公开(公告)号：US09637480B2

公开(公告)日：2017-05-02

申请号：US13885184

申请日：2011-11-18

申请人： Takeshi Mita ,  Yukihiro Maizuru ,  Ken-ichi Toyama ,  Motoyoshi Iwasa ,  Hotaka Imanaka ,  Hiroto Matsui

发明人： Takeshi Mita ,  Yukihiro Maizuru ,  Ken-ichi Toyama ,  Motoyoshi Iwasa ,  Hotaka Imanaka ,  Hiroto Matsui

IPC分类号： A61K31/42 ,  A61K31/435 ,  C07D413/12 ,  C07D207/18 ,  C07D261/04 ,  C07D401/04 ,  C07D401/14 ,  C07D413/04 ,  C07D413/14 ,  A01N43/36 ,  A01N43/56 ,  A01N43/76 ,  A01N43/78 ,  A01N43/80 ,  C07D409/14

CPC分类号： C07D413/12 ,  A01N43/36 ,  A01N43/40 ,  A01N43/56 ,  A01N43/76 ,  A01N43/78 ,  A01N43/80 ,  A61K31/42 ,  A61K31/435 ,  C07D207/18 ,  C07D261/04 ,  C07D401/04 ,  C07D401/14 ,  C07D409/14 ,  C07D413/04 ,  C07D413/14

摘要： There is provided a novel agent for controlling harmful arthropods or nematodes that are parasites and hygienic pests for animals. An ecto- or endo-parasiticide for mammals or the like comprising as active ingredient, one or more selected from substituted benzamide compounds of formula (1) or salts thereof: wherein A1 is C—X3 or nitrogen atom, etc., A2 and A3 are C—H, etc., A4 is C—H or nitrogen atom, etc., G is G-2a, etc., W is oxygen atom or sulfur atom, X1 is halogen atom, trifluoromethyl, etc., X2 is hydrogen atom, halogen atom, trifluoromethyl, etc., X3 is hydrogen atom, halogen atom, etc., Y1 is hydrogen atom, halogen atom, methyl, etc., R1 is trifluoromethyl, etc., R2 is E-3a, etc., R3 is hydrogen atom, etc., p is an integer of 0 to 2.

公开(公告)号：US20130338197A1

公开(公告)日：2013-12-19

申请号：US13885184

申请日：2011-11-18

申请人： Takeshi Mita ,  Yukihiro Maizuru ,  Ken-ichi Toyama ,  Motoyoshi Iwasa ,  Hotaka Imanaka ,  Hiroto Matsui

发明人： Takeshi Mita ,  Yukihiro Maizuru ,  Ken-ichi Toyama ,  Motoyoshi Iwasa ,  Hotaka Imanaka ,  Hiroto Matsui

IPC分类号： C07D413/12 ,  C07D409/14

CPC分类号： C07D413/12 ,  A01N43/36 ,  A01N43/40 ,  A01N43/56 ,  A01N43/76 ,  A01N43/78 ,  A01N43/80 ,  A61K31/42 ,  A61K31/435 ,  C07D207/18 ,  C07D261/04 ,  C07D401/04 ,  C07D401/14 ,  C07D409/14 ,  C07D413/04 ,  C07D413/14

摘要： There is provided a novel agent for controlling harmful arthropods or nematodes that are parasites and hygienic pests for animals. An ecto- or endo-parasiticide for mammals or the like comprising as active ingredient, one or more selected from substituted benzamide compounds of formula (1) or salts thereof: wherein A1 is C—X3 or nitrogen atom, etc., A2 and A3 are C—H, etc., A4 is C—H or nitrogen atom, etc., G is G-2a, etc., W is oxygen atom or sulfur atom, X1 is halogen atom, trifluoromethyl, etc., X2 is hydrogen atom, halogen atom, trifluoromethyl, etc., X3 is hydrogen atom, halogen atom, etc., Y1 is hydrogen atom, halogen atom, methyl, etc., R1 is trifluoromethyl, etc., R2 is E-3a, etc., R3 is hydrogen atom, etc., p is an integer of 0 to 2.

摘要翻译： 提供了一种用于控制作为动物的寄生虫和卫生有害生物的有害节肢动物或线虫的新型药剂。 包含作为活性成分的一种或多种选自取代的式（1）的苯甲酰胺化合物或其盐的哺乳动物的外消旋物或杀虫剂：其中A1是C-X3或氮原子等，A2和A3 是CH等，A4是CH或氮原子等，G是G-2a等，W是氧原子或硫原子，X 1是卤素原子，三氟甲基等，X 2是氢原子，卤素原子 三氟甲基等，X3为氢原子，卤素原子等，Y1为氢原子，卤原子，甲基等，R1为三氟甲基等，R2为E-3a等，R3为氢原子 等，p为0〜2的整数。