公开(公告)号：US20110306639A1

公开(公告)日：2011-12-15

申请号：US12740673

申请日：2008-11-25

申请人： ZhaoHai Qin ,  Yongqiang Ma ,  Wangcang Su ,  Lei Wang ,  Zheng Zhang ,  Bengbin Zhao ,  Jiangsheng Fang

发明人： ZhaoHai Qin ,  Yongqiang Ma ,  Wangcang Su ,  Lei Wang ,  Zheng Zhang ,  Bengbin Zhao ,  Jiangsheng Fang

IPC分类号： A01N43/40 ,  A01P7/04 ,  C07D405/12 ,  A01N47/44 ,  C07C281/16 ,  C07D213/53

CPC分类号： C07C281/18 ,  A01N51/00

摘要： The present invention discloses hydrocarbylidene nitrohydrozinecarboximidamides and the use thereof as well as a method for making the same. The structural general formula of the compounds are shown in formula I, wherein, R1 is C1-C10 saturated and/or unsaturated aliphatic hydrocarbonyl, benzyl, substituted benzyl, halogenated picolyl, halogenated thiazolyl methyl, tetrahydrofuryl methyl or oxazolyl methyl; R2 is hydrogen, C1-C5 saturated and/or unsaturated aliphatic hydrocarbonyl, phenyl, substituted phenyl, pyridyl or substituted pyridyl; R3 is hydrogen, C1-C10 saturated and/or unsaturated aliphatic hydrocarbonyl, furyl, phenyl, substituted phenyl, benzyl or substituted benzyl. The tests of insecticidal activity show that the hydrocarbylidene nitrohydrozinecarboximidamides shown by formula (I) have high preventive efficiency against insect pests of plants, such as aphid, plant hopper, cotton bollworm, asparagus caterpillar, and the like, and can be used as plant insecticides.

摘要翻译： 本发明公开了亚烃基硝基氢亚肟酰亚胺及其用途及其制备方法。 化合物的结构通式如式I所示，其中R1为C1-C10饱和和/或不饱和脂族烃基，苄基，取代苄基，卤代吡啶甲基，卤代噻唑基甲基，四氢呋喃基甲基或恶唑基甲基; R2是氢，C1-C5饱和和/或不饱和脂族烃基，苯基，取代的苯基，吡啶基或取代的吡啶基; R3是氢，C1-C10饱和和/或不饱和脂族烃基，呋喃基，苯基，取代的苯基，苄基或取代的苄基。 杀虫活性试验表明，式（I）所示的亚烃基硝基氢化胂甲酰胺对蚜虫，植物料斗，棉铃虫，芦笋毛虫等植物的害虫具有较高的预防效果，可用作植物杀虫剂 。