2-Substituted 7-Aminoazolopyrimidines, Processes For Their Preparation And Their Use For Controlling Harmful Fungi, And Compositions Comprising These Compounds
    4.
    发明申请
    2-Substituted 7-Aminoazolopyrimidines, Processes For Their Preparation And Their Use For Controlling Harmful Fungi, And Compositions Comprising These Compounds 审中-公开
    2-取代的7-氨基偶氮嘧啶,其制备方法及其用于控制​​有害真菌和包含这些化合物的组合物

    公开(公告)号:US20080139581A1

    公开(公告)日:2008-06-12

    申请号:US11885536

    申请日:2006-03-02

    IPC分类号: A01N43/90 A01P3/00 C07D487/04

    CPC分类号: C07D487/04

    摘要: 2-Substituted 7-aminoazolopyrimidines of the formula I in which the substituents are as defined below: R1 is hydrogen, halogen, cyano, alkyl, haloalkyl, alkenyl, alkynyl, cycloalkyl, alkoxy, alkoxyalkyl, benzyloxyalkyl, alkoxyalkenyl or alkoxyalkynyl; R2 is hydrogen, halogen, cyano, alkyl, haloalkyl, alkenyl, alkynyl, cycloalkyl, alkoxy, alkoxyalkyl and alkylthioalkyl, where the carbon chains in R1 and/or R2 may be substituted according to the description; R3 is halogen, cyano, NRARB, hydroxyl, mercapto, alkyl, haloalkyl, cycloalkyl, alkoxy, alkylthio, cycloalkoxy, cycloalkylthio, carboxyl, formyl, alkylcarbonyl, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, phenyl, phenoxy, phenylthio, benzyloxy, benzylthio, alkyl-S(O)m—; A is N and CRx; Rx is hydrogen or one of the groups mentioned under R3; processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

    摘要翻译: 2-取代的式I的7-氨基偶氮嘧啶,其中取代基如下:R 1是氢,卤素,氰基,烷基,卤代烷基,烯基,炔基,环烷基,烷氧基,烷氧基烷基,苄氧基烷基 ,烷氧基烯基或烷氧基炔基; R 2是氢,卤素,氰基,烷基,卤代烷基,烯基,炔基,环烷基,烷氧基,烷氧基烷基和烷硫基烷基,其中R 1和/或R 2可以根据描述代替; R 3是卤素,氰基,NR B,B,羟基,巯基,烷基,卤代烷基,环烷基,烷氧基,烷硫基,环烷氧基,环烷硫基 ,羧基,甲酰基,烷基羰基,烷氧基羰基,烯氧基羰基,炔氧基羰基,苯基,苯氧基,苯硫基,苄氧基,苄硫基,烷基-S(O) A是N和CR R x是氢或R 3中提到的基团之一; 制备这些化合物的方法和中间体,包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

    7-Aminomethyl-1,2,4-Triazolo[1,5-A]Pyrimidine Compounds And Their Use For Controlling Pathogenic Fungi
    5.
    发明申请
    7-Aminomethyl-1,2,4-Triazolo[1,5-A]Pyrimidine Compounds And Their Use For Controlling Pathogenic Fungi 审中-公开
    7-氨基甲基-1,2,4-三唑并[1,5-A]嘧啶化合物及其用于控制​​致病真菌

    公开(公告)号:US20080076785A1

    公开(公告)日:2008-03-27

    申请号:US11663982

    申请日:2005-09-27

    IPC分类号: A01N43/54 A01P3/00 C07D239/70

    CPC分类号: A01N43/90 C07D487/04

    摘要: The invention relates to 7-aminomethyl-1,2,4-triazolo[1,5-a]pyrimidine compounds of general formula (I) and the agriculturally compatible salts of said compounds. In said formula: R1 and R2 represent hydrogen, alkyl, haloalkyl, alkoxy, cycloalkyl, bicycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a 5- or 6-membered saturated, partially unsaturated or aromatic heterocycle, containing 1 to 4 heteroatoms from the group containing O, N or S, or R1 and R2, together with the nitrogen atom to which they are bonded, can also form a five- or six-membered heterocyclyl or heteroaryl, which is bonded by means of N and can contain 1 to 3 additional heteroatoms from the group containing O, N and S as the ring member and can be substituted according to the description; R3 and R4 represent hydrogen, alkyl, haloalkyl, haloalkoxy, alkoxy, or alkoxyalkyl; X represents halogen, cyano, a 5- or 6-membered saturated, partially unsaturated or aromatic heterocycle, containing 1, 2 or 3 heteroatoms from the group containing O, N or S as the ring member, alkyl, alkoxy, alkenyl or alkynyl, whereby the latter 4 groups can be substituted according to the description; L is defined as cited in the claims and the description; and m represents 0, 1, 2, 3, 4 or 5. The invention also relates to the use of the triazolopyrimidine compounds of general formula (I) and their agriculturally compatible salts for controlling plant-pathogenic fungi, to a method for controlling plant-pathogenic fungi, containing at least one compound of general formula (I) and/or an agriculturally compatible salt of said compound and at least one liquid or solid carrier.

    摘要翻译: 本发明涉及通式(I)的7-氨基甲基-1,2,4-三唑并[1,5-a]嘧啶化合物和所述化合物的农业上相容的盐。 在所述式中:R 1和R 2表示氢,烷基,卤代烷基,烷氧基,环烷基,二环烷基,卤代环烷基,烯基,链烯基,卤代烯基,环烯基,卤代环烯基,炔基,卤代炔基或苯基,萘基或5-或6-元饱和, 部分不饱和或芳族杂环,含有1至4个含有O,N或S的杂原子,或R 1和R 2与它们所键合的氮原子一起也可以形成五元或六元杂环基或杂芳基 ,其通过N键合并且可以含有来自含有O,N和S的基团的1至3个另外的杂原子作为环成员,并且可以根据描述进行取代; R3和R4代表氢,烷基,卤代烷基,卤代烷氧基,烷氧基或烷氧基烷基; X代表卤素,氰基,含有1,2或3个杂原子的5-或6-元饱和的部分不饱和或芳族杂环,所述杂环含有作为环成员的O,N或S,烷基,烷氧基,烯基或炔基, 由此后4个组可以根据描述被替代; L定义为权利要求书和说明书中引用的; 和m表示0,1,2,3,4或5.本发明还涉及通式(I)的三唑并嘧啶化合物及其农业上相容的盐用于控制植物致病真菌的用途,用于控制植物的方法 致病真菌,含有至少一种通式(I)的化合物和/或所述化合物的农业上相容的盐和至少一种液体或固体载体。