公开(公告)号：US4948417A

公开(公告)日：1990-08-14

申请号：US212835

申请日：1988-06-29

申请人： Markus Lindig ,  Karlfried Dickore ,  Kurt Findeisen ,  Hans-Joachim Santel ,  Robert R. Schmidt ,  Harry Strang

发明人： Markus Lindig ,  Karlfried Dickore ,  Kurt Findeisen ,  Hans-Joachim Santel ,  Robert R. Schmidt ,  Harry Strang

IPC分类号： C07D401/06 ,  A01N47/38 ,  C07D249/12 ,  C07D401/12

CPC分类号： C07D401/12 ,  A01N47/38 ,  C07D249/12

摘要： Herbicidal substituted triazolinones of the formula ##STR1## in which R.sup.1 represents hydrogen, alkyl, alkenyl, alkynyl, halogenoalkyl, halogenoalkenyl, halogenoalkynyl, alkoxyalkyl, alkoxy, cycloalkylalkyl, cycloalkyl or in each case optionally substituted aralkyl or aryl,R.sup.2 represents alkyl, alkenyl, alkynyl, halogenoalkyl, halogenoalkenyl, halogenoalkynyl, alkoxyalkyl, alkoxy, cycloalkylalkyl, cycloalkyl or in each case optionally substituted aralkyl or aryl,R.sup.3 and R.sup.4 independently of one another each represent hydrogen, alkyl, alkenyl, alkynyl, halogenoalkyl, halogenoalkenyl, halogenoalkinyl, cyanoalkyl, hydroxyalkyl, alkoxyalkyl, alkoximinoalkyl, alkoxycarbonylalkyl, alkoxycarbonylalkenyl, alkylaminoalkyl, dialkylaminoalkyl, in each case optionally substituted cycloalkyl, cycloalkylalkyl, cyclcalkenyl or cycloalkenylalkyl, optionally substituted heterocyclylalkyl, in each case optionally substituted aralkyl, aroyl or aryl, alkoxy, alkenyloxy, alkynyloxy, aralkyloxy or aryloxy or, together with the nitrogen atom to which they are bonded, represent an optionally substituted heterocycle,X represents oxygen or sulphur andY represents oxygen or sulphur,where X represents sulphur only, when at least one of the radicals R.sup.3 or R.sup.4 does not simultaneously represent hydrogen, methyl or ethyl.

摘要翻译： R 1代表氢，烷基，烯基，炔基，卤代烷基，卤代烯基，卤代炔基，烷氧基烷基，烷氧基，环烷基烷基，环烷基或在各种情况下是任选取代的芳烷基或芳基的除草取代的三唑啉酮，其中R 1表示烷基， ，烯基，炔基，卤代烷基，卤代烯基，卤代炔基，烷氧基烷基，烷氧基，环烷基烷基，环烷基或在每种情况下任选取代的芳烷基或芳基，R 3和R 4彼此独立地表示氢，烷基，烯基，炔基，卤代烷基，卤代烯基，卤代烯基 烷氧基烷基，烷氧基羰基烷基，烷氧基羰基烯基，烷基氨基烷基，二烷基氨基烷基，在各种情况下均为任选取代的环烷基，环烷基烷基，环烯基或环烯基烷基，任选取代的杂环基烷基，在任何情况下均为任选取代的芳烷基，芳酰基或芳基，烷氧基，烯氧基， ，芳烷氧基或芳氧基 r与其键合的氮原子一起代表任选取代的杂环，X表示氧或硫，Y表示氧或硫，其中X表示仅硫，当基团R3或R4中的至少一个不同时 代表氢，甲基或乙基。

公开(公告)号：US4909830A

公开(公告)日：1990-03-20

申请号：US269809

申请日：1988-11-10

申请人： Uta Jensen-Korte ,  Hans-Joachim Santel ,  Robert R. Schmidt ,  Harry Strang

发明人： Uta Jensen-Korte ,  Hans-Joachim Santel ,  Robert R. Schmidt ,  Harry Strang

IPC分类号： A01N43/56 ,  C07C67/00 ,  C07C241/00 ,  C07C257/04 ,  C07C257/06 ,  C07C313/00 ,  C07C323/62 ,  C07D231/52

CPC分类号： C07D231/52 ,  C07C257/06

摘要： Herbicidal 3-aminopyrazolin-5-ones of the formula ##STR1## in which R.sup.1 stands for alkyl, alkenyl, halogenoalkyl, halogenoalkenyl, alkoxyalkyl, alkylthioalkyl, cycloalkyl, for optionally substituted aralkyl or for optionally substituted aryl,R.sup.2 stands for hydrogen or alkyl,R.sup.3 stands for hydrogen or alkyl,R.sup.4 stands for hydrogen, alkyl, alkenyl, alkinyl, alkoxyalkyl, alkylthioalkyl, alkoxycarbonylalkyl or alkanoyl, orR.sup.3 and R.sup.4 together stand for an alkylene or alkenylene radical, each of which is divalent,X stands for halogen, alkyl, alkoxy, alkylthio, halogenoalkyl. halogenoalkoxy or halogenoalkylthio, andZ stands for hydrogen, halogen, alkyl, alkoxy, alkylthio, halogenoalkyl, halogenoalkoxy or halogenoalkylthio,and acid addition salts thereof. Intermediates of the formula ##STR2## are also disclosed.

摘要翻译： R1代表烷基，烯基，卤代烷基，卤代烯基，烷氧基烷基，烷硫基烷基，环烷基，任选取代的芳烷基或任选取代的芳基的式（Ⅰ）的除草3-氨基吡唑啉-5-酮代表氢 或烷基，R3代表氢或烷基，R4代表氢，烷基，烯基，炔基，烷氧基烷基，烷硫基烷基，烷氧基羰基烷基或烷酰基，或R3和R4一起代表一个亚烷基或亚烯基， 卤素，烷基，烷氧基，烷硫基，卤代烷基。 卤代烷氧基或卤代烷硫基，Z代表氢，卤素，烷基，烷氧基，烷硫基，卤代烷基，卤代烷氧基或卤代烷硫基，及其酸加成盐。 还公开了式（II）的中间体。