Quinoline-3-carboxamides, their manufacture and use
    1.
    发明授权
    Quinoline-3-carboxamides, their manufacture and use 失效
    喹啉-3-甲酰胺,其制造和使用

    公开(公告)号:US5972841A

    公开(公告)日:1999-10-26

    申请号:US988765

    申请日:1997-12-11

    IPC分类号: A01N43/42 C07D215/56

    CPC分类号: A01N43/42 C07D215/56

    摘要: Quinoline-3-carboxamides I ##STR1## where R.sup.1 is hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, and the organic radicals may be substituted or unsubstituted;R.sup.2 is hydrogen, hydroxyl, alkoxy, alkenyloxy, dialkylamino, alkyl, alkenyl, alkynyl, cycloalkyl, and the organic radicals may be substituted or unsubstituted;orR.sup.1, R.sup.2 together denote an alkylene chain of 4 to 7 members and which may be interrupted by oxygen, sulfur or N-methyl;R.sup.3 -R.sup.6 are hydrogen, alkyl, alkoxy, haloalkyl, haloalkoxy, alkylthio, haloalkylthio, halogen, cyano or nitro;X is oxygen or sulfur;with the proviso that R.sup.2 is not hydrogen, C.sub.1 -C.sub.3 -alkyl, n-butyl, 3-methylbutyl, cyclohexyl, hexyl, heptyl, octyl, 2-chlorobenzyl, 3-(dimethylamino)propyl, 3-(diethylamino)propyl, 2-morpholinoethyl or 2-(3,4-dimethoxyphenyl)ethyl when R.sup.1 and R.sup.3 to R.sup.6 are hydrogen and X is oxygen, and that R.sup.2 is not benzyl when R.sup.1 is methyl, R.sup.3 to R.sup.6 are hydrogen and X is oxygen, and that R.sup.1 and R.sup.2 do not jointly denote morpholino when R.sup.3 to R.sup.6 are hydrogen and X is oxygen.

    摘要翻译: 其中R 1是氢,烷基,烯基,炔基,环烷基和有机基团的喹啉-3-甲酰胺I可以是取代或未取代的; R2是氢,羟基,烷氧基,烯氧基,二烷基氨基,烷基,烯基,炔基,环烷基,有机基可以是取代或未取代的; 或R 1,R 2一起表示4至7个成员的亚烷基链,并且可被氧,硫或N-甲基中断; R3-R6是氢,烷基,烷氧基,卤代烷基,卤代烷氧基,烷硫基,卤代烷硫基,卤素,氰基或硝基; X是氧或硫; 条件是R2不是氢,C1-C3-烷基,正丁基,3-甲基丁基,环己基,己基,庚基,辛基,2-氯苄基,3-(二甲基氨基)丙基,3-(二乙基氨基)丙基, 当R 1和R 3至R 6为氢且X为氧时,R 2为苄基,R 3为R 6为氢,X为氧时,R 2为苄基, 当R 3至R 6为氢且X为氧时,R 2不共同表示吗啉代。

    Hydroxypyridonecarboxamides, their manufacture and use as herbicides
    3.
    发明授权
    Hydroxypyridonecarboxamides, their manufacture and use as herbicides 失效
    羟基吡啶甲酰胺,其制备和用作除草剂

    公开(公告)号:US5344813A

    公开(公告)日:1994-09-06

    申请号:US981361

    申请日:1992-11-25

    摘要: Hydroxypyridonecarboxamides of the formula I ##STR1## where: X is oxygen or sulfur;R.sup.1, R.sup.2 independently of each other are hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkylalkyl or alkoxy, and these organic radicals are substituted or unsubstituted;R.sup.3 is hydrogen, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, haloalkylthio, halogen or nitro;R.sup.4 is alkyl, alkenyl, alkynyl, cycloalkyl, alkoxy, alkylthio, phenyl or a 5- or 6-membered heterocyclic, aliphatic or aromatic radical containing from one to three heteroatoms selected from the group consisting of oxygen, sulfur and nitrogen, and these radicals are substituted or unsubstituted;with the exception of 6-methyl-4-hydroxypyrid-2-one-3-carboxamide and 6-methyl-4-hydroxypyrid-2-one-3-carboxylic acid-tert-butylamide.

    摘要翻译: 式I的羟基吡啶甲酰胺(I)其中:X是氧或硫; R 1,R 2彼此独立地是氢,烷基,烯基,炔基,环烷基,环烷基烷基或烷氧基,并且这些有机基团是取代或未取代的; R3是氢,烷基,卤代烷基,烷氧基,卤代烷氧基,烷硫基,卤代烷硫基,卤素或硝基; R 4是烷基,烯基,炔基,环烷基,烷氧基,烷硫基,苯基或含有1至3个选自氧,硫和氮的杂原子的5或6元杂环,脂族或芳族基团, 是取代或未取代的; 除了6-甲基-4-羟基吡啶-2-酮-3-甲酰胺和6-甲基-4-羟基吡啶-2-酮-3-羧酸 - 叔丁基酰胺之外。

    Quinoline-3-carboxamides, their manufacture and use
    5.
    发明授权
    Quinoline-3-carboxamides, their manufacture and use 失效
    喹啉-3-甲酰胺,其制造和使用

    公开(公告)号:US5798451A

    公开(公告)日:1998-08-25

    申请号:US794572

    申请日:1997-02-03

    IPC分类号: A01N43/42 C07D215/56

    CPC分类号: A01N43/42 C07D215/56

    摘要: Quinoline-3-carboxamides I ##STR1## where R.sup.1 is hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, and the organic radicals may be substituted or unsubstituted; R.sup.2 is hydrogen, hydroxyl, alkoxy, alkenyloxy, dialkylamino, alkyl, alkenyl, alkynyl, cycloalkyl, and the organic radicals may be substituted or unsubstituted; or R.sup.1, R.sup.2 together denote an alkylene chain of 4 to 7 members and which may be interrupted by oxygen, sulfur or N-methyl; R.sup.3 -R.sup.6 are hydrogen, alkyl, alkoxy, haloalkyl, haloalkoxy, alkylthio, haloalkylthio, halogen, cyano or nitro; X is oxygen or sulfur; with the proviso that R.sup.2 is not hydrogen, C.sub.1 -C.sub.3 -alkyl, n-butyl, 3-methylbutyl, cyclohexyl, hexyl, heptyl, octyl, 2-chlorobenzyl, 3-(dimethylamino)propyl, 3-(diethylamino)propyl, 2-morpholinoethyl or 2-(3,4-dimethoxyphenyl)ethyl when R.sup.1 and R.sup.3 to R.sup.6 are hydrogen and X is oxygen, and that R.sup.2 is not benzyl when R.sup.1 is methyl, R.sup.3 to R.sup.6 are hydrogen and X is oxygen, and that R.sup.1 and R.sup.2 do not jointly denote morpholino when R.sup.3 to R.sup.6 are hydrogen and X is oxygen.

    摘要翻译: 喹啉-3-甲酰胺其中R 1是氢,烷基,烯基,炔基,环烷基和有机基团可以是取代或未取代的(I) R2是氢,羟基,烷氧基,烯氧基,二烷基氨基,烷基,烯基,炔基,环烷基,有机基可以是取代或未取代的; 或R 1,R 2一起表示4至7个成员的亚烷基链,并且可被氧,硫或N-甲基中断; R3-R6是氢,烷基,烷氧基,卤代烷基,卤代烷氧基,烷硫基,卤代烷硫基,卤素,氰基或硝基; X是氧或硫; 条件是R2不是氢,C1-C3-烷基,正丁基,3-甲基丁基,环己基,己基,庚基,辛基,2-氯苄基,3-(二甲基氨基)丙基,3-(二乙基氨基)丙基, 当R 1和R 3至R 6为氢且X为氧时,R 2为苄基,R 3为R 6为氢,X为氧时,R 2为苄基, 当R 3至R 6为氢且X为氧时,R 2不共同表示吗啉代。