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1.INDAZOLES, BENZISOXAZOLES AND BENZISOTHIAZOLES AND THEIR USE AS ESTROGENIC AGENTS 失效
标题翻译: 丁唑,苯唑沙和苯并噻唑及其作为雌激素的用途公开(公告)号:US20110237624A1
公开(公告)日:2011-09-29
申请号:US13152433
申请日:2011-06-03
申请人: Benoit RONDOT , Jean LAFAY , Paule BONNET , Thierry CLERC , Igor DUC , Eric DURANTI , François PUCCIO , Jacqueline SHIELDS , Christian BLOT , Philippe MAILLOS
发明人: Benoit RONDOT , Jean LAFAY , Paule BONNET , Thierry CLERC , Igor DUC , Eric DURANTI , François PUCCIO , Jacqueline SHIELDS , Christian BLOT , Philippe MAILLOS
IPC分类号: A61K31/454 , C07D231/56 , C07D401/06 , C07D261/20 , C07D413/12 , C07D275/04 , A61K31/416 , A61K31/423 , A61K31/428 , A61P35/00 , A61P19/10 , A61P15/00 , A61P25/24
CPC分类号: C07D231/56 , C07D261/20 , C07D275/04 , C07D275/06 , C07D491/06
摘要: The present invention relates to compounds of formula (I): in which R1, R2, R3, X, Y and A are as defined in the specification.The compounds are modulators of the estrogen receptors.
摘要翻译: 本发明涉及式(I)化合物:其中R1,R2,R3,X,Y和A如说明书中所定义。 这些化合物是雌激素受体的调节剂。