-
公开(公告)号:US08895497B2
公开(公告)日:2014-11-25
申请号:US12960805
申请日:2010-12-06
申请人: Chun-Cheng Lin , Wun-Shaing Wayne Chang , Biing-Jiun Uang , Jang-Yang Chang , Jo-Chun Chen , Hsing-Pang Hsieh
发明人: Chun-Cheng Lin , Wun-Shaing Wayne Chang , Biing-Jiun Uang , Jang-Yang Chang , Jo-Chun Chen , Hsing-Pang Hsieh
IPC分类号: C07D295/215 , C07D307/68
CPC分类号: C07C261/04 , C07C237/22 , C07C2601/02 , C07C2601/04 , C07C2601/14 , C07C2601/18 , C07C2603/18 , C07D209/42 , C07D217/26 , C07D241/24 , C07D249/18 , C07D295/215 , C07D307/68 , C07D309/32 , C07D319/18 , C07D333/24
摘要: Cathepsin S inhibitors having formula (I), (II), (III) or (IV) as shown in the specification. These inhibitors can be used to treat cancer and autoimmune/inflammatory diseases.
摘要翻译: 具有式(I),(II),(III)或(IV)的组织蛋白酶S抑制剂,如说明书所示。 这些抑制剂可用于治疗癌症和自身免疫/炎性疾病。
-
公开(公告)号:US20110166141A1
公开(公告)日:2011-07-07
申请号:US12960805
申请日:2010-12-06
申请人: Chun-Cheng Lin , Wun-Shaing Wayne Chang , Biing-Jiun Uang , Jang-Yang Chang , Jo-Chun Chen , Hsing-Pang Hsieh
发明人: Chun-Cheng Lin , Wun-Shaing Wayne Chang , Biing-Jiun Uang , Jang-Yang Chang , Jo-Chun Chen , Hsing-Pang Hsieh
IPC分类号: A61K31/5375 , C07C69/66 , A61K31/235 , C07D241/10 , A61K31/4965 , C07D295/18 , A61P35/00
CPC分类号: C07C261/04 , C07C237/22 , C07C2601/02 , C07C2601/04 , C07C2601/14 , C07C2601/18 , C07C2603/18 , C07D209/42 , C07D217/26 , C07D241/24 , C07D249/18 , C07D295/215 , C07D307/68 , C07D309/32 , C07D319/18 , C07D333/24
摘要: Cathepsin S inhibitors having formula (I), (II), (III) or (IV) as shown in the specification. These inhibitors can be used to treat cancer and autoimmune/inflammatory diseases.
摘要翻译: 具有式(I),(II),(III)或(IV)的组织蛋白酶S抑制剂,如说明书所示。 这些抑制剂可用于治疗癌症和自身免疫/炎性疾病。
-