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    Pyridyl cyclopropane derivatives with fungicidal activity
    3.
    发明公开
    Pyridyl cyclopropane derivatives with fungicidal activity 失效
    Fungizide。

    公开(公告)号：EP0436348A2

    公开(公告)日：1991-07-10

    申请号：EP90313836.0

    申请日：1990-12-18

    申请人： ZENECA LIMITED ,  ICI AMERICAS INC.

    发明人： Worthington, Paul Antohony ,  Matthews, Ian Richard ,  Bartholomew, David ,  Crowley, Patrick Jelf ,  Baker, Don Robert ,  Fisher, Karl Joseph

    IPC分类号： C07D213/75 ,  C07D213/74 ,  A01N53/00 ,  C07C61/04 ,  C07C51/245

    CPC分类号： C07D213/75 ,  A01N53/00 ,  C07C51/29 ,  C07C61/15

    摘要： Compounds of having the general formula (I):

    and stereoisomers thereof, wherein R¹ is hydrogen, halogen, C₁₋₄ alkoxy, C₁₋₄ alkyl, C₂₋₄ alkenyl, C₂₋₄ alkynyl, C₁₋₄ haloalkyl, C₁₋₄ haloalkoxy, COR or cyano; R², R³ and R⁴ are independently hydrogen, halogen or methyl, provided that R², R³ and R⁴ are not all hydrogen and provided that when one of them is methyl then at least one of the other two is not hydrogen;

    wherein R⁵ is hydrogen, C₁₋₄ alkyl (optionally substituted by hydrogen or cyano), optionally substituted benzyl, C₂₋₄ alkenyl, C₂₋₄ alkynyl, cyano, COR C₁₋₄ thioalkoxy C₁₋₄ thiohaloalkoxy or SNR⁷R⁸; R⁷ and R⁸ are independently C₁₋₄ alkyl or CO₂R; Y is oxygen or sulphur; R⁶ is C₁₋₄ alkoxy, C₁₋₄ thioalkoxy or -NR⁹ R¹⁰ ; and R⁹ and R¹⁰ are independently hydrogen, C₁₋₄ alkyl, aryl or aralkyl or R⁹ and R¹⁰ join to form an optionally substituted heterocyclic ring and R is C₁₋₄ alkyl or C₃₋₇ cycloalkyl. These compounds are fungicidally active.

    摘要翻译： 具有通式（I）：的化合物及其立体异构体，其中R 1是氢，卤素，C 1-4烷氧基，C 1-4烷基，C 2-4烯基，C 2-4炔基，C 1-4 卤代烷基，C 1-4卤代烷氧基，COR或氰基; R 2，R 3和R 4独立地为氢，卤素或甲基，条件是R 2，R 3和R 4不全部为氢，条件是当其中一个为 甲基，则其他两个中的至少一个不是氢; 其中R 5为氢，C 1-4烷基（任选被氢或氰基取代），任选取代的苄基，C 2-4烯基，C 2-4炔基，氰基，COR C 1-4硫烷氧基C 1-4硫代卤代烷氧基或 SNR <7> - [R <8>; R 7和R 8独立地是C 1-4烷基或CO 2 R; Y是氧或硫; R 6是C 1-4烷氧基，C 1-4硫代烷氧基或-NR 9 R 1; 并且R 9和R 1独立地是氢，C 1-4烷基，芳基或芳烷基或R 9和R 1连接形成任选被取代的杂环，R是C1 -4-烷基或C 3-7环烷基。 这些化合物是杀真菌活性的。

    Fungicides
    4.
    发明公开
    Fungicides 失效
    杀菌剂

    公开(公告)号：EP0769495A1

    公开(公告)日：1997-04-23

    申请号：EP96307315.0

    申请日：1996-10-08

    申请人： ZENECA LIMITED

    发明人： Matthews, Ian Richard ,  De Fraine, Paul John ,  Crowley, Patrick Jelf ,  Williams, John

    IPC分类号： C07D265/36 ,  C07D265/32 ,  C07D211/86 ,  C07D211/74 ,  C07D215/22 ,  C07D267/14 ,  C07D279/16 ,  A01N43/84

    CPC分类号： C07D215/227 ,  A01N43/36 ,  A01N43/42 ,  A01N43/72 ,  A01N43/76 ,  A01N43/84 ,  C07D211/74 ,  C07D211/86 ,  C07D265/32 ,  C07D265/36 ,  C07D267/14 ,  C07D279/16

    摘要： Compounds, useful as plant fungicides, having the formula (I):
    or a stereoisomer thereof, wherein A is CH or N, B is OCH 3 or NHCH 3 , X is CH 2 , CH 2 O, O or S, Y is R 1 -C=C-R 2 or R 1 -CH-CH-R 2 wherein R 1 and R 2 are independently H, halo, hydroxy, alkyl, haloalkyl, alkoxy, haloalkoxy, cyano, nitro, amino, mono- or dialkylamino, alkanoylamino, carboxy, alkoxycarbonyl, aminocarbonyl, mono- or di-alkylaminocarbonyl, alkylcarbonyloxy, optionally substituted aryl, optionally substituted aralkyl or optionally substituted aryloxy or R 1 and R 2 join to form with the carbon atoms to which they are attached an optionally substituted benzene ring, and Z is CH 2 , CHCH 3 , C(CH 3 ) 2 or C=O.

    摘要翻译： 其中A为CH或N，B为OCH3或NHCH3，X为CH2，CH2O，O或S，Y为R1-C = C- 其中R 1和R 2独立地为H，卤素，羟基，烷基，卤代烷基，烷氧基，卤代烷氧基，氰基，硝基，氨基，单或二烷基氨基，烷酰基氨基，羧基，烷氧羰基，氨基羰基， 或二烷基氨基羰基，烷基羰基氧基，任选取代的芳基，任选取代的芳烷基或任选取代的芳氧基，或者R 1和R 2与它们所连接的碳原子一起形成任选取代的苯环，Z为CH 2，CHCH 3，C ）2或C = O。

    Pyridyl cyclopropane derivatives with fungicidal activity
    5.
    发明公开
    Pyridyl cyclopropane derivatives with fungicidal activity 失效
    具有杀真菌活性的吡啶基环丙烷衍生物

    公开(公告)号：EP0436348A3

    公开(公告)日：1991-12-11

    申请号：EP90313836.0

    申请日：1990-12-18

    申请人： ZENECA LIMITED ,  ICI AMERICAS INC.

    发明人： Worthington, Paul Antohony ,  Matthews, Ian Richard ,  Bartholomew, David ,  Crowley, Patrick Jelf ,  Baker, Don Robert ,  Fisher, Karl Joseph

    IPC分类号： C07D213/75 ,  C07D213/74 ,  A01N53/00 ,  C07C61/04 ,  C07C51/245

    CPC分类号： C07D213/75 ,  A01N53/00 ,  C07C51/29 ,  C07C61/15

    摘要： Compounds of having the general formula (I):

    and stereoisomers thereof, wherein R¹ is hydrogen, halogen, C₁₋₄ alkoxy, C₁₋₄ alkyl, C₂₋₄ alkenyl, C₂₋₄ alkynyl, C₁₋₄ haloalkyl, C₁₋₄ haloalkoxy, COR or cyano; R², R³ and R⁴ are independently hydrogen, halogen or methyl, provided that R², R³ and R⁴ are not all hydrogen and provided that when one of them is methyl then at least one of the other two is not hydrogen;

    wherein R⁵ is hydrogen, C₁₋₄ alkyl (optionally substituted by hydrogen or cyano), optionally substituted benzyl, C₂₋₄ alkenyl, C₂₋₄ alkynyl, cyano, COR C₁₋₄ thioalkoxy C₁₋₄ thiohaloalkoxy or SNR⁷R⁸; R⁷ and R⁸ are independently C₁₋₄ alkyl or CO₂R; Y is oxygen or sulphur; R⁶ is C₁₋₄ alkoxy, C₁₋₄ thioalkoxy or -NR⁹ R¹⁰ ; and R⁹ and R¹⁰ are independently hydrogen, C₁₋₄ alkyl, aryl or aralkyl or R⁹ and R¹⁰ join to form an optionally substituted heterocyclic ring and R is C₁₋₄ alkyl or C₃₋₇ cycloalkyl. These compounds are fungicidally active.

    摘要翻译： 具有通式（Ⅰ）的化合物及其立体异构体，其中R 1是氢，卤素，C 1-4烷氧基，C 1-4烷基，C 2-4链烯基，C 2-4炔基，C 1-4卤代烷基，C 1-4卤代烷氧基 ，COR或氰基; R 2，R 3和R 4独立地为氢，卤素或甲基，条件是R 2，R 3和R 4不全是氢，并且条件是当它们中的一个是甲基时，则另外两个中的至少一个不是氢; 其中R 5是氢，C 1-4烷基（任选被氢或氰基取代），任选取代的苄基，C 2-4链烯基，C 2-4炔基，氰基，COR C 1-4硫代烷氧基C 1-4硫代卤代烷氧基或SNR 6 R 7; R 8和R 9独立地为C 1-4烷基或CO 2 R; Y是氧或硫; R 6是C 1-4烷氧基，C 1-4硫代烷氧基或-NR 9 R 10; R 9和R 10独立地是氢，C 1-4烷基，芳基或芳烷基，或者R 8和R 10连接形成任意取代的杂环，R是C 1-4烷基或C 3-8环烷基。 这些化合物具有杀真菌活性。

    Fungicides
    7.
    发明公开
    Fungicides 失效
    Fungizide

    公开(公告)号：EP0858997A1

    公开(公告)日：1998-08-19

    申请号：EP98105183.2

    申请日：1996-10-08

    申请人： ZENECA LIMITED

    发明人： Matthews, Ian Richard ,  De Fraine,Paul John ,  Crowley, Patrick Jelf ,  Williams, John

    IPC分类号： C07D211/86 ,  C07D211/90 ,  C07D265/32 ,  A01N43/84 ,  A01N43/40

    CPC分类号： C07D215/227 ,  A01N43/36 ,  A01N43/42 ,  A01N43/72 ,  A01N43/76 ,  A01N43/84 ,  C07D211/74 ,  C07D211/86 ,  C07D265/32 ,  C07D265/36 ,  C07D267/14 ,  C07D279/16

    摘要： Compounds, useful as plant fungicides, having the formula (I):
    or a stereoisomer thereof, wherein A is CH or N, B is OCH 3 or NHCH 3 , X is CH 2 , CH 2 O, O or S, Y is R 1 -C=C-R 2 or R 1 -CH-CH-R 2 wherein R 1 and R 2 are independently H, halo, hydroxy, alkyl, haloalkyl, alkoxy, haloalkoxy, cyano, nitro, amino, mono- or dialkylamino, alkanoylamino, carboxy, alkoxycarbonyl, aminocarbonyl, mono- or dialkylaminocarbonyl, alkylcarbonyloxy, optionally substituted aryl, optionally substituted aralkyl or optionally substituted aryloxy and Z is CH 2 , CHCH 3 , C(CH 3 ) 2 or C=O.

    摘要翻译： 可用作植物杀真菌剂的化合物，其具有式（I）：其中A为CH或N，B为OCH 3或NHCH 3，X为CH 2，CH 2 O，O或S，Y为R 1 -C = CR 2或R 1 -CH-CH-R 2其中R 1和R 2独立地是H，卤素，羟基，烷基，卤代烷基，烷氧基，卤代烷氧基，氰基， 硝基，氨基，一烷基氨基或二烷基氨基，烷酰基氨基，羧基，烷氧基羰基，氨基羰基，单 - 或二烷基氨基羰基，烷基羰氧基，任选取代的芳基，任选取代的芳烷基或任选取代的芳氧基，Z是CH 2，CHCH 3，C（CH 3） O.

    Process for the preparation of intermediates for oxime ether- or 2-phenyl-3-methyl propenoate-fungicides
    8.
    发明公开
    Process for the preparation of intermediates for oxime ether- or 2-phenyl-3-methyl propenoate-fungicides 失效
    一种制备中间体化合物的肟醚或2-苯基-3-甲氧基 - propenester杀真菌剂处理

    公开(公告)号：EP0711751A1

    公开(公告)日：1996-05-15

    申请号：EP96102169.8

    申请日：1992-09-09

    申请人： ZENECA LIMITED

    发明人： Matthews, Ian Richard ,  Clouch, John Martin ,  Godfrey, Christopher Richard Ayles

    IPC分类号： C07C249/12 ,  C07C251/48 ,  C07D311/76 ,  C07D307/83 ,  C07C69/96

    CPC分类号： C07D213/75 ,  A01N47/06 ,  A01N47/12 ,  A01N47/16 ,  A01N47/18 ,  A01N47/20 ,  A01N47/22 ,  C07C69/734 ,  C07C69/96 ,  C07C249/04 ,  C07C249/12 ,  C07C251/48 ,  C07C271/28 ,  C07C271/64 ,  C07C317/42 ,  C07C323/36 ,  C07C327/48 ,  C07C329/02 ,  C07C329/04 ,  C07C333/08 ,  C07D295/205 ,  C07D311/76

    摘要： Fungicidal compounds having the formula (I):

    wherein W is CH₃O.CH=CCO₂CH₃, CH₃ON=CCONR³R⁴ or CH₃ON=CCO₂CH₃ and stereoisomers thereof; n is O or 1; X is oxygen or sulphur; Z is oxygen, sulphur or NR¹; R¹ is hydrogen or alkyl optionally substituted with halogen, C₁₋₆ alkoxy, C₂₋₆ alkenyl, C₂₋₆ alkynyl, C₃₋₆ cycloalkyl or aryl; R² is alkyl, haloalkyl, alkenyl, alkynyl, alkoxycarbonyl(C₁₋₄)alkyl, optionally substituted aryl, optionally substituted heteroaryl, optionally substituted aryl(C₁₋₄)alkyl, optionally substituted heteroaryl(C₁₋₄)alkyl, optionally substituted aryloxy(C₁₋₄)alkyl, optionally substituted heteroaryloxy(C₁₋₄)alkyl, optionally substituted aryloxy(C₂₋₄)alkenyl, optionally substituted heteroaryloxy(C₂₋₄)alkenyl, optionally substituted aryl(C₂₋₄)alkenyl, optionally substituted heteroaryl(C₂₋₄)alkenyl, optionally substituted arylcarbonyl(C₁₋₄)alkyl, optionally substituted heteroarylcarbonyl(C₁₋₄)alkyl, optionally substituted aryloxycarbonyl(C₁₋₄)alkyl, optionally substituted heteroaryloxycarbonyl-(C₁₋₄)alkyl or -COR⁵; or R¹ and R² together form an optionally substituted 4-, 5- or 6-membered heterocyclic ring system; R³ and R⁴ are independently hydrogen or methyl; and R⁵ is optionally substituted heteroaryl or optionally substituted aryl; and processes for preparing, compositions comprising and methods of combating fungi using compounds of formula (I). Also provided is a process for the preparation of a compound of formula (XX):

    wherein p is 0 or 1.

    摘要翻译： 具有式（I）的杀真菌化合物： worin W是CH3O.CH = CCO2CH3，CH3ON = CCONR <3> [R <4>或= CH3ON CCO2CH3和立体异构体; n是0或1; X是氧或硫; Z是氧，硫或NR <1>; [R <1>是氢或烷基被卤素OPTIONALLY substituiertem，C 1-6烷氧基，C 2-6烯基，C 2-6炔基，C 3-6环烷基或芳基; [R <2>的烷基，卤代烷基，烯基，炔基，烷氧基羰基（C 1-4）烷基，芳基OPTIONALLY substituiertem，任选substituiertem杂芳基，任选substituiertem芳基（C 1-4）烷基，任选substituiertem杂芳基（C 1-4）烷基，任选 取代的芳氧基（C 1-4）烷基，任选取代的杂芳氧基（C 1-4）烷基，任选取代的芳氧基（C 2-4）烯基，任选取代的杂芳氧基（C 2-4）烯基，任选取代的芳基（C 2-4）烯基，任选 取代的杂芳基（C 2-4）烯基，任选substituiertem芳基羰基（C 1-4）烷基，任选substituiertem杂芳（C 1-4）烷基，任选substituiertem芳氧基羰基（C 1-4）烷基，任选substituiertem杂芳氧，（C 1-4）烷基或 COR <5>; 或R <1>和R <2>一起形成在OPTIONALLY substituiertem 4-，5-或6元杂环环系; [R <3>和R <4>是unabhängig氢或甲基; 且R <5>任选substituiertem杂芳基或任选substituiertem芳基; 和制备打击使用式（I）的化合物真菌的，组合物和方法，其包括处理。 所以提供了一种用于制备式（XX）的化合物的制备： worin p是0或第一