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公开(公告)号:US09700558B2
公开(公告)日:2017-07-11
申请号:US14771109
申请日:2014-03-17
申请人: VERONA PHARMA PLC
IPC分类号: A61K31/519 , A61K31/46 , A61K31/40 , A61K45/06 , A61K9/00 , A61K31/137 , A61K31/167 , A61K31/44 , A61K9/48 , A61M15/00
CPC分类号: A61K31/519 , A61K9/0075 , A61K9/0078 , A61K9/008 , A61K9/0095 , A61K9/4858 , A61K31/137 , A61K31/167 , A61K31/40 , A61K31/44 , A61K31/46 , A61K45/06 , A61M15/009 , A61M2202/064 , A61K2300/00
摘要: The invention provides a composition which comprises (a) a PDE3/PDE4 inhibitor which is 9,10-Dimethoxy-2-(2,4,6-trimethylphenylimino)-3-(N-carbamoyl-2-aminoethyl)-3,4,6,7-tetrahydro-2H-pyrimido[6,1-a]isoquinolin-4-one or a pharmaceutically acceptable acid addition salt thereof and (b) a muscarinic receptor antagonist.
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公开(公告)号:US10471063B2
公开(公告)日:2019-11-12
申请号:US15614440
申请日:2017-06-05
申请人: VERONA PHARMA PLC
IPC分类号: A61K31/519 , A61K31/40 , A61K45/06 , A61K9/00 , A61K31/137 , A61K31/167 , A61K31/44 , A61K31/46 , A61K9/48 , A61M15/00
摘要: The invention provides a composition which comprises (a) a PDE3/PDE4 inhibitor which is 9,10-Dimethoxy-2-(2,4,6-trimethylphenylimino)-3-(N-carbamoyl-2-aminoethyl)-3,4,6,7-tetrahydro-2H-pyrimido[6,1-a]isoquinolin-4-one or a pharmaceutically acceptable acid addition salt thereof and (b) a muscarinic receptor antagonist.
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公开(公告)号:US09717732B2
公开(公告)日:2017-08-01
申请号:US14771097
申请日:2014-03-17
申请人: VERONA PHARMA PLC
IPC分类号: A61K31/505 , A61K31/519 , A61K31/40 , A61K45/06 , A61K9/00 , A61K31/137 , A61K31/167 , A61K31/44 , A61K31/46 , A61K9/48 , A61M15/00
CPC分类号: A61K31/519 , A61K9/0075 , A61K9/0078 , A61K9/008 , A61K9/0095 , A61K9/4858 , A61K31/137 , A61K31/167 , A61K31/40 , A61K31/44 , A61K31/46 , A61K45/06 , A61M15/009 , A61M2202/064 , A61K2300/00
摘要: The invention provides a composition which comprises (a) a PDE3/PDE4 inhibitor which is 9,10-Dimethoxy-2-(2,4,6-trimethylphenylimino)-3-(N-carbamoyl-2-aminoethyl)-3,4,6,7-tetrahydro-2H-pyrimido[6,1-a]isoquinolin-4-one or a pharmaceutically acceptable acid addition salt thereof and (b) a β2-adrenergic receptor agonist.
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