公开(公告)号：EP2872519A1

公开(公告)日：2015-05-20

申请号：EP13732493.5

申请日：2013-06-27

申请人： UNIVERSITE DE BORDEAUX ,  Centre National de la Recherche Scientifique

发明人： PUCHEAULT, Mathieu Jonathan Damien ,  MARCIASINI, Ludovic Daniel Alain ,  VAULTIER, Michel

IPC分类号： C07F5/02

CPC分类号： C07F5/04 ,  C07F5/02 ,  C07F5/027

摘要： The present invention relates to a new process for the preparation of an arylborane compound, by arylation of a B-H bond, which comprises a step (1) of contacting an arenediazonium salt or a heteroarenediazonium salt with an organoboron compound containing at least one B-H bond, in a reaction medium containing a solvent, in the absence of base, in the absence or in the presence of an activating agent, for the preparation of an arylborane compound, and a possible step (2) of recovery and purification of said arylborane compound obtained at the step (1), said arylborane being in particular an aminoarylborane, and a possible step (3) of refunctionalisation of said arylborane obtained at step (1) or (2) for the preparation of aryl boronic derivatives or arylborates.