公开(公告)号：US08680290B2

公开(公告)日：2014-03-25

申请号：US11574648

申请日：2005-08-17

申请人： Andrew Plant ,  Jutta Elisabeth Boehmer ,  Janice Black ,  Timothy David Sparks

发明人： Andrew Plant ,  Jutta Elisabeth Boehmer ,  Janice Black ,  Timothy David Sparks

IPC分类号： C07D261/10 ,  A61K31/421

CPC分类号： C07D261/10 ,  C07D413/12 ,  C07D417/12

摘要： Compounds of formula (I) wherein the substituents are as defined in claim 1, are suitable for use as herbicides. Also claimed is a process for the preparation of compounds of the formula I, wherein m is 2 and n is 1, and the other substituents are defined as in claim 1, formula (Ia) by reacting a compound of the formula Ia in a single step or stepwise in succession with compounds of the formula R5—X and/or R6—X, wherein R5 and R6 are as defined in claim 1, and X is a leaving group, and a process for the preparation of compounds of the formula I, wherein R6 is C1-C10alkyl or halogen, m is 2 and n is 1, and the other substituents are defined as in claim 1, formula (Ib) by reacting a compound of the formula Ib with a compound of the formula R5—X, wherein R5 is as defined in claim 1, and X is a leaving group, and a process for the preparation of compounds of the formula I, wherein R5 is chlorine, bromine or iodine, m is 1 or 2, and n is 1, and the other substituents are defined as in claim 1, formula (Ic) by reacting a compound of the formula 1e with an N-halosuccinimide and an oxidising agent.

摘要翻译： 其中取代基如权利要求1中所定义的式（I）化合物适合用作除草剂。 还要求保护的是制备式I化合物的方法，其中m为2且n为1，其它取代基如权利要求1，式（Ia）所定义，通过使式Ia化合物在单一 与式R 5 -X和/或R 6 -X的化合物连续进行步骤或分步步骤，其中R 5和R 6如权利要求1中所定义，X为离去基团，以及制备式I化合物的方法 其中R 6为C 1 -C 10烷基或卤素，m为2且n为1，其它取代基如权利要求1所定义，式（Ib）通过式Ib化合物与式R 5 -X 其中R 5如权利要求1所定义，X为离去基团，以及制备式Ⅰ化合物的方法，其中R 5为氯，溴或碘，m为1或2，n为1， 并且其它取代基如权利要求1所定义，式（Ic）通过使式1e的化合物与N-卤代琥珀酰亚胺和氧化剂反应。

公开(公告)号：US20080139390A1

公开(公告)日：2008-06-12

申请号：US11574648

申请日：2005-08-17

申请人： Andrew Plant ,  Jutta Elisabeth Boehmer ,  Janice Black ,  Timothy David Sparks

发明人： Andrew Plant ,  Jutta Elisabeth Boehmer ,  Janice Black ,  Timothy David Sparks

IPC分类号： A01N43/80 ,  A01P13/00 ,  C07D261/10 ,  C07D413/12 ,  C07D417/12

CPC分类号： C07D261/10 ,  C07D413/12 ,  C07D417/12

摘要： Compounds of formula (I) wherein the substituents are as defined in claim 1, are suitable for use as herbicides. Also claimed is a process for the preparation of compounds of the formula I, wherein m is 2 and n is 1, and the other substituents are defined as in claim 1, formula (Ia) by reacting a compound of the formula Ia in a single step or stepwise in succession with compounds of the formula R5—X and/or R6—X, wherein R5 and R6 are as defined in claim 1, and X is a leaving group, and a process for the preparation of compounds of the formula I, wherein R6 is C1-C10alkyl or halogen, m is 2 and n is 1, and the other substituents are defined as in claim 1, formula (Ib) by reacting a compound of the formula Ib with a compound of the formula R5—X, wherein R5 is as defined in claim 1, and X is a leaving group, and a process for the preparation of compounds of the formula I, wherein R5 is chlorine, bromine or iodine, m is 1 or 2, and n is 1, and the other substituents are defined as in claim 1, formula (Ic) by reacting a compound of the formula 1e with an N-halosuccinimide and an oxidising agent.

摘要翻译： 其中取代基如权利要求1中所定义的式（I）化合物适合用作除草剂。 还要求保护的是制备式I化合物的方法，其中m为2且n为1，其它取代基如权利要求1，式（Ia）所定义，通过使式Ia化合物在单一 与式R 5 -X和/或R 6 -X的化合物相继步骤或逐步进行，其中R 5和R 0 > 6 如权利要求1中所定义，X是离去基团，以及制备式I化合物的方法，其中R 6为C 1 烷基或卤素，m是2，n是1，其它取代基如权利要求1式（Ib）所定义，通过使式Ib化合物与 式R 5 -X的化合物，其中R 5如权利要求1中所定义，X为离去基团，和其制备方法 式I其中R 5为氯，溴或碘，m为1或2，n为1，其它取代基定义如下： m 1，式（Ic）通过使式1e的化合物与N-卤代琥珀酰亚胺和氧化剂反应。