公开(公告)号：US08114991B2

公开(公告)日：2012-02-14

申请号：US10771649

申请日：2004-02-03

Applicant: Hartmut Ahrens ,  Hansjörg Dietrich ,  Klemens Minn ,  Thomas Auler ,  Hermann Bieringer ,  Martin Hills ,  Heinz Kehne ,  Hubert Menne

Inventor： Hartmut Ahrens ,  Hansjörg Dietrich ,  Klemens Minn ,  Thomas Auler ,  Hermann Bieringer ,  Martin Hills ,  Heinz Kehne ,  Hubert Menne

IPC: C07D251/48 ,  A01N43/68

CPC classification number: C07D405/12 ,  A01N43/68 ,  C07D251/18 ,  C07D311/68 ,  C07D401/12

Abstract: Amino-1,3,5-triazines N-substituted with chiral bicyclic radicals, process for their preparation, compositions thereof, and their use as herbicides and plant growth regulators.The invention relates to an optically active compound of formula (I) or a salt thereof: wherein the various symbols are as defined in the description, to processes for their preparation, to compositions thereof, and to their use as herbicides or plant growth regulators. The invention also relates to novel intermediates of formula (III), (V) and (XIII) as defined in the description.

Abstract translation: 用手性双环基团N-取代的氨基-1,3,5-三嗪，其制备方法，其组合物及其作为除草剂和植物生长调节剂的用途。 本发明涉及式（I）的光学活性化合物或其盐：其中各种符号如说明书中所定义，其制备方法，组合物及其作为除草剂或植物生长调节剂的用途。 本发明还涉及如说明书中定义的式（III），（V）和（XIII）的新型中间体。

公开(公告)号：US07569519B2

公开(公告)日：2009-08-04

申请号：US11807820

申请日：2007-05-30

Applicant: Andreas Van Almsick ,  Lothar Willms ,  Hermann Bieringer ,  Hubert Menne ,  Thomas Auler

Inventor： Andreas Van Almsick ,  Lothar Willms ,  Hermann Bieringer ,  Hubert Menne ,  Thomas Auler

IPC: C07D231/12 ,  C07D231/14 ,  A01N43/56

CPC classification number: C07D307/18 ,  C07D307/20 ,  C07D307/33 ,  C07D309/12 ,  C07D309/18 ,  C07D319/06 ,  C07D405/12

Abstract: What is described are derivatives of benzoyl derivatives of the formula (I) and their use as herbicides. In this formula (I), R1, R2 and R3 are different radicals, X is a bridge atom selected from the group consisting of oxygen and sulfur and Het is a saturated heterocyclic group which comprises oxygen and carbon atoms.

Abstract translation: 所描述的是式（I）的苯甲酰基衍生物的衍生物及其作为除草剂的用途。 在该式（I）中，R 1，R 2和R 3是不同的基团，X是选自氧和硫的桥原子，Het是包含氧和碳原子的饱和杂环基。

公开(公告)号：US07211673B2

公开(公告)日：2007-05-01

申请号：US11325957

申请日：2006-01-05

Applicant: Michael G. Hoffmann ,  Hendrik Helmke ,  Lothar Willms ,  Thomas Auler ,  Hermann Bieringer ,  Hubert Menne

Inventor： Michael G. Hoffmann ,  Hendrik Helmke ,  Lothar Willms ,  Thomas Auler ,  Hermann Bieringer ,  Hubert Menne

IPC: C07D409/14 ,  A01N43/76

CPC classification number: C07D409/14 ,  A01N43/56 ,  C07D401/14 ,  C07D413/14 ,  C07D417/14

Abstract: A description is given of 4-trifluoromethylpyrazolyl-substituted pyridines and pyrimidines of formula (I) and of their use as herbicides. In this formula (I) R1, R2, R3 and R4 are various radicals, A is an aromatic or heteroaromatic radical, and Z is a nitrogen or carbon atom.

Abstract translation: 给出了式（I）的4-三氟甲基吡唑基取代的吡啶和嘧啶及其作为除草剂的用途的描述。 在该式（I）中，R 1，R 2，R 3和R 4是各种基团，A 是芳族或杂芳族基团，Z是氮或碳原子。

公开(公告)号：US20070066481A1

公开(公告)日：2007-03-22

申请号：US11529087

申请日：2006-09-28

Applicant: Frank Ziemer ,  Hermann Bieringer ,  Christopher Rosinger ,  Erwin Hacker ,  Lothar Willms

Inventor： Frank Ziemer ,  Hermann Bieringer ,  Christopher Rosinger ,  Erwin Hacker ,  Lothar Willms

IPC: A01N25/32

CPC classification number: A01N25/32 ,  A01N43/56 ,  A01N2300/00

Abstract: What is described are herbicidal compositions comprising herbicidal compounds of the formula (I) and a compound of the formula (II) which acts as a safener. In the formulae (I) and (II), the symbols R1 to R17 denote hydrogen, halogen, nitro and various organic radicals. These herbicidal compositions have a particularly high compatibility with useful plants.

Abstract translation: 所描述的是包含式（I）的除草化合物和作为安全剂的式（II）化合物的除草组合物。 在式（I）和（II）中，符号R 1至R 17表示氢，卤素，硝基和各种有机基团。 这些除草组合物与有用植物具有特别高的相容性。

公开(公告)号：US07135434B2

公开(公告)日：2006-11-14

申请号：US10265925

申请日：2002-10-07

Applicant: Frank Ziemer ,  Lothar Willms ,  Hermann Bieringer ,  Erwin Hacker

Inventor： Frank Ziemer ,  Lothar Willms ,  Hermann Bieringer ,  Erwin Hacker

IPC: A01N25/32 ,  A01N43/50 ,  A01P13/00

CPC classification number: A01N43/18 ,  A01N25/32 ,  A01N43/56 ,  A01N43/80 ,  A01N2300/00 ,  A01N43/78

Abstract: This invention provides for, inter alia, a herbicidal composition comprising a mixture of: A. a herbicidally effective amount of at least one compound of the formula where V and Z are defined in the specification; and B. an antidote.

公开(公告)号：US07078369B2

公开(公告)日：2006-07-18

申请号：US10659201

申请日：2003-09-09

Applicant: Hansjörg Dietrich ,  Christian Waldraff ,  Lothar Willms ,  Hermann Bieringer ,  Christopher Rosinger ,  Felix Thürwächter ,  Thomas Auler

Inventor： Hansjörg Dietrich ,  Christian Waldraff ,  Lothar Willms ,  Hermann Bieringer ,  Christopher Rosinger ,  Felix Thürwächter ,  Thomas Auler

IPC: C07D251/42 ,  C07D251/48 ,  C07D251/52 ,  A01N43/68 ,  A01N47/36

CPC classification number: C07D521/00 ,  A01N47/36 ,  C07C311/16 ,  C07C311/39 ,  C07D207/32 ,  C07D239/42 ,  C07D239/47 ,  C07D239/52 ,  C07D251/42 ,  C07D251/46 ,  C07D295/155 ,  C07D403/12

Abstract: Phenylsulfonyl ureas are disclosed for controlling harmful plants in crops of useful plants. Also disclosed are processes for the preparation of phenylsulfonyl ureas, and their use as herbicides and plant growth regulators.

Abstract translation: 公开了苯磺酰脲用于控制有用植物作物中的有害植物。 还公开了制备苯磺酰脲的方法及其作为除草剂和植物生长调节剂的用途。

公开(公告)号：US20060111240A1

公开(公告)日：2006-05-25

申请号：US11323085

申请日：2005-12-30

Applicant: Erwin Hacker ,  Hermann Bieringer ,  Lothar Willms

Inventor： Erwin Hacker ,  Hermann Bieringer ,  Lothar Willms

IPC: A01N57/00

CPC classification number: A01N57/20 ,  A01N2300/00

Abstract: Herbicide combinations (A)+(B), if appropriate in the presence of safeners, with an effective content of (A) broad-spectrum herbicides from the group (A1) glufosinate (salts) and related compounds (A2) glyphosate (salts) and related compounds such as sulfosate, (A3) imidazolinones, (A4) herbicidal azoles from the group of the protoporphyrinogen oxidase inhibitors (PPO inhibitors) (A5) cyclohexanedione herbicides and (A6) heteroaryloxyphenoxypropionic acid herbicides and (B) one or more herbicides from the group of the compounds consisting of (B0) one or more structurally different herbicides from the abovementioned group (A) or (B1) foliar- and soil-acting herbicides against monocotyledonous and dicotyledonous harmful plants or (B2) herbicides which can be employed selectively in maize against dicots, or (B3) foliar- and soil-acting herbicides which can be employed selectively in maize, predominantly against dicotyledonous harmful plants, or herbicides from several of groups (B0) to (B3) are suitable for controlling harmful plants in maize which consists of tolerant or resistant mutants or transgenic maize plants and the maize crops are tolerant to the herbicides (A) and (B), if appropriate in the presence of safeners, which are contained in the combination.

Abstract translation: （A）+（B），如果适合，在安全剂存在下，有效含量（A）来自（A1）草铵膦（盐）和相关化合物（A2）的广谱除草剂草甘膦（盐） 以及来自原卟啉原氧化酶抑制剂（PPO抑制剂）（A5）环己二酮除草剂和（A6）杂芳基氧基苯氧基丙酸除草剂组的磺酰基，（A3）咪唑啉酮，（A4）除草唑等相关化合物和（B）一种或多种除草剂 由（B0）组成的一组化合物，所述组合物来自上述组（A）中的一种或多种结构不同的除草剂或（B1）对单子叶和双子叶植物有害植物的叶面和土壤作用除草剂或（B2）除草剂，其可以选择性地使用 在玉米对双子叶植物中，或（B3）叶面和土壤作用的除草剂，其可以选择性地用于玉米，主要是针对双子叶植物有害植物或来自几个组（B0）至（B 3）适用于控制由耐受性或抗性突变体或转基因玉米植物组成的玉米中的有害植物，并且玉米作物对除草剂（A）和（B）是有耐受性的，如果适用，则在安全剂存在下 组合。

公开(公告)号：US20060014643A1

公开(公告)日：2006-01-19

申请号：US10531830

申请日：2003-10-01

Applicant: Erwin Hacker ,  Hermann Bieringer ,  Hans Huff ,  Lothar Willms

Inventor： Erwin Hacker ,  Hermann Bieringer ,  Hans Huff ,  Lothar Willms

IPC: A01N43/56 ,  A01N43/647 ,  A01N43/713 ,  A01N43/72

CPC classification number: A01N43/56 ,  A01N43/76 ,  A01N2300/00

Abstract: Combinations of a compound of formula (I) or a salt thereof in which R1, R2, R3, R4 and n are as defined in the description, and one or more aryloxyphenoxypropionate herbicides or agriculturally acceptable salts thereof are useful for increasing weed control.

Abstract translation: 式（I）化合物或其盐的组合，其中R 1，R 2，R 3，R 4，R 4， 和n如说明书中所定义，并且一种或多种芳氧基苯氧基丙酸酯除草剂或其农业上可接受的盐可用于增加杂草控制。

公开(公告)号：US20050267184A1

公开(公告)日：2005-12-01

申请号：US11058951

申请日：2005-02-16

Applicant: Thomas Seitz ,  Andreas Almsick ,  Lothar Willms ,  Thomas Auler ,  Hermann Bieringer ,  Hubert Menne

Inventor： Thomas Seitz ,  Andreas Almsick ,  Lothar Willms ,  Thomas Auler ,  Hermann Bieringer ,  Hubert Menne

IPC: A01N43/56 ,  C07D209/08 ,  C07D231/20 ,  C07D403/12 ,  A61K31/4196 ,  A61K31/4152 ,  C07D231/44

CPC classification number: C07D231/20 ,  A01N43/56 ,  C07D403/12

Abstract: A description is given of derivatives of benzoylpyrazoles of the formula (I) and of their use as herbicides. In this formula (I) R1a, R1b, R1c, R2, R3, R4 and R5 stand for various radicals, X for a bridging atom, L for a carbon chain and Y for a chalcogen atom.

Abstract translation: 给出式（I）的苯甲酰基吡唑衍生物及其作为除草剂的用途的描述。 在该式（I）中，R 1a，R 1b，R 1c，R 2，R 2， 3个，R 4和R 5代表各种基团，X代表桥连原子，L代表碳链，Y代表硫属原子。

公开(公告)号：US06750177B2

公开(公告)日：2004-06-15

申请号：US10382004

申请日：2003-03-05

Applicant: Erwin Hacker ,  Hermann Bieringer ,  Hansjörg Krähmer

Inventor： Erwin Hacker ,  Hermann Bieringer ,  Hansjörg Krähmer

IPC: A01N4736

CPC classification number: A01N47/36 ,  A01N43/80 ,  A01N43/70 ,  A01N37/40 ,  A01N37/22 ,  A01N25/32 ,  A01N2300/00

Abstract: Herbicidal compositions with acylated aminophenylsulfonylureas Herbicide combinations with an effective content of components (A), (B) and (C) have improved herbicidal effects: (A) one or more herbicides selected from the group of the compounds of the formula (I) or their salts, (B) denotes one or more herbicides from the group of the compounds of the formula (II) and their salts, (C) denotes one or more herbicides from the group of the compounds consisting of (C1) flumioxazin (C2) alachlor (C3) metolachlor (C4) acetochlor (C5) dimethenamid (C6) pethoxamid (C7) atrazine (C8) simazone (C9) cyanazine (C10) terbuthylazine (C11) metribuzin (C12) isoxaflutole (C13) fluthiamid (C14) terbutryne (C15) nicosulfuron (C16) rimsulfuron (C17) primsulfuron (C18) pendimethalin (C19) sulcotrione (C20) dicamba (C21) mesotrione (C22) linuron (C23) benoxacor (C24) metosulam (C25) flumetsulam (C26) sethoxydim (C27) cycloxydim (C28) clethodim (C29) clefoxidim (C30) aclonifen (C31) MCPA (C32) 2, 4-D (C33) bromoxynil (C34) bentazone (C35) fluthiacet (C36) pyridate (C37) diflufenzopyr (C38) carfentrazone (C39) clopyralid (C40) halosulfuron (C41) thifensulfuron (C42) prosulfuron (C43) tritosulfuron (C44) sulfosulfuron (C45) ethoxysulfuron (C46) tribenuron (C47) amidosulfuron (C48) mecoprop (C49) dichlorporp (C50) fluroxypyr (C51) profluazol (C52) amicarbazone (C53) trifloxysulfuron (C54) glufosinate (C55) glufosinate-ammonium (C56) glyphosate (C57) glyphosate-isopropytammonium (C58) imazapyr (C59) imazethapyr (C60) imazamethabenz (C61) imazamox (C62) imazaquin and (C63) imazapic (AC 263,222).

Abstract translation: 具有酰化氨基苯基磺酰脲的除草组合物与组分（A），（B）和（C）有效含量的除草剂组合具有改善的除草效果：（A）一种或多种选自式（I）化合物或其 盐，（B）表示来自式（II）化合物及其盐的一种或多种除草剂，（C）表示一种或多种由（C1）氟草胺（C2）甲草胺 （C3）异丙甲草胺（C4）乙草胺（C5）二甲酰氨基（C6）花青素（C7）莠去津（C8）西蒙松（C9）氰嗪（C10）特丁津（C11）甲基溴（C12）异唑（C13） ）C（C）（C26）苯磺隆（C16）嘧磺隆（C17）头孢磺隆（C18）二甲戊乐宁（C19）三氧六环（C20）麦草畏（C21）甲基磺草酮（C22） （C28）烯草酮（C29）clefoxidim（C30）aclonifen（C31）MCPA（C32）2,4-D（C33） （C34）苯磺隆（C34）苯扎硫酮（C35）氟磺隆（C36）吡啶（C37）二氟苯并吡喃（C38）氟哌唑酮（C39）氯吡磺隆（C40）卤磺隆（C41）噻吩磺隆（C42） C54）草甘膦（C47）草甘膦（C47）草甘膦（C47）二氯甲氧基丙酸（C49）二氯弹（C50）氟草烟（C51）丙酰脲（C52）氨基脲（C53）三氟嘧磺隆（C54）草铵膦 异丙基铵（C58）咪草烟（C59）咪草烟（C60）咪草螨辛（C61）咪唑莫斯（C62）咪草胺和（C63）咪唑（AC 263,222）。