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公开(公告)号:US06943162B2
公开(公告)日:2005-09-13
申请号:US10466847
申请日:2002-01-23
申请人: Ronnie Lee Hale , Brad Richard Henke , Millard Hurst Lambert, III , Amy Tsai Lu , Paul Kenneth Spearing , Philip Stewart Turnbull
发明人: Ronnie Lee Hale , Brad Richard Henke , Millard Hurst Lambert, III , Amy Tsai Lu , Paul Kenneth Spearing , Philip Stewart Turnbull
IPC分类号: A61P5/30 , C07D251/38 , C07D251/70 , C07D401/12 , C07D417/12 , C07D403/02 , A61K31/53 , A61P35/00
CPC分类号: C07D401/12 , C07D251/38 , C07D251/70 , C07D417/12
摘要: Triazine derivatives of formula (I), which exhibit pharmacological activity at estrogen receptors alpha (ER alpha) and beta (ER beta) are described herein. The described invention also includes compositions and medicaments containing the triazine derivatives as well as processes for the preparation and use of such compounds, compositions and medicaments.
摘要翻译: 本文描述了在雌激素受体α(ERα)和β(ERβ))表现出药理活性的式(I)的三嗪衍生物。 所述发明还包括含有三嗪衍生物的组合物和药物以及这些化合物,组合物和药物的制备和使用方法。