib malate form 1 have been prepared and described.
-
公开(公告)号：EP2207777A2
公开(公告)日：2010-07-21
申请号：EP08843260.4
申请日：2008-10-23
发明人： SIMO, ondrej , FILIPCIK, Jiri , MARTAUS, Alexandr , JEGOROV, Alexandr , GAVENDA, Ales , ARONHIME, Judith , VRASPIR, Pavel , KOLTAI, Tamas , FAUSTMANN, Jiri , GABRIEL, Roman
IPC分类号： C07D417/12 , A61K31/506 , A61P35/00
CPC分类号： C07D417/12
摘要： Provided is dasatinib, solvates thereof and their crystalline forms, methods for their preparation, and pharmaceutical compositions thereof. Formula (I).
-
公开(公告)号：EP2220072A2
公开(公告)日：2010-08-25
申请号：EP08852503.5
申请日：2008-11-21
发明人： GAVENDA, Ales , BIGATTI, Ettore , JEGOROV, Alexandr , CANAVESI, Augusto , VRASPIR, Pavel , ARONHIME, Judith , MACDONALD, Peter, Lindsay , SCARPITTA, Francesca , VILLA, Marco , ANGIOLETTI, Paolo
IPC分类号： C07D403/06 , A61K31/404 , A61P35/00
CPC分类号： C07D403/06
摘要： The present invention provides polymorphs of Sunitinib base and processes for preparation thereof.
-
-
-
搜索结果
4 条记录 (耗时 0.011 秒)
