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    Process for the preparation of 9-amino substituted 9,10-dihydropyrrolo[2,1-b][1,3]benzotiazepines
    1.
    发明授权
    Process for the preparation of 9-amino substituted 9,10-dihydropyrrolo[2,1-b][1,3]benzotiazepines 失效
    制备9-氨基取代的9,10-二氢吡咯并[2,1-b] [1,3]苯并氮杂的方法

    公开(公告)号：US07078521B2

    公开(公告)日：2006-07-18

    申请号：US10343629

    申请日：2001-07-20

    申请人： Patrizia Minetti ,  Domenico Mastrojanno

    发明人： Patrizia Minetti ,  Domenico Mastrojanno

    IPC分类号： C07D513/04

    CPC分类号： C07D513/04

    摘要： A process is described for the preparation of compounds with the following formula where the groups are as defined below; in particular, R1 is a substituted amine; said process includes essentially the reaction of pyrrolobenzothiazepin-9-one with amine R1H to give the corresponding enamine, which is subsequently transformed into the final compound

    摘要翻译： 描述了用于制备具有下式的化合物的方法，其中基团如下所定义; 特别地，R 1是取代的胺; 所述方法基本上包括吡咯并苯并硫氮杂-9-酮与胺R 1 H的反应，得到相应的烯胺，随后将其转化为最终化合物