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    Indazole derivatives
    1.
    发明授权
    Indazole derivatives 失效
    吲唑衍生物

    公开(公告)号：US07919517B2

    公开(公告)日：2011-04-05

    申请号：US12275614

    申请日：2008-11-21

    申请人： Yoshihisa Ohta ,  Fumihiko Kanai ,  Shinji Nara ,  Yutaka Kanda ,  Hiroshi Umehara ,  Yukimasa Shiotsu ,  Tomoki Naoe ,  Hitoshi Kiyoi ,  Keiko Kawashima ,  Hiromi Ando ,  Motoki Miyama

    发明人： Yoshihisa Ohta ,  Fumihiko Kanai ,  Shinji Nara ,  Yutaka Kanda ,  Hiroshi Umehara ,  Yukimasa Shiotsu ,  Tomoki Naoe ,  Hitoshi Kiyoi ,  Keiko Kawashima ,  Hiromi Ando ,  Motoki Miyama

    IPC分类号： A61K31/416 ,  C07D231/56

    CPC分类号： C07D231/56

    摘要： The present invention provides a compound represented by Formula (I): [wherein R1 represents CONR1aR1b (wherein R1a and R1b may be the same or different and each represents a hydrogen atom, substituted or unsubstituted lower alkyl, substituted or unsubstituted aryl, substituted or unsubstituted ararkyl or a substituted or unsubstituted heterocyclic group, or R1a and R1b are combined together with the adjacent nitrogen atom thereto to form a substituted or unsubstituted heterocyclic group) or the like, R2 represents a hydrogen atom, CONR2aR2b (wherein R2a and R2b may be the same or different and each represents a hydrogen atom, substituted or unsubstituted lower alkyl, substituted or unsubstituted aryl, substituted or unsubstituted ararkyl or a substituted or unsubstituted heterocyclic group, or R2a and R2b are combined together with the adjacent nitrogen atom thereto to form a substituted or unsubstituted heterocyclic group), NR2cR2d (wherein R2c and R2d may be the same or different and each represents a hydrogen atom, substituted or unsubstituted lower alkyl, substituted or unsubstituted lower alkanoyl, substituted or unsubstituted aroyl, substituted or unsubstituted heteroaroyl, substituted or unsubstituted ararkyl, substituted or unsubstituted lower alkylsulfonyl or substituted or unsubstituted lower arylsulfonyl) or the like].

    摘要翻译： 本发明提供由式（I）表示的化合物：[其中R1表示CONR1aR1b（其中R1a和R1b可以相同或不同，各自表示氢原子，取代或未取代的低级烷基，取代或未取代的芳基，取代或未取代的 芳基或取代或未取代的杂环基，或者R1a和R1b与相邻的氮原子一起形成取代或未取代的杂环基）等，R2表示氢原子，CONR2aR2b（其中R2a和R2b可以是 各自表示氢原子，取代或未取代的低级烷基，取代或未取代的芳基，取代或未取代的芳基或取代或未取代的杂环基，或者R 2a和R 2b与相邻的氮原子一起形成取代基 或未取代的杂环基），NR2cR2d（其中R2c和R2d可以相同或不同 取代或未取代的杂芳酰基，取代或未取代的芳酰基，取代或未取代的低级烷基磺酰基或取代或未取代的低级芳基磺酰基）等，其中R 1表示氢原子，取代或未取代的低级烷基，取代或未取代的低级烷酰基，取代或未取代的芳酰基， 。

    Magnetic recording and reproducing apparatus with selective loading of different sized magnetic tapes
    2.
    发明授权
    Magnetic recording and reproducing apparatus with selective loading of different sized magnetic tapes 失效
    具有选择性加载不同尺寸磁带的磁记录和再现装置

    公开(公告)号：US4866550A

    公开(公告)日：1989-09-12

    申请号：US171746

    申请日：1988-03-22

    申请人： Keiichi Ohashi ,  Hiroshi Umehara ,  Hajime Nagahashi

    发明人： Keiichi Ohashi ,  Hiroshi Umehara ,  Hajime Nagahashi

    IPC分类号： H02M7/219 ,  G11B15/665 ,  G11B15/675 ,  G11B25/06

    CPC分类号： G11B15/6653 ,  G11B15/67544 ,  G11B15/67565 ,  G11B25/066

    摘要： A magnetic recording and reproducing apparatus which enables selective loading of a plurality of kinds of magnetic tape cassettes of different sizes, including a slider which receives a large magnetic tape cassette horizontally from an insertion position of the large magnetic tape cassette so as to displace the large magnetic tape cassette horizontally and then, lowers the large magnetic tape cassette vertically and an adapter chassis into which a small magnetic tape cassette is fitted so as to be locked thereto. Upon detection of fitting of the small magnetic tape cassette into the adapter chassis, a magnetic tape is drawn from the small magnetic tape cassette by first and second tape drawing arms mounted on the adapter chassis and upon detection of a state in which the magnetic tape has been drawn from the small magnetic tape cassette and the slider has been displaced to a position for performing recording and reproduction, the adapter chassis is loaded onto the slider located at the position for performing recording and reproduction.

    摘要翻译： 一种磁记录和再现装置，其能够选择性地装载多种不同尺寸的磁带盒（1,3），包括滑块（6），滑块（6）从大的磁带盒（3）的水平插入位置 使大型磁带盒（3）水平移位，然后使大型磁带盒（3）垂直移动，并将适配器底盘（14）放入小型磁带盒（1）中， ）被装配以便被锁定在其上。 在检测到小型磁带盒（1）装配到适配器底座（14）中时，通过第一和第二带状拉伸臂（22,23）从小型磁带盒（1）中抽出磁带（1a） 安装在适配器底盘（14）上，并且在检测到磁带（1a）已经从小型磁带盒（1）中被拉出并且滑块（6）已经移位到位置（6P）的状态下 执行记录和再现时，适配器底盘（14）被加载到位于位置（6P）处的用于执行记录和再现的滑块（6）上。

    INDAZOLE DERIVATIVES
    4.
    发明申请
    INDAZOLE DERIVATIVES 失效
    吲哚衍生物

    公开(公告)号：US20090082348A1

    公开(公告)日：2009-03-26

    申请号：US12275614

    申请日：2008-11-21

    申请人： Yoshihisa Ohta ,  Fumihiko Kanai ,  Shinji Nara ,  Yutaka Kanda ,  Hiroshi Umehara ,  Yukimasa Shiotsu ,  Tomoki Naoe ,  Hitoshi Kiyoi ,  Keiko Kawashima ,  Hiromi Ando ,  Motoki Miyama

    发明人： Yoshihisa Ohta ,  Fumihiko Kanai ,  Shinji Nara ,  Yutaka Kanda ,  Hiroshi Umehara ,  Yukimasa Shiotsu ,  Tomoki Naoe ,  Hitoshi Kiyoi ,  Keiko Kawashima ,  Hiromi Ando ,  Motoki Miyama

    IPC分类号： A61K31/5377 ,  A61K31/416 ,  A61K31/496 ,  A61K31/454 ,  A61K31/506 ,  A61K31/4439 ,  A61P35/00

    CPC分类号： C07D231/56

    摘要： The present invention provides a compound represented by Formula (I): [wherein R1 represents CONR1aR1b (wherein R1a and R1b may be the same or different and each represents a hydrogen atom, substituted or unsubstituted lower alkyl, substituted or unsubstituted aryl, substituted or unsubstituted ararkyl or a substituted or unsubstituted heterocyclic group, or R1a and R1b are combined together with the adjacent nitrogen atom thereto to form a substituted or unsubstituted heterocyclic group) or the like, R2 represents a hydrogen atom, CONR2aR2b (wherein R2a and R2b may be the same or different and each represents a hydrogen atom, substituted or unsubstituted lower alkyl, substituted or unsubstituted aryl, substituted or unsubstituted ararkyl or a substituted or unsubstituted heterocyclic group, or R2a and R2b are combined together with the adjacent nitrogen atom thereto to form a substituted or unsubstituted heterocyclic group), NR2cR2d (wherein R2c and R2d may be the same or different and each represents a hydrogen atom, substituted or unsubstituted lower alkyl, substituted or unsubstituted lower alkanoyl, substituted or unsubstituted aroyl, substituted or unsubstituted heteroaroyl, substituted or unsubstituted ararkyl, substituted or unsubstituted lower alkylsulfonyl or substituted or unsubstituted lower arylsulfonyl) or the like].

    摘要翻译： 本发明提供由式（I）表示的化合物：[其中R1表示CONR1aR1b（其中R1a和R1b可以相同或不同，各自表示氢原子，取代或未取代的低级烷基，取代或未取代的芳基，取代或未取代的 芳基或取代或未取代的杂环基，或者R1a和R1b与相邻的氮原子一起形成取代或未取代的杂环基）等，R2表示氢原子，CONR2aR2b（其中R2a和R2b可以是 各自表示氢原子，取代或未取代的低级烷基，取代或未取代的芳基，取代或未取代的芳基或取代或未取代的杂环基，或者R 2a和R 2b与相邻的氮原子一起形成取代基 或未取代的杂环基），NR2cR2d（其中R2c和R2d可以相同或不同 取代或未取代的芳酰基，取代或未取代的芳酰基，取代或未取代的低级烷基磺酰基或取代或未取代的低级芳基磺酰基）等。 。

    Indazole derivatives
    5.
    发明授权
    Indazole derivatives 失效
    吲唑衍生物

    公开(公告)号：US07470717B2

    公开(公告)日：2008-12-30

    申请号：US10548475

    申请日：2004-07-30

    申请人： Yoshihisa Ohta ,  Fumihiko Kanai ,  Shinji Nara ,  Yutaka Kanda ,  Hiroshi Umehara ,  Yukimasa Shiotsu ,  Tomoki Naoe ,  Hitoshi Kiyoi ,  Keiko Kawashima ,  Hiromi Ando ,  Motoki Miyama

    发明人： Yoshihisa Ohta ,  Fumihiko Kanai ,  Shinji Nara ,  Yutaka Kanda ,  Hiroshi Umehara ,  Yukimasa Shiotsu ,  Tomoki Naoe ,  Hitoshi Kiyoi ,  Keiko Kawashima ,  Hiromi Ando ,  Motoki Miyama

    IPC分类号： A61K31/416 ,  C07D231/56

    CPC分类号： C07D231/56

    摘要： The present invention provides a compound represented by Formula (I): [wherein R1 represents CONR1aR1b (wherein R1a and R1b may be the same or different and each represents a hydrogen atom, substituted or unsubstituted lower alkyl, substituted or unsubstituted aryl, substituted or unsubstituted ararkyl or a substituted or unsubstituted heterocyclic group, or R1a and R1b are combined together with the adjacent nitrogen atom thereto to form a substituted or unsubstituted heterocyclic group) or the like, R2 represents a hydrogen atom, CONR2aR2b (wherein R2a and R2b may be the same or different and each represents a hydrogen atom, substituted or unsubstituted lower alkyl, substituted or unsubstituted aryl, substituted or unsubstituted ararkyl or a substituted or unsubstituted heterocyclic group, or R2a and R2b are combined together with the adjacent nitrogen atom thereto to form a substituted or unsubstituted heterocyclic group), NR2cR2d (wherein R2c and R2d may be the same or different and each represents a hydrogen atom, substituted or unsubstituted lower alkyl, substituted or unsubstituted lower alkanoyl, substituted or unsubstituted aroyl, substituted or unsubstituted heteroaroyl, substituted or unsubstituted ararkyl, substituted or unsubstituted lower alkylsulfonyl or substituted or unsubstituted lower arylsulfonyl) or the like].

    摘要翻译： 本发明提供由式（I）表示的化合物：[其中R1表示CONR1aR1b（其中R1a和R1b可以相同或不同，各自表示氢原子，取代或未取代的低级烷基，取代或未取代的芳基，取代或未取代的 芳烷基或取代或未取代的杂环基，或者R1a和R1b与相邻的氮原子一起形成取代或未取代的杂环基）等，R2表示氢原子，CONR2aR2b（其中R2a和R2b可以是 各自表示氢原子，取代或未取代的低级烷基，取代或未取代的芳基，取代或未取代的芳烷基或取代或未取代的杂环基，或R 2a和R 2b与相邻的氮原子一起形成取代基 或未取代的杂环基），NR2cR2d（其中R2c和R2d可以相同或不同 取代或未取代的杂芳酰基，取代或未取代的芳烷基，取代或未取代的低级烷基磺酰基或取代或未取代的低级芳基磺酰基）等，其中R 1代表氢原子，取代或未取代的低级烷基，取代或未取代的低级烷酰基，取代或未取代的芳酰基， 。

    DISASTER-PREVENTING DEVICE
    6.
    发明申请
    DISASTER-PREVENTING DEVICE 审中-公开
    防灾装置

    公开(公告)号：US20120285710A1

    公开(公告)日：2012-11-15

    申请号：US13558535

    申请日：2012-07-26

    申请人： Hiroshi Umehara ,  Yuji Sugie

    发明人： Hiroshi Umehara ,  Yuji Sugie

    IPC分类号： A62C37/36

    CPC分类号： A62C5/006 ,  A62C3/16 ,  A62C37/36 ,  G08B17/00 ,  G08B17/113 ,  G08B25/007

    摘要： [Problem to be Solved] A low-cost simple extinguishing device, which is installed in small space such as the interior of a board and carries out fire detection and extinguishment, is provided.[Solution] A disaster-preventing device 10 is provided with: a battery that supplies a power source; a fire detecting unit 12 that detects fire; and an aerosol generating unit 14 that generates and discharges, to outside, aerosol for extinguishment by combustion of a solid extinguishing agent when the fire detecting unit 12 detects the fire. The fire detecting unit 12 outputs fire warning by sound and display when the fire is detected. The disaster-preventing device 10 can be installed at an arbitrary position in the interior of the board by a magnet sheet 32.

    摘要翻译： [待解决的问题]提供了一种安装在诸如板内部的小空间中并执行火灾探测和熄灭的低成本简单灭火装置。 [解决方案]防灾装置10具备：供给电源的电池; 检测火灾的火灾检测单元12; 以及气雾发生单元14，其在火灾检测单元12检测到火灾时，通过固体灭火剂的燃烧产生并排出气溶胶以熄灭。 火灾检测单元12在检测到火灾时，通过声音输出火灾警报和显示。 防灾装置10可以通过磁片32安装在板的内部的任意位置。

    Indazole derivatives
    8.
    发明申请
    Indazole derivatives 失效
    吲唑衍生物

    公开(公告)号：US20070117856A1

    公开(公告)日：2007-05-24

    申请号：US10548475

    申请日：2004-07-30

    申请人： Yoshihisa Ohta ,  Fumihiko Kanai ,  Shinji Nara ,  Yutaka Kanda ,  Hiroshi Umehara ,  Yukimasa Shiotsu ,  Tomoki Naoe ,  Hitoshi Kiyoi ,  Keiko Kawashima ,  Hiromi Ando ,  Motoki Miyama

    发明人： Yoshihisa Ohta ,  Fumihiko Kanai ,  Shinji Nara ,  Yutaka Kanda ,  Hiroshi Umehara ,  Yukimasa Shiotsu ,  Tomoki Naoe ,  Hitoshi Kiyoi ,  Keiko Kawashima ,  Hiromi Ando ,  Motoki Miyama

    IPC分类号： A61K31/416 ,  C07D231/56

    CPC分类号： C07D231/56

    摘要： The present invention provides a compound represented by Formula (I): [wherein R1 represents CONR1aR1b (wherein R1a and R1b may be the same or different and each represents a hydrogen atom, substituted or unsubstituted lower alkyl, substituted or unsubstituted aryl, substituted or unsubstituted ararkyl or a substituted or unsubstituted heterocyclic group, or R1a and R1b are combined together with the adjacent nitrogen atom thereto to form a substituted or unsubstituted heterocyclic group) or the like, R2 represents a hydrogen atom, CONR2aR2b (wherein R2a and R2b may be the same or different and each represents a hydrogen atom, substituted or unsubstituted lower alkyl, substituted or unsubstituted aryl, substituted or unsubstituted ararkyl or a substituted or unsubstituted heterocyclic group, or R2a and R2b are combined together with the adjacent nitrogen atom thereto to form a substituted or unsubstituted heterocyclic group), NR2cR2d (wherein R2c and R2d may be the same or different and each represents a hydrogen atom, substituted or unsubstituted lower alkyl, substituted or unsubstituted lower alkanoyl, substituted or unsubstituted aroyl, substituted or unsubstituted heteroaroyl, substituted or unsubstituted ararkyl, substituted or unsubstituted lower alkylsulfonyl or substituted or unsubstituted lower arylsulfonyl) or the like].

    摘要翻译： 本发明提供由式（I）表示的化合物：[其中R 1表示CONR 1a 1b 1b（其中R 1a） R 1b和R 1b可以相同或不同，各自表示氢原子，取代或未取代的低级烷基，取代或未取代的芳基，取代或未取代的芳烷基或取代或未取代的杂环基， 或R 1a和R 1b与相邻的氮原子一起形成取代或未取代的杂环基）等，R 2 O， >表示氢原子，其中R 2a，R 2b和R 2b可以相同或不同， 各自表示氢原子，取代或未取代的低级烷基，取代或未取代的芳基，取代或未取代的芳烷基或取代或未取代的杂环基，或R 2b和R 2b >与t结合在一起 它与氮原子相邻以形成取代或未取代的杂环基），NR 2c R 2d（其中R 2c和R 2d） 取代或未取代的低级烷酰基，取代或未取代的芳酰基，取代或未取代的杂芳酰基，取代或未取代的芳烷基，取代或未取代的低级烷基磺酰基或 取代或未取代的低级芳基磺酰基等）。

    Ab1 KINASE INHIBITORS
    10.
    发明申请
    Ab1 KINASE INHIBITORS 审中-公开
    Ab1激酶抑制剂

    公开(公告)号：US20120329794A1

    公开(公告)日：2012-12-27

    申请号：US12305146

    申请日：2007-06-29

    申请人： Yukimasa Shiotsu ,  Kenichi Ishii ,  Hiroshi Umehara ,  Shiro Akinaga

    发明人： Yukimasa Shiotsu ,  Kenichi Ishii ,  Hiroshi Umehara ,  Shiro Akinaga

    IPC分类号： A61K31/416 ,  A61K31/4439 ,  C12N9/99 ,  A61K31/454 ,  A61P35/00 ,  A61P35/02 ,  A61K31/5377 ,  A61K31/496

    CPC分类号： C07D231/56 ,  A61K31/416 ,  A61K31/4439 ,  A61K31/454 ,  A61K31/496 ,  A61K31/5377 ,  C07D401/06 ,  C07D403/10 ,  C07D413/12

    摘要： The present invention provides an Abelson kinase (Abl kinase) inhibitor which comprises, as an active ingredient, an indazole derivative represented by Formula (I) (wherein R1 represents substituted or unsubstituted aryl or a substituted or unsubstituted heterocyclic group) or a pharmaceutically acceptable salt thereof,an Abl kinase inhibitor which comprises, as an active ingredient, an indazole derivative represented by Formula (Ia) [wherein R2 represents CONR4aR4b (wherein R4a and R4b may be the same or different and each represents a hydrogen atom, substituted or unsubstituted lower alkyl, or the like, or R4a and R4b are combined together with the adjacent nitrogen atom thereto to form a substituted or unsubstituted heterocyclic group) or the like, and R3 represents a hydrogen atom, substituted or unsubstituted lower alkyl, or the like] or a pharmaceutically acceptable salt thereof, and the like.

    摘要翻译： 本发明提供了一种Abelson激酶（Abl激酶）抑制剂，其包含式（I）表示的吲唑衍生物作为活性成分（其中R 1表示取代或未取代的芳基或取代或未取代的杂环基）或其药学上可接受的盐 其包含作为活性成分的由式（Ia）表示的吲唑衍生物（其中R 2表示CONR 4 aR 4 b（其中R 4a和R 4b可以相同或不同，各自表示氢原子，取代或未取代的低级）的Abl激酶抑制剂 烷基等，或者R4a和R4b与相邻的氮原子一起形成取代或未取代的杂环基）等，R 3表示氢原子，取代或未取代的低级烷基等，或 其药学上可接受的盐等。