公开(公告)号：US20070135453A1

公开(公告)日：2007-06-14

申请号：US10579395

申请日：2004-12-14

Applicant: Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

Inventor： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC: A01N43/90 ,  C07D487/04

CPC classification number: C07D487/04 ,  A01N43/90

Abstract: The present invention relates to 6-(2,4,6-trihalophenyl)triazolopyrimidines of the formula I in which the substituents are as defined below: R1 is alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl or a five- or six-member saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R2 is hydrogen or one of the groups mentioned under R1, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain one to three further heteroatoms from the group consisting of O, N and S as ring members; R1 and/or R2 may be substituted as defined in the description; L1, L2, L3 are chlorine or fluorine, where at least one group is chlorine; X is cyano, alkyl, alkoxy, alkenyloxy, haloalkoxy or haloalkenyloxy; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

Abstract translation: 本发明涉及式I的6-（2,4,6-三卤代苯基）三唑并嘧啶，其中取代基如下：R 1是烷基，卤代烷基，环烷基，卤代环烷基，烯基， 卤代烯基，环烯基，卤代环烯基，炔基，卤代炔基或苯基，萘基或五或六元饱和的部分不饱和或芳族杂环，其含有一至四个由O，N和S组成的组的杂原子，R 2 R 1是氢或R 1，R 2和R 2中所提及的基团之一，与它们的氮原子一起 还可以形成通过N连接的五元或六元杂环基或杂芳基，并且可以含有一个至三个其它由O，N和S组成的组的杂原子作为环成员; R 1和/或R 2可以如说明书中所定义的取代; L 1，L 2，L 3 3是氯或氟，其中至少一个基团是氯; X是氰基，烷基，烷氧基，烯氧基，卤代烷氧基或卤代烯氧基; 制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20070054926A1

公开(公告)日：2007-03-08

申请号：US10566360

申请日：2004-07-07

Applicant: Jordi Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

Inventor： Jordi Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

IPC: A01N43/64 ,  A01N43/90

CPC classification number: A01N43/90 ,  A01N2300/00

Abstract: Fungicidal mixtures comprising, as active components, 1) the triazolopyrimidine derivative of the formula I and 2) epoxiconazole of the formula II, in a synergistically effective amount, methods for controlling harmful fungi from the class of the Oomycetes using mixtures of the compound I with the compound II, the use of the compound I with the compound II for preparing such mixtures and compositions comprising these mixtures are described.

Abstract translation: 包含作为活性组分的1）式I的三唑并嘧啶衍生物和2）式II的环氧唑的协同有效量的方法，使用化合物I与化合物I的混合物来控制来自卵菌纲的有害真菌的方法 描述了化合物II，化合物I与化合物II用于制备这些混合物的用途和包含这些混合物的组合物。

公开(公告)号：US07186672B2

公开(公告)日：2007-03-06

申请号：US10466168

申请日：2002-01-17

Applicant: Bernd Müller ,  Ingo Rose ,  Eberhard Ammermann ,  Reinhard Stierl ,  Gisela Lorenz ,  Siegfried Strathmann ,  Maria Scherer ,  Klaus Schelberger ,  Joachim Leyendecker ,  Egon Haden

Inventor： Bernd Müller ,  Ingo Rose ,  Eberhard Ammermann ,  Reinhard Stierl ,  Gisela Lorenz ,  Siegfried Strathmann ,  Maria Scherer ,  Klaus Schelberger ,  Joachim Leyendecker ,  Egon Haden

IPC: A01N25/26

CPC classification number: A01N35/04 ,  A01N47/24 ,  A01N43/653 ,  A01N2300/00

Abstract: Fungicidal mixtures comprising a) a benzophenone of the formula I, b) a carbamate of the formula II, and c) an azole derivative of the formula III in a synergistically effective amount, and a method for controlling harmful fungi using mixtures of the compounds I, II and III are described. The active compounds of the formulae I, II and III are defined in the description.

Abstract translation: 杀真菌混合物，其包含a）式I的二苯甲酮，b）式II的氨基甲酸酯，和c）协同有效量的式III的唑衍生物，以及使用化合物I的混合物来控制有害真菌的方法 ，II和III。 式I，II和III的活性化合物在说明书中定义。

公开(公告)号：US20060241128A1

公开(公告)日：2006-10-26

申请号：US10532719

申请日：2003-11-04

Applicant: Jordi Tormo I Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

Inventor： Jordi Tormo I Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC: A01N43/90 ,  C07D487/04

CPC classification number: C07C69/65 ,  A01N43/90 ,  C07D487/04

Abstract: Substituted 6-(2-halogenphenyl)-triazolopyrimidines of formula I in which R1 denote alkyl, alkenyl, alkynyl, alkadienyl, haloalkyl, haloalkenyl, cycloalkyl, phenyl, naphthyl, or a 5- or 6-membered saturated, unsaturated, or aromatic heterocycle, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, wherein R1 and R2 radicals may be substituted as defined in the description, R2 denote hydrogen, or a group mentioned for R1; or R1 and R2 together with the interjacent nitrogen atom represent a 5- or 6-membered heterocycle, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which ring may be substituted as defined in the description; Hal is halogen; L1, L3 independently denote hydrogen, halogen, or alkyl; L2 is hydrogen, halogen, haloalkyl, or NH2, NHRb, or N(Rb)2, wherein Rb is as defined in the description, wherein at least one from L1, L2, and L3 is not hydrogen; X is halogen, cyano, alkyl, alkoxy, haloalkoxy or alkenyloxy. processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi.

Abstract translation: 其中R 1表示烷基，烯基，炔基，链二烯基，卤代烷基，卤代烯基，环烷基，苯基，萘基或5-或6-元的取代的6-（2-卤代苯基） - 三唑并嘧啶， 含有1至4个氮原子或1至3个氮原子和1个硫或氧原子的饱和，不饱和或芳族杂环，其中R 1和R 2可以是 如说明书中所定义，R 2表示氢或R 1所提及的基团; 或R 1和R 2连同中间的氮原子代表含有1-4个氮原子或一至三个氮原子的一个或多个六元杂环，一个 硫或氧原子，该环可以如说明书中所定义取代; 卤素是卤素; L 1，L 3独立地表示氢，卤素或烷基; L 2是氢，卤素，卤代烷基或NH 2，NHR b或/或N（R b） 其中R b如描述中所定义，其中至少一个L 1，L 2， ，而L 3不是氢; X是卤素，氰基，烷基，烷氧基，卤代烷氧基或烯氧基。 其制备方法，含有它们的组合物及其用于对抗植物病原真菌的用途。

公开(公告)号：US20060217400A1

公开(公告)日：2006-09-28

申请号：US10539559

申请日：2003-12-17

Applicant: Bernd Müller ,  Jordi Blasco ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

Inventor： Bernd Müller ,  Jordi Blasco ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

IPC: A01N43/90 ,  C07D487/04

CPC classification number: C07D487/04 ,  A01N43/90

Abstract: Triazolopyrimidines of the formula I in which the index n and the substituents R1, R2 and R3 are as defined in the description, and processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.

Abstract translation: 其中指数n和取代基R 1，R 2和R 3的式I的三唑并嘧啶如说明书中所定义，以及 描述了制备这些化合物的方法，包含它们的组合物及其用于控制​​有害真菌的用途。

公开(公告)号：US20060211573A1

公开(公告)日：2006-09-21

申请号：US10548690

申请日：2004-03-24

Applicant: Jordi Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schalfer ,  Frank Schieweck ,  Anja Schwogler ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

Inventor： Jordi Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schalfer ,  Frank Schieweck ,  Anja Schwogler ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC: A01N43/90 ,  C07D487/04

CPC classification number: C07D487/04 ,  A01N43/90

Abstract: 7-(Alkenylamino)triazolopyrimidines of the formula I wherein the substituents have the following meanings: L is halogen, alkyl, haloalkyl, alkoxy, amino, NHR or NR2; R is alkyl or alkyl-carbonyl; m is 1, 2, 3, 4 or 5; X is halogen, cyano, alkyl, haloalkyl or alkoxy; R1 is alkyl or haloalkyl; R2 is hydrogen, alkyl or haloalkyl; R3 is alkenyl, which can be unsubstituted or partially or completely halogenated or can be substituted according to the Description; R4 is hydrogen or alkyl, R3 and R4 can also, together with the nitrogen atom to which they are bonded, form a five- or six-membered unsaturated ring which can be interrupted by an atom from the group consisting of O, N and S and/or can carry one or more sub-stituents. Processes for the preparation of these compounds, preparations comprising them and their use in the control of harmful phytopathogenic fungi.

Abstract translation: 式（I）的7-（烯基氨基）三唑并嘧啶，其中取代基具有以下含义：L是卤素，烷基，卤代烷基，烷氧基，氨基，NHR或NR 2。 R是烷基或烷基 - 羰基; m为1,2,3,4或5; X是卤素，氰基，烷基，卤代烷基或烷氧基; R 1是烷基或卤代烷基; R 2是氢，烷基或卤代烷基; R 3是烯基，其可以是未取代的或部分的或完全卤化的或可以根据描述被取代; R 4是氢或烷基，R 3和R 4也可以与它们所键合的氮原子一起形成五元环 - 或六元不饱和环，其可以被来自O，N和S的原子中断，和/或可以携带一个或多个亚取代基。 制备这些化合物的方法，包含它们的制剂及其在控制有害植物病原真菌中的用途。

公开(公告)号：US07071334B2

公开(公告)日：2006-07-04

申请号：US10474461

申请日：2002-04-06

Applicant: Jordi Tormo i Blasco ,  Hubert Sauter ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

Inventor： Jordi Tormo i Blasco ,  Hubert Sauter ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC: C07D487/04 ,  A01N43/90

CPC classification number: C07D487/04 ,  A01N43/90

Abstract: 6-(2-Chloro-6-fluoro-phenyl)-triazolopyrimidines of formula (I), in which R1 and R2 independently denote hydrogen or alkyl, alkenyl, alkynyl, alkadienyl, or haloalkyl, cycloalkyl, bicycloalkyl, phenyl, naphthyl, or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or where R1 and R2 radicals may be unsubstituted or partially or fully halogenated or may be substituted as defined in the description. R1 and R2 together with the interjacent nitrogen atom represent a 5- or 6-membered heterocyclic ring, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which may be substituted; X is cyano, alkoxy, haloalkoxy or alkenyloxy; processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi

Abstract translation: 式（I）的6-（2-氯-6-氟 - 苯基） - 三唑并嘧啶，其中R 1和R 2独立地表示氢或烷基，烯基， 炔基，链烯基或卤代烷基，环烷基，二环烷基，苯基，萘基或含有1-4个氮原子或1-3个氮原子和一个硫或氧原子的5-或6-元杂环基，或5-或6-元 含有一至四个氮原子或一至三个氮原子和一个硫或氧原子的杂芳基，或其中R 1和R 2基团可以是未取代的或部分或完全的 卤化的或可以如说明书中所定义的取代。 R 1和R 2与中间的氮原子一起表示含有1-4个氮原子或一至三个氮原子的一个5-或6-元杂环，一个 硫或氧原子，其可以被取代; X是氰基，烷氧基，卤代烷氧基或烯氧基; 其制备方法，含有它们的组合物及其用于对抗植物病原真菌的用途

公开(公告)号：US20060100220A1

公开(公告)日：2006-05-11

申请号：US10532769

申请日：2003-11-14

Applicant: Jordi Tormo I Blasco ,  Thomas Grote ,  Eberhard Ammermann ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

Inventor： Jordi Tormo I Blasco ,  Thomas Grote ,  Eberhard Ammermann ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

IPC: A01N43/90 ,  A01N43/80 ,  A01N43/50

CPC classification number: A01N43/90 ,  A01N2300/00

Abstract: Fungicidal mixtures, comprising A) the triazolopyrimidine of the formula I and B) imidazole derivatives of the formula II where X1 and X2 are halogen and phenyl which may be substituted by halogen or alkyl or X1 and X2 together with the bridging C═C double bond form a difluoromethylenedioxyphenyl group; X3 is cyano or halogen, and X4 is dialkylamino or isoxazol-4-yl which may carry two alkyl radicals, in a synergistically effective amount, methods for controlling harmful fungi using mixtures of the compounds I and II, compositions comprising these compounds and the use of the compounds I and II for preparing such mixtures are described.

Abstract translation: 杀真菌混合物，其包含A）式I的三唑并嘧啶和B）式II的咪唑衍生物，其中X 1和X 2是卤素和可以被 卤素或烷基或X 1和X 2连同桥连CC双键形成二氟亚甲二氧基苯基; X 3是氰基或卤素，X 4是可以以协同有效量存在两个烷基的二烷基氨基或异恶唑-4-基，用于控制有害真菌的方法 描述了使用化合物I和II的混合物，包含这些化合物的组合物和化合物I和II用于制备这些混合物的用途。

公开(公告)号：US20060079537A1

公开(公告)日：2006-04-13

申请号：US10531898

申请日：2003-11-14

Applicant: Jordi Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

Inventor： Jordi Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC: A61K31/519 ,  C07D487/04

CPC classification number: C07D487/04 ,  A01N43/90

Abstract: 2-Substituted triazolopyrimidines of the formula I, in which the substituents are as defined below: L are halogen, cyano, nitro, alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, —C(═O)-A or S(═O)pA′; A and A′ are as defined in the description; p is 0, 1 or 2; m is 0, 1, 2, 3, 4 or 5; X is cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; R1,R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, phenyl, naphthyl or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered ring which may be interrupted by an atom from the group consisting of O, N and S, where R1 and/or R2 may be substituted as defined in the description; and R3 is cyano, hydroxyl, alkoxy, alkenyloxy, haloalkoxy, haloalkenyloxy, NR1R2 or S(O)nR31, where n and R31 are as defined in the description; Processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi are described.

Abstract translation: 氰基，硝基，烷基，烯基，炔基，卤代烷基，卤代烯基，烷氧基，烯氧基，炔氧基，卤代烷氧基，-C（ - O） - 取代的取代基如下： -A或S（-O） A'; A和A'如说明书所定义; p为0,1或2; m为0,1,2,3,4或5; X是氰基，烷基，卤代烷基，烷氧基或卤代烷氧基; R 1，R 2是氢，烷基，卤代烷基，环烷基，卤代环烷基，烯基，链二烯基，卤代烯基，环烯基，炔基，卤代炔基或环炔基，苯基，萘基或五 - 至十元饱和的，部分不饱和的或芳族杂环，其含有一至四个由O，N和S组成的组的杂原子，R 1和R 2连同 它们所连接的氮原子也可以形成可被来自O，N和S的原子间隔的五元或六元环，其中R 1和/或 R 2可以如说明书中定义的取代; 和R 3是氰基，羟基，烷氧基，烯氧基，卤代烷氧基，卤代烯氧基，NR 1 R 2或S（O）n 其中n和R 31如在说明书中所定义的; 描述了制备这些化合物的方法和中间体，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20060074093A1

公开(公告)日：2006-04-06

申请号：US10532770

申请日：2003-11-14

Applicant: Jordi Blasco ,  Thomas Grote ,  Eberhard Ammermann ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

Inventor： Jordi Blasco ,  Thomas Grote ,  Eberhard Ammermann ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

IPC: A01N43/40 ,  A01N43/90

CPC classification number: A01N43/90 ,  A01N43/40 ,  A01N2300/00

Abstract: Fungicidal mixtures, comprising A) the triazolopyrimidine of the formula I and B) amide compounds of the formula II where X1 and X2 are halogen, nitro, cyano, alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl, haloalkynyl, alkoxy, haloalkoxy, haloalkylthio, alkylsulfinyl or alkylsulfonyl; x is 1, 2, 3 or 4; and y is 1, 2, 3, 4 or 5; in a synergistically effective amount, methods for controlling harmful fungi using mixtures of the compounds I and II, compositions comprising these compounds and the use of the compounds I and II for preparing such mixtures are described.

Abstract translation: 杀真菌混合物，其包含A）式I的三唑并嘧啶和B）式II的酰胺化合物，其中X 1和X 2是卤素，硝基，氰基，烷基， 烯基，炔基，卤代烷基，卤代烯基，卤代炔基，烷氧基，卤代烷氧基，卤代烷硫基，烷基亚磺酰基或烷基磺酰基; x为1,2,3或4; y为1,2,3,4或5; 在协同有效量下，描述了使用化合物I和II的混合物来控制有害真菌的方法，包含这些化合物的组合物以及化合物I和II用于制备这种混合物的用途。