Benzimidazole derivatives, agricultural and horticultural fungicides
containing the same as an active ingredient and intermediate compounds
thereof
    11.
    发明授权
    Benzimidazole derivatives, agricultural and horticultural fungicides containing the same as an active ingredient and intermediate compounds thereof 失效
    苯并咪唑衍生物,含有与活性成分相同的农业和园艺杀真菌剂及其中间体化合物

    公开(公告)号:US5310747A

    公开(公告)日:1994-05-10

    申请号:US894007

    申请日:1992-06-02

    CPC分类号: C07D491/04 A01N43/90

    摘要: A benzimidazole derivative having the formula, ##STR1## wherein R is cyano or thiocarbamoyl; Q is lower alkyl or a group represented by the formula NQ.sup.1 Q.sup.2, in which Q.sup.1 and Q.sup.2 are independently lower alkyl, lower alkyl substituted with phenyl, lower alkenyl or lower alkynyl, or they form a lower alkylene ring when taken together at their ends which ring may include a hetero atom; X is hydrogen or halogen; and Z is a group which consists of (a) one oxygen atom or two non-adjacent oxygen atom, (b) --CF.sub.2 -- group and (c) any one of a single bond, --CF.sub.2 --, --CFH--, CFCl-- and --CH.sub.2 -- groups and forms a five-membered or six membered ring together with two adjacent carbon atoms of the benzene ring; is obtained by reacting a corresponding 2-cyanobenzimidazole compound and a sulfamoyl chloride derivative. The benzimidazole derivative is incorporated into agricultural and horticultural fungicides as an active ingredient.

    摘要翻译: 具有下式的苯并咪唑衍生物,其中R是氰基或硫代氨基甲酰基; Q是低级烷基或由式NQ1Q2表示的基团,其中Q1和Q2独立地是低级烷基,被苯基,低级链烯基或低级炔基取代的低级烷基,或者当它们的末端相互结合时,它们形成低级亚烷基环 可以包括杂原子; X是氢或卤素; Z为由(a)一个氧原子或两个不相邻氧原子组成的基团,(b)-CF2-基团和(c)单键,-CF2-,-CFH-,CFCl- 和-CH 2 - 基团,并与苯环的两个相邻碳原子一起形成五元或六元环; 是通过使相应的2-氰基苯并咪唑化合物和氨磺酰氯衍生物反应得到的。 苯并咪唑衍生物作为活性成分掺入农业和园艺杀真菌剂中。