SYSTEM FOR CONTROLLING THE REACTIVITY OF BORONIC ACIDS
    2.
    发明公开
    SYSTEM FOR CONTROLLING THE REACTIVITY OF BORONIC ACIDS 有权
    系统ZUR STEUERUNG DERREAKTIVITÄTVONBORONSÄURE

    公开(公告)号:EP2181103A1

    公开(公告)日:2010-05-05

    申请号:EP07844994.9

    申请日:2007-11-08

    IPC分类号: C07D307/80 C07F5/02

    摘要: A protected organoboronic acid includes a boron having an sp3 hybridization, a conformationally rigid protecting group bonded to the boron, and an organic group bonded to the boron through a boron-carbon bond. A method of performing a chemical reaction includes contacting a protected organoboronic acid with a reagent, the protected organoboronic acid including a boron having an sp3 hybridization, a conformationally rigid protecting group bonded to the boron, and an organic group bonded to the boron through a boron-carbon bond. The organic group is chemically transformed, and the boron is not chemically transformed.

    摘要翻译: 受保护的有机硼酸包括具有sp 3杂交的硼,与硼结合的构象刚性保护基,以及通过硼 - 碳键与硼结合的有机基团。 进行化学反应的方法包括使受保护的有机硼酸与试剂接触,受保护的有机硼酸包括具有sp3杂交的硼,与硼结合的构象刚性保护基,和通过硼键合到硼上的有机基团 碳键。 有机基团被化学转化,硼不进行化学转化。