公开(公告)号：US3914427A

公开(公告)日：1975-10-21

申请号：US43888774

申请日：1974-02-01

Applicant: BAYER AG

Inventor： KRAMER WOLFGANG ,  BUCHEL KARL HEINZ ,  MEISER WERNER ,  FROHBERGER PAUL-ERNST ,  SCHEINPFLUG HANS

IPC: A01N43/50 ,  A01P3/00 ,  C07C45/63 ,  C07C45/75 ,  C07D233/60 ,  C07D521/00 ,  A01N9/22

CPC classification number: C07D231/12 ,  C07C45/63 ,  C07C45/75 ,  C07D233/56 ,  C07D249/08 ,  C07C49/255

Abstract: Compositions containing and methods of using 1-ethylimidazoles of the formula

in which R1 and R3 each individually is hydrogen, alkyl, alkenyl, cycloalkyl, cycloalkenyl, optionally substituted aryl or optionally substituted aralkyl, R2 is alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, optionally substituted aryl or optionally substituted aralkyl, Y is oxygen or sulfur, and X is a keto group or a functional derivative of a keto group, AS SUCH OR IN THE FORM OF SALTS, FOR COMBATING FUNGI.

Abstract translation: 含有式（I）的1-乙基咪唑的组合物和其中R 1和R 3各自独立地为氢，烷基，烯基，环烷基，环烯基，任选取代的芳基或任选地 取代的芳烷基，R 2是烷基，烯基，炔基，环烷基，环烯基，任选取代的芳基或任选取代的芳烷基，Y是氧或硫，X是酮基或酮基的官能衍生物， 用于组合真菌。

公开(公告)号：US3890442A

公开(公告)日：1975-06-17

申请号：US39620273

申请日：1973-09-11

Applicant: BAYER AG

Inventor： MEISER WERNER ,  KRAMER WOLFGANG ,  BUCHEL KARL HEINZ ,  PLEMPEL MANFRED

IPC: C07C45/00 ,  C07C45/63 ,  C07C45/70 ,  C07C45/71 ,  C07C49/213 ,  C07C49/255 ,  C07D249/08 ,  C07D521/00 ,  A61K27/00

CPC classification number: C07D231/12 ,  C07C45/004 ,  C07C45/63 ,  C07C45/70 ,  C07C45/71 ,  C07C49/213 ,  C07C49/255 ,  C07D233/56 ,  C07D249/08 ,  C07C49/233 ,  C07C49/84

Abstract: Antimycotic compositions are produced which comprise an antimycotically effective amount of a 1,2,4-triazole of the formula:

OR A PHARMACEUTICALLY ACCEPTABLE NON-TOXIC SALT THEREOF WHEREIN X 1 is hydrogen or alkyl; X2 is hydrogen or alkyl; R1 is alkyl, unsubstituted or substituted aryl or unsubstituted or substituted aralkyl; R2 is hydrogen, alkyl or unsubstituted or substituted aryl; R3 is alkyl, cycloalkyl, unsubstituted or substituted aryl or unsubstituted or substituted aralkyl; and Y is a keto group or a functional derivative of a keto group, in combination with a pharmaceutically acceptable non-toxic, inert diluent or carrier.

Abstract translation: 产生抗真菌组合物，其包含抗真菌有效量的下式的1,2,4-三唑：

公开(公告)号：US3912752A

公开(公告)日：1975-10-14

申请号：US31896372

申请日：1972-12-27

Applicant: BAYER AG

Inventor： MEISER WERNER ,  BUCHEL KARL HEINZ ,  KRAMER WOLFGANG ,  GREWE FERDINAND

IPC: A01N43/653 ,  A01P3/00 ,  C07C45/63 ,  C07C45/70 ,  C07C49/213 ,  C07D249/08 ,  C07D521/00

CPC classification number: C07D231/12 ,  C07C45/63 ,  C07C45/70 ,  C07C49/213 ,  C07D233/56 ,  C07D249/08 ,  C07C49/255 ,  C07C49/233

Abstract: in which X1 represents hydrogen or an alkyl radical, X2 represents hydrogen or an alkyl radical, R1 represents an alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl or optionally substituted aryl or aralkyl radical, R2 represents hydrogen or an alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl or optionally substituted aryl or aralkyl radical, R3 represents hydrogen or an alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl or optionally substituted aryl or aralkyl radical, and Y represents a keto group or a functional keto derivative, WHICH POSSESS FUNGICIDAL PROPERTIES.
1-SUBSTITUTED-1,2,4-TRIAZOLES OF THE FORMULA

Abstract translation: 其中X 1表示氢或烷基，X 2表示氢或烷基，R 1表示烷基，烯基，炔基，R 1表示烷基，链烯基，炔基， ，环烷基，环烯基或任选取代的芳基或芳烷基，R 2表示氢或烷基，烯基，炔基，环烷基，环烯基或任选取代的芳基或芳烷基，R 3表示氢或烷基，烯基，炔基，环烷基，环烯基或任选地 取代的芳基或芳烷基，Y表示酮基或官能酮衍生物，其具有无害的杀真菌性质。

公开(公告)号：US6423726B2

公开(公告)日：2002-07-23

申请号：US91126301

申请日：2001-07-23

Applicant: BAYER AG

Inventor： DUTZMANN STEFAN ,  ERDELEN CHRISTOPH ,  ANDERSCH WOLFRAM ,  DEHNE HEINZ-WILHELM ,  HARTWIG JUERGEN ,  STENZEL KLAUS ,  KRAMER WOLFGANG

IPC: A01N47/40 ,  A01N51/00 ,  A01N43/40 ,  A01N47/10

CPC classification number: A01N47/40 ,  A01N51/00 ,  A01N61/00 ,  A01N59/02 ,  A01N53/00 ,  A01N47/44 ,  A01N47/38 ,  A01N47/26 ,  A01N47/14 ,  A01N47/04 ,  A01N43/84 ,  A01N43/707 ,  A01N43/66 ,  A01N43/653 ,  A01N43/40 ,  A01N43/36 ,  A01N37/46 ,  A01N2300/00

Abstract: A composition includes synergistic amounts of:(a) a compound formula (I)wherein X represents =CH- or =N-; E represents an electron-withdrawing radical; R represents optionally substituted hetarylalkyl; A represents hydrogen, alkyl, or a bifunctional group which is linked to the radical Z; Z represents alkyl, -NH-alkyl, -N(alkyl)2 or a bifunctional group which is linked to the radical A, and(b) a fungicidal active compound, excluding cyclopropylcarboxamide derivatives and azolylmethylcycloalkanes. The combination of imidacloprid and a fungicidal active compound selected from the group consisting of tebuconazole and compounds of the formulais excluded.

Abstract translation: 组合物包括协同量的：（a）其中X表示= CH-或= N-的化合物式（I） E代表吸电子基团; R代表任选取代的杂芳基烷基; A表示与基团Z连接的氢，烷基或双官能团; Z表示烷基，-NH-烷基，-N（烷基）2或与基团A连接的双官能团，和（b）杀真菌活性化合物，不包括环丙基甲酰胺衍生物和唑基甲基环烷烃。 将吡虫啉和选自戊唑醇和式的化合物的杀真菌活性化合物的组合排除在外。

公开(公告)号：US3898341A

公开(公告)日：1975-08-05

申请号：US46993874

申请日：1974-05-14

Applicant: BAYER AG

Inventor： MEISER WERNER ,  BUCHEL KARL HEINZ ,  KRAMER WOLFGANG ,  GREWE FERDINAND ,  FROHBERGER PAUL-ERNST

IPC: A01N43/50 ,  A01P1/00 ,  A01P3/00 ,  C07C45/63 ,  C07C45/71 ,  C07D233/60 ,  C07D249/08 ,  C07D521/00 ,  A01N9/22

CPC classification number: C07D231/12 ,  C07C45/63 ,  C07C45/71 ,  C07D233/56 ,  C07D249/08 ,  C07C49/84

Abstract: Combating fungi with imidazole derivatives of the formula

IN WHICH R1 and R3 each independently is an optionally substituted alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, aryl or aralkyl radical, and R2 is hydrogen or one of the radicals recited for R1, X is oxygen or sulfur, and Y is a keto group or a functional derivative of a keto group, AND THEIR SALTS.

Abstract translation: 用下式的咪唑衍生物与R1反应：R1和R3各自独立地为任选取代的烷基，烯基，炔基，环烷基，环烯基，芳基或芳烷基，R2为氢或为R1所述的基团之一，X为氧 或硫，Y是酮基的酮基或官能衍生物，以及它们的盐。