公开(公告)号：US09497970B2

公开(公告)日：2016-11-22

申请号：US14903887

申请日：2014-07-14

Applicant: BASF SE

Inventor： Arun Narine ,  Nina Gertrud Bandur ,  Joachim Dickhaut ,  Raffael Koller ,  Wolfgang Von Deyn ,  Jean-Yves Wach ,  Vincent Salgado

IPC: C07D235/02 ,  C07D401/12 ,  C07D417/12 ,  C07D491/04 ,  C07D495/04 ,  A01N43/50 ,  A01N47/30 ,  A01N43/56 ,  A01N43/647 ,  A01N43/78 ,  A01N43/80 ,  A01N43/86 ,  A01N47/20 ,  A01N47/36 ,  A01N47/48 ,  C07D231/56 ,  C07D235/06 ,  C07D249/22 ,  C07D261/20 ,  C07D275/04

CPC classification number: A01N47/30 ,  A01N43/56 ,  A01N43/647 ,  A01N43/78 ,  A01N43/80 ,  A01N43/86 ,  A01N47/20 ,  A01N47/36 ,  A01N47/48 ,  C07D231/56 ,  C07D235/02 ,  C07D235/06 ,  C07D249/22 ,  C07D261/20 ,  C07D275/04 ,  C07D401/12 ,  C07D417/12 ,  C07D491/04 ,  C07D495/04

Abstract: The present invention relates to novel compounds of the formula I and the N-oxides, stereoisomers, tautomers and agriculturally or veterinarily acceptable salts thereof wherein C1 is C or CH; C2 is C or CH; A1 is N or C; A2 is N, C(R2), N(R3), O, S or C(R4,R5); and A3 is N, O, S, N(R6), C(R7) or C(R8,R9); where one or two non-adjacent bonds in the 5-membered ring formed by C1, C2, A1, A2 and A3 are double bonds, while the others are single bonds, provided that the bond between A1 and A2 or the bond between A1 and C1 or the bond between A2 and A3 or the bond between C1 and C2 or the bond between A3 and C2 is a double bond further provided that at least one of A1, A2 and A3 is N, N(R3) or N(R6), and where Ar, R1, R2, R3, R4, R5, R6, R7, R8, R9 and (R)k are as defined in the claims and in the description, which are useful for combating or controlling invertebrate pests, in particular arthropod pests and nematodes. The invention also relates to a method for controlling invertebrate pests by using these compounds and to plant propagation material and to an agricultural and a veterinary composition comprising said compounds.

公开(公告)号：US20150087509A1

公开(公告)日：2015-03-26

申请号：US14398239

申请日：2013-04-29

Applicant: BASF SE

Inventor： Karsten Körber ,  Florian Kaiser ,  Gemma Veitch ,  Wolfgang Von Deyn ,  Nina Gertrud Bandur ,  Joachim Dickhaut ,  Arun Narine ,  Deborah L. Culbertson ,  Paul Neese ,  Koshi Gunjima

IPC: C07D403/04 ,  A01N43/56 ,  A61K45/06 ,  A61K31/506 ,  A01N47/34 ,  C07D403/14 ,  C07F9/6558 ,  A01N57/24 ,  A61K31/675 ,  C07D405/14 ,  C07D409/14

CPC classification number: C07D403/04 ,  A01N43/56 ,  A01N47/34 ,  A01N47/36 ,  A01N57/24 ,  A01N57/32 ,  A61K31/506 ,  A61K31/675 ,  A61K45/06 ,  C07D403/14 ,  C07D405/14 ,  C07D409/14 ,  C07F9/247 ,  C07F9/65583

Abstract: The present invention relates to substituted pyrazole-containing compounds of formula (I), and the stereoisomers and salts thereof, wherein the substituents are as defined in the description.The present invention further relates to a method for combating or controlling invertebrate pests, to a method for protecting plant propagation material and/or the plants which grow therefrom, to plant propagation material comprising at least one compound according to the present invention, to a method for treating or protecting an animal from infestation or infection by parasites, to a process for the preparation of a composition for treating infested or infected animals and/or for protecting animals against infestation or infection by parasites, and to a compound according to the invention for use as a medicament.

Abstract translation: 本发明涉及式（I）的取代的含吡唑化合物及其立体异构体和盐，其中取代基如说明书中所定义。 本发明还涉及一种防治无脊椎害虫的方法，一种用于保护植物繁殖材料和/或从其生长的植物的方法，包括至少一种根据本发明的化合物的植物繁殖材料的方法， 用于治疗或保护动物免受寄生虫感染或感染，涉及制备用于治疗感染或感染动物的组合物和/或用于保护动物免受寄生虫感染或感染的方法，以及根据本发明的化合物 用作药物。

公开(公告)号：US11019820B2

公开(公告)日：2021-06-01

申请号：US15656293

申请日：2017-07-21

Applicant: BASF SE

Inventor： Arun Narine ,  Nina Gertrud Bandur ,  Joachim Dickhaut ,  Swetlana Derksen ,  Raffael Koller ,  Wolfgang Von Deyn ,  Jean-Yves Wach ,  Deborah L. Culbertson

IPC: A01N43/90 ,  C07D471/04 ,  C07D487/04 ,  C07D513/04 ,  C07D498/04

Abstract: Substituted pyrimidinium compounds of the general formula (I) and their uses for combating animal pests
The present invention relates to substituted pyrimidinium compounds of formula (I), to the stereoisomers, salts, tautomers and N-oxides thereof and to compositions comprising such compounds. The invention also relates to methods and uses of these substituted pyrimidinium compounds and of compositions thereof, for combating and controlling animal pests. Furthermore the invention relates also to pesticidal methods of applying such substituted pyrimidinium compounds.
The substituted pyrimidinium compounds of the present invention are defined by the following general formula (I): wherein X, Y, Z, R1, R2, A and Het are defined as in the description.

公开(公告)号：US10757938B2

公开(公告)日：2020-09-01

申请号：US16245471

申请日：2019-01-11

Applicant: BASF SE

Inventor： Martin John McLaughlin ,  Nina Gertrud Bandur ,  Matthias Pohlman ,  Jochen Dietz ,  Wolfgang Von Deyn

IPC: A01N43/40 ,  C07D405/14 ,  C07D401/06 ,  C07D405/06 ,  C07D417/06 ,  A01N43/54 ,  A01N43/78 ,  A01N53/00 ,  C07D401/14 ,  C07D417/14

Abstract: The present invention relates to N-acylimino compound of formula (I): wherein X is O or S, in particular O; m is an integer selected from 0, 1, 2, 3, 4, 5 or 6; Het is a 5 or 6 membered carbon-bound or nitrogen-bound heterocyclic ring, W1-W2-W3-W4 represents a carbon chain group connected to N and C═N, and thus forming a saturated, unsaturated, or partially unsaturated 5 or 6 membered nitrogen containing heterocycle, wherein W1, W2, W3 and W4 each individually represent CRvRw, R1, R2 may be hydrogen, halogen, etc. R3 may be hydrogen, halogen, CN, C1-C6-alkyl, etc. R4a, R4b if present, may be hydrogen, halogen, C1-C6-alkyl, etc. R5 may be hydrogen, halogen, C1-C6-alkyl, C1-C6-alkenyl, C1-C6-alkinyl, C3-C8-cycloalkyl, S(O)nNR9aR9b, NR9aR9b, C(═O)OR8, C(═O)NR9aR9b, C(═S)NR9aR9b, C(═O)R7a, C(═S)R7a, NR9a—C(═O)R7a, NR9a—C(═S)R7a, NR9a—S(O)nR8a, a moitey Q-phenyl, where the phenyl ring is optionally substituted with one or more, e.g. 1, 2, 3, 4 or 5 identical or different substituents R10, or a moiety Q-Het#, or R3 and R5 together may also form with the carbon atom they are bound to, a 3, 4, 5 or 6 membered saturated partially unsaturated carbocycle or heterocycle. The invention also relates to the use of the N-acylimino heterocyclic compounds, their stereoisomers, their tautomers and their salts, for combating invertebrate pests. Furthermore the invention relates also to methods of combating invertebrate pests, which comprises applying such compounds.

公开(公告)号：US09422280B2

公开(公告)日：2016-08-23

申请号：US14387600

申请日：2013-03-25

Applicant: BASF SE

Inventor： Nina Gertrud Bandur ,  Ralph Paulini ,  Florian Kaiser ,  Arun Narine ,  Joachim Dickhaut ,  Karsten Körber ,  Wolfgang Von Deyn ,  Swetlana Derksen ,  Deborah L. Culbertson ,  Nancy B. Rankl

IPC: A01N43/42 ,  C07D471/04 ,  A01N43/90 ,  C07D487/04

CPC classification number: C07D471/04 ,  A01N43/90 ,  C07D487/04

Abstract: The invention relates to N-substituted hetero-bicyclic compounds of formula (I), to the enantiomers, diastereomers and salts thereof and to compositions comprising such compounds. The invention also relates to methods and uses of these N-substituted hetero-bicyclic compounds, and of compositions comprising thereof, for combating and controlling animal pests. Furthermore the invention relates also to pesticidal methods of applying such N-substituted hetero-bicyclic compounds.The N-substituted hetero-bicyclic compounds of the present invention are defined by the following formula I: wherein A, B, X, Het, R1, R2, W1, W2, W3 and W4 are defined as in the description.

公开(公告)号：US20150166528A1

公开(公告)日：2015-06-18

申请号：US14407731

申请日：2013-06-04

Applicant: BASF SE

Inventor： Florian Kaiser ,  Arun Narine ,  Joachim Dickhaut ,  Karsten Körber ,  Nina Gertrud Bandur

IPC: C07D417/14 ,  A01N43/78

CPC classification number: C07D417/14 ,  A01N43/78 ,  A61K31/4439 ,  C07D417/04 ,  C07D417/12

Abstract: The present invention relates to pesticidal methods for the use and application of substituted 3-pyridyl thiazole compounds and the stereoisomers, salts, tautomers and N-oxides thereof and to compositions comprising the same. The invention also relates to insecticidal substituted 3-pyridyl thiazole compounds or of the compositions comprising such compounds for combating invertebrate pests and uses thereof.The substituted 3-pyridyl thiazole compounds of the present invention are defined by the following general formula (I): wherein m, k, R1, R2, R6, G, and A are defined as in the description.

Abstract translation: 本发明涉及使用和应用取代的3-吡啶基噻唑化合物及其立体异构体，盐，互变异构体和N-氧化物及其组合物的杀虫方法。 本发明还涉及杀虫取代的3-吡啶基噻唑化合物或包含用于防治无脊椎害虫的化合物的组合物及其用途。 本发明的取代的3-吡啶基噻唑化合物由以下通式（I）定义：其中m，k，R1，R2，R6，G和A如说明书所定义。

公开(公告)号：US20150057280A1

公开(公告)日：2015-02-26

申请号：US14389125

申请日：2013-03-27

Applicant: BASF SE

Inventor： Nina Gertrud Bandur ,  Ralph Paulini ,  Florian Kaiser ,  Arun Narine ,  Joachim Dickhaut ,  Karsten Korber

IPC: C07D213/50 ,  C07D213/48 ,  C07D401/14 ,  A01N43/54 ,  A01N43/78 ,  A01N43/84 ,  C07D213/52 ,  C07D213/53 ,  C07D401/06 ,  C07D417/06 ,  A01N43/40 ,  A01N43/56

CPC classification number: C07D213/50 ,  A01N43/40 ,  A01N43/54 ,  A01N43/56 ,  A01N43/60 ,  A01N43/76 ,  A01N43/78 ,  A01N43/84 ,  C07D213/46 ,  C07D213/48 ,  C07D213/52 ,  C07D213/53 ,  C07D213/61 ,  C07D401/06 ,  C07D401/14 ,  C07D405/06 ,  C07D413/06 ,  C07D417/06

Abstract: The invention relates to pyridylidene compounds of formula (I), to the enantiomers, diastereomers and salts thereof and to compositions comprising such compounds. The invention also relates to methods and uses of these N-substituted pyridylidene compounds, and of compositions comprising thereof, for combating and controlling animal pests. Furthermore the invention relates also to pesticidal methods of applying such N-substituted pyridylidene compounds.The N-substituted pyridylidene compounds of the present invention are defined by the following formula I: wherein X, Het, R1, R2, R3, R4 and R6 are defined as in the description.

Abstract translation: 本发明涉及式（I）的吡啶亚基化合物，其涉及其对映体，非对映异构体和盐以及包含这些化合物的组合物。 本发明还涉及这些N-取代的吡啶亚基化合物及其组合物的方法和用途，用于对抗和控制动物害虫。 此外，本发明还涉及施用这种N-取代的吡啶亚基化合物的杀虫方法。 本发明的N-取代的吡啶亚基化合物由下式I定义：其中X，Het，R 1，R 2，R 3，R 4和R 6如描述中所定义。