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1.COMPOUNDS HAVING MUSCARINIC RECEPTOR ANTAGONIST AND BETA2 ADRENERGIC RECEPTOR AGONIST ACTIVITY 有权
Title translation: 具有肌钙蛋白受体拮抗剂和BETA2 ADRENERGIC受体激动剂的化合物公开(公告)号:US20160346271A1
公开(公告)日:2016-12-01
申请号:US15168466
申请日:2016-05-31
Applicant: CHIESI FARMACEUTICI S.p.A.
Inventor: Laura CARZANIGA , Fabio RANCATI , Andrea RIZZI , Ian LINNEY , Wolfgang SCHMIDT , Michael BARNES , Chris KNIGHT
IPC: A61K31/4709 , A61M16/14 , A61M15/00 , C07D453/02 , A61K9/00
CPC classification number: A61K31/4709 , A61K9/0073 , A61M15/009 , A61M16/14 , A61M2202/064 , C07D453/02
Abstract: Compounds of formula I, defined herein, act both as muscarinic receptor antagonists and beta2 adrenergic receptor agonists and are useful for treating diseases of the respiratory tract.
Abstract translation: 式I定义的化合物既作为毒蕈碱受体拮抗剂和β2肾上腺素能受体激动剂,也可用于治疗呼吸道疾病。