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![Processes for the preparation of O-[5-(4-amino-thiazol-2-yl)-pyridin-2-ylmethyl]-hydroxylamine](/abs-image/US/2010/11/30/US07842813B2/abs.jpg.150x150.jpg)
1.发明授权Processes for the preparation of O-[5-(4-amino-thiazol-2-yl)-pyridin-2-ylmethyl]-hydroxylamine 有权制备O- [5-（4-氨基 - 噻唑-2-基） - 吡啶-2-基甲基] - 羟胺的方法公开(公告)号：US07842813B2
公开(公告)日：2010-11-30
申请号：US12437636
申请日：2009-05-08
申请人： Datong Tang , Yinglin Han , Yanhe Huang , Ly Tam Phan , Yat Sun Or , Zhe Wang
发明人： Datong Tang , Yinglin Han , Yanhe Huang , Ly Tam Phan , Yat Sun Or , Zhe Wang
IPC分类号： C07D417/04
CPC分类号： C07D417/04
摘要： The present invention relates generally to novel methods for the synthesis of O-[5-(4-amino-thiazol-2-yl)-pyridin-2-ylmethyl]-hydroxylamine which is an essential reagent in the synthesis of one of the bridged erythromycin derivatives and their respective pharmaceutically acceptable salts in PCT Application WO 03/097659 A1. In particular, the present invention relates to processes and intermediates for the preparation of a compound of formula (Ia):
摘要翻译： 本发明一般涉及合成O- [5-（4-氨基 - 噻唑-2-基） - 吡啶-2-基甲基] - 羟胺的新方法，其是合成桥接的 红霉素衍生物及其各自的药学上可接受的盐在PCT申请WO 03/097659 A1中。 特别地，本发明涉及制备式（Ia）化合物的方法和中间体：
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![PROCESSES FOR THE PREPARATION OF O-[5-(4-AMINO-THIAZOL-2-YL)-PYRIDIN-2-YLMETHYL]-HYDROXYLAMINE](/abs-image/US/2009/11/12/US20090281324A1/abs.jpg.150x150.jpg)
2.发明申请PROCESSES FOR THE PREPARATION OF O-[5-(4-AMINO-THIAZOL-2-YL)-PYRIDIN-2-YLMETHYL]-HYDROXYLAMINE 有权制备O- [5-（4-氨基 - 噻唑-2-基） - 吡啶-2-基]甲基] - 羟基甲酰胺的方法公开(公告)号：US20090281324A1
公开(公告)日：2009-11-12
申请号：US12437636
申请日：2009-05-08
申请人： Datong Tang , Yinglin Han , Yanhe Huang , Ly Tam Phan , Yat Sun Or , Zhe Wang
发明人： Datong Tang , Yinglin Han , Yanhe Huang , Ly Tam Phan , Yat Sun Or , Zhe Wang
IPC分类号： C07D417/04
CPC分类号： C07D417/04
摘要： The present invention relates generally to novel methods for the synthesis of O-[5-(4-amino-thiazol-2-yl)-pyridin-2-ylmethyl]-hydroxylamine which is an essential reagent in the synthesis of one of the bridged erythromycin derivatives and their respective pharmaceutically acceptable salts in PCT Application WO 03/097659 A1. In particular, the present invention relates to processes and intermediates for the preparation of a compound of formula (Ia):
摘要翻译： 本发明一般涉及合成O- [5-（4-氨基 - 噻唑-2-基） - 吡啶-2-基甲基] - 羟胺的新方法，其是合成桥接的 红霉素衍生物及其各自的药学上可接受的盐在PCT申请WO 03/097659 A1中。 特别地，本发明涉及制备式（Ia）化合物的方法和中间体：
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