公开(公告)号：US06177462B1

公开(公告)日：2001-01-23

申请号：US09237403

申请日：1999-01-26

Applicant: Zhang Lixin ,  Li Zongcheng ,  Li Zhinian ,  Zhang Hong ,  Liu Changling ,  Li Bin ,  Steven Howard Shaber

Inventor： Zhang Lixin ,  Li Zongcheng ,  Li Zhinian ,  Zhang Hong ,  Liu Changling ,  Li Bin ,  Steven Howard Shaber

IPC: C07C32700

CPC classification number: A01N37/36 ,  A01N37/50 ,  A01N43/40 ,  C07C251/60 ,  C07D213/53 ,  C07D307/52

Abstract: Compounds with fungicidal and insecticidal properties having formula wherein X is N or CH; Y is O, S or NR6; A is independently hydrogen, halo, cyano, (C1-C12)alkyl, or (C1-C12)alkoxy; R1 and R6 is independently hydrogen or (C1-C4)alkyl; R2 is independently hydrogen, (C1-C12)alkyl, halo(C1-C12)alkyl, (C3-C7)cycloalkyl, (C2-C8)alkenyl, halo(C2-C8)alkenyl, (C2-C8)alkynyl, halo(C2-C8)alkynyl, aryl, aralkyl, heterocyclic, or heterocyclic(C1-C4)alkyl; R3 is independently hydrogen or (C1-C4)alkyl; R4 and R5 is independently hydrogen, (C1-C4)alkyl, aryl, aralkyl, aryl(C2-C8)alkenyl, aryl(C2-C8)alkynyl, heterocyclic, or heterocyclic(C1-C4)alkyl wherein if one of R4 and R5 is hydrogen or (C1-C4)alkyl than the other of R4 and R5 is other than hydrogen or (C1-C4)alkyl, and its enantiomers and stereoisomers and agronomically acceptable salts.

Abstract translation: 具有杀虫和杀虫性质的化合物，其具有式（X）的化合物是N或CH; Y是O，S或NR6; A独立地是氢，卤素，氰基，（C1-C12）烷基或（C1-C12）烷氧基; R1和R6独立地是氢或（C1-C4）烷基; R2独立地是氢 ，（C 1 -C 12）烷基，（C 1 -C 12）烷基，（C 3 -C 7）环烷基，（C 2 -C 8）烯基，卤代（C 2 -C 8）烯基，（C 2 -C 8）炔基， （C 1 -C 4）烷基; R 4和R 5独立地是氢，（C 1 -C 4）烷基，芳基，芳烷基，芳基（C 1 -C 4） （C 2 -C 8）烷基，其中如果R 4和R 5中的一个是氢或（C 1 -C 4）烷基，其中R 4和R 5中的另一个不是 氢或（C 1 -C 4）烷基，及其对映异构体和立体异构体和农艺学上可接受的盐。