Patent search ap:("LEO Pharma A/S") AND inv:"Tine Marianne DUUS" Page 1

1.

发明申请
METHODS FOR THE PREPARATION OF 1,3-BENZODIOXOLE HETEROCYCLIC COMPOUNDS 审中-公开

公开(公告)号：US20200262842A1

公开(公告)日：2020-08-20

申请号：US16062760

申请日：2016-12-16

Applicant: LEO Pharma A/S

Inventor： Allan Carsten DAHL , Gitte Holm JENSEN , Tine Marianne DUUS

IPC: C07D495/10

Abstract: The present invention relates to novel methods for the preparation of 1,3-benzo-dioxole heterocyclic compounds and intermediates for the same. The compounds are useful as PDE4 inhibitors.

2.

发明申请
NOVEL AMINO-IMIDAZOPYRIDINE DERIVATIVES AS JANUS KINASE INHIBITORS AND PHARMACEUTICAL USE THEREOF 审中-公开

公开(公告)号：US20190367512A1

公开(公告)日：2019-12-05

申请号：US16477249

申请日：2018-01-10

Applicant: LEO Pharma A/S

Inventor： Jens LARSEN , Mogens LARSEN , Lars Kyhn RASMUSSEN , Andreas RITZEN , Tine Marianne DUUS

IPC: C07D471/04

Abstract: The present invention relates to a compound according to formula (I) or pharmaceutically acceptable salts, hydrates, or solvates thereof; wherein R1 is C1-alkyl, R2 is C1-alkyl, R3 is C2-alkyl, R4 is hydrogen, R5 is hydrogen. The invention relates further to said compounds for use in therapy, to pharmaceutical compositions comprising said compounds, to said compounds for use in the treatment autoimmune diseases and to intermediates for the preparation of said compounds.

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