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1.Process for preparing triazole substituted azaindoleoxoacetic piperazine derivatives and novel salt forms produced therein 有权
标题翻译: 制备三唑取代的亚氮杂双氧乙酸哌嗪衍生物的方法及其中生成的新型盐形式公开(公告)号:US07601715B2
公开(公告)日:2009-10-13
申请号:US11455338
申请日:2006-06-19
申请人: Nachimuthu Soundararajan , Yuping Qiu , Wenhao Hu , David R. Kronenthal , Pierre Sirard , Jean Lajeunesse , Robert Droghini , Ramakrishnan Chidambaram , Xinhua Qian , Kenneth J. Natalie , Shawn K. Pack , Nathan Reising , Erqing Tang , Michael G. Fakes , Qi Gao , Feng Qian , Blisse J. Vakkalagadda , Chiajen Lai , Shan-Ming Kuang
发明人: Nachimuthu Soundararajan , Yuping Qiu , Wenhao Hu , David R. Kronenthal , Pierre Sirard , Jean Lajeunesse , Robert Droghini , Ramakrishnan Chidambaram , Xinhua Qian , Kenneth J. Natalie , Shawn K. Pack , Nathan Reising , Erqing Tang , Michael G. Fakes , Qi Gao , Feng Qian , Blisse J. Vakkalagadda , Chiajen Lai , Shan-Ming Kuang
IPC分类号: A01N43/58 , A61K31/50 , A61K31/497 , C07D239/00 , C07D239/02 , C07D241/00 , C07D241/02 , C07D295/00
CPC分类号: C07D471/04 , C07C311/49 , C07D213/26
摘要: A process is provided for preparing triazole substituted azaindoleoxoacetic piperazine derivative. Novel intermediates produced in the above process, and novel N-1 and amorphous forms of a 1,2,3-triazole substituted azaindoloxoacetic piperazine derivatives and processes for producing such novel forms are also provided.
摘要翻译: 提供制备三唑取代的氮杂糊精乙酸哌嗪衍生物的方法。 还提供了在上述方法中制备的新型中间体和新的N-1和无定形形式的1,2,3-三唑取代的氮杂寡脱氧乙酸哌嗪衍生物及其制备方法。
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2.Process for preparing triazole substituted azaindoleoxoacetic piperazine derivatives and novel salt forms produced therein 有权
标题翻译: 制备三唑取代的亚氮杂双氧乙酸哌嗪衍生物的方法及其中生成的新型盐形式公开(公告)号:US07968718B2
公开(公告)日:2011-06-28
申请号:US12548809
申请日:2009-08-27
申请人: Nachimuthu Soundararajan , Yuping Qiu , Wenhao Hu , David R. Kronenthal , Pierre Sirard , Jean Lajeunesse , Robert Droghini , Ramakrishnan Chidambaram , Xinhua Qian , Kenneth J. Natalie , Shawn K. Pack , Nathan Reising , Erqing Tang , Michael G. Fakes , Qi Gao , Feng Qian , Blisse J. Vakkalagadda , Chiajen Lai , Shan-Ming Kuang
发明人: Nachimuthu Soundararajan , Yuping Qiu , Wenhao Hu , David R. Kronenthal , Pierre Sirard , Jean Lajeunesse , Robert Droghini , Ramakrishnan Chidambaram , Xinhua Qian , Kenneth J. Natalie , Shawn K. Pack , Nathan Reising , Erqing Tang , Michael G. Fakes , Qi Gao , Feng Qian , Blisse J. Vakkalagadda , Chiajen Lai , Shan-Ming Kuang
IPC分类号: C07D471/02
CPC分类号: C07D471/04 , C07C311/49 , C07D213/26
摘要: A process is provided for preparing triazole substituted azaindoleoxoacetic piperazine derivative. Novel intermediates produced in the above process, and novel N-1 and amorphous forms of a 1,2,3-triazole substituted azaindoloxoacetic piperazine derivatives and processes for producing such novel forms are also provided.
摘要翻译: 提供制备三唑取代的氮杂糊精乙酸哌嗪衍生物的方法。 还提供了在上述方法中制备的新型中间体和新的N-1和无定形形式的1,2,3-三唑取代的氮杂寡脱氧乙酸哌嗪衍生物及其制备方法。
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3.PROCESS FOR PREPARING TRIAZOLE SUBSTITUTED AZAINDOLEOXOACETIC PIPERAZINE DERIVATIVES AND NOVEL SALT FORMS PRODUCED THEREIN 有权
标题翻译: 制备三唑取代的氮杂双环氧哌嗪衍生物及其生产的新型盐形式的方法公开(公告)号:US20100076191A1
公开(公告)日:2010-03-25
申请号:US12548809
申请日:2009-08-27
申请人: NACHIMUTHU SOUNDARARAJAN , Yuping Qiu , Wenhao Hu , David R. Kronenthal , Pierre Sirard , Jean Lajeunesse , Robert Droghini , Ramakrishnan Chidambaram , Xinhua Qian , Kenneth J. Natalie , Shawn K. Pack , Nathan Reising , Erqing Tang , Michael G. Fakes , Qi Gao , Feng Qian , Blisse J. Vakkalagadda , Chiajen Lai , Shan-Ming Kuang
发明人: NACHIMUTHU SOUNDARARAJAN , Yuping Qiu , Wenhao Hu , David R. Kronenthal , Pierre Sirard , Jean Lajeunesse , Robert Droghini , Ramakrishnan Chidambaram , Xinhua Qian , Kenneth J. Natalie , Shawn K. Pack , Nathan Reising , Erqing Tang , Michael G. Fakes , Qi Gao , Feng Qian , Blisse J. Vakkalagadda , Chiajen Lai , Shan-Ming Kuang
IPC分类号: C07D471/04
CPC分类号: C07D471/04 , C07C311/49 , C07D213/26
摘要: A process is provided for preparing triazole substituted azaindoleoxoacetic piperazine derivative. Novel intermediates produced in the above process, and novel N-1 and amorphous forms of a 1,2,3-triazole substituted azaindoloxoacetic piperazine derivatives and processes for producing such novel forms are also provided.
摘要翻译: 提供制备三唑取代的氮杂糊精乙酸哌嗪衍生物的方法。 还提供了在上述方法中制备的新型中间体和新的N-1和无定形形式的1,2,3-三唑取代的氮杂寡脱氧乙酸哌嗪衍生物及其制备方法。
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公开(公告)号:US20060293304A1
公开(公告)日:2006-12-28
申请号:US11455338
申请日:2006-06-19
申请人: Nachimuthu Soundararajan , Yuping Qiu , Wenhao Hu , David Kronenthal , Pierre Sirard , Jean Lajeunesse , Robert Droghini , Ramakrishnan Chidambaram , Xinhua Qian , Kenneth Natalie , Shawn Pack , Nathan Reising , Erqing Tang , Michael Fakes , Qi Gao , Feng Qian , Blisse Vakkalagadda , Chiajen Lai , Shan-Ming Kuang
发明人: Nachimuthu Soundararajan , Yuping Qiu , Wenhao Hu , David Kronenthal , Pierre Sirard , Jean Lajeunesse , Robert Droghini , Ramakrishnan Chidambaram , Xinhua Qian , Kenneth Natalie , Shawn Pack , Nathan Reising , Erqing Tang , Michael Fakes , Qi Gao , Feng Qian , Blisse Vakkalagadda , Chiajen Lai , Shan-Ming Kuang
IPC分类号: C07D471/02 , A61K31/55 , A61K31/5377 , A61K31/496 , A61K31/4745
CPC分类号: C07D471/04 , C07C311/49 , C07D213/26
摘要: A process is provided for preparing triazole substituted azaindoleoxoacetic piperazine derivative. Novel intermediates produced in the above process, and novel N-1 and amorphous forms of a 1,2,3-triazole substituted azaindoloxoacetic piperazine derivatives and processes for producing such novel forms are also provided.
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