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公开(公告)号：US4079069A
公开(公告)日：1978-03-14
申请号：US794771
申请日：1977-05-09
IPC分类号： C07D471/04 , A23K1/16 , A61K31/505 , A61K31/675 , A61P33/02 , C07D521/00
CPC分类号： A61K31/505 , A23K20/116 , A61K31/675
摘要： 5-Deazariboflavin, its phosphate ester and nontoxic salts thereof and its novel bis(loweralkoxymethylene) derivatives have antiprotozoal and antiparasitic activity. They are particularly useful for controlling cecal and/or intestinal coccidiosis when administered in minor quantities to animals, in particular to poultry, usually in admixture with animal sustenance. The compounds are included in compositions useful for the prevention and treatment of coccidiosis in poultry.
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公开(公告)号：US4290966A
公开(公告)日：1981-09-22
申请号：US193790
申请日：1980-10-03
IPC分类号： C07C59/76 , C07D317/30 , C11C1/00
CPC分类号： C07D317/30 , C07C59/76
摘要： Traumatin, 12-oxo-trans (E) -10-docecenoic acid, is prepared from 10-oxomethyldecanoate by reaction with (triphenylphosphoranylene)acetaldehyde to form 12-oxomethyldodecenoate; blocking the 12-oxo group; hydrolyzing the ester group; and deblocking the 12-oxo group.
摘要翻译： 通过与（三苯基亚磷酰）乙醛反应，由10-氧代甲基癸酸酯制备外消旋，12-氧代 - 反式（E）-10-十六烯酸，形成十二碳烯酸12-氧代甲酯; 封闭了12个氧代基团; 水解酯基; 并将12-氧代基团解封。
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公开(公告)号：US4173631A
公开(公告)日：1979-11-06
申请号：US911619
申请日：1978-06-01
申请人： Donald W. Graham , Edward F. Rogers
发明人： Donald W. Graham , Edward F. Rogers
IPC分类号： C07D475/14 , A61K31/525 , C07H19/04
CPC分类号： C07D475/14
摘要： The novel compound 7-methyl-8-methylamino-10-(1'-D-ribityl)isoalloxazine is prepared. This compound has anticoccidial, antiprotozoal and antiparasitic activity. It is particularly useful for controlling cecal and/or intestinal coccidiosis when administered in minor quantities to animals, in particular to poultry, usually in admixture with animal sustenance.
摘要翻译： 制备新化合物7-甲基-8-甲基氨基-10-（1'-D-核糖基）异吲哚啉。 该化合物具有抗球虫，抗原虫和抗寄生虫活性。 当以少量施用于动物，特别是通常与动物饲养物混合的家禽时，对于控制盲肠和/或肠球虫病尤其有用。
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4.发明授权Compositions for treating coccidiosis containing 5-deazariboflavin and its derivatives 失效用于治疗含有5-二氮唑吗啉及其衍生物的结肠病的组合物
公开(公告)号：US4053602A
公开(公告)日：1977-10-11
申请号：US737890
申请日：1976-11-02
IPC分类号： C07D471/04 , A23K1/16 , A61K31/505 , A61K31/675 , A61P33/02
CPC分类号： A61K31/505 , A23K20/116 , A61K31/675
摘要： 5-Deazariboflavin, its phosphate ester and non-toxic salts thereof and its novel bis(loweralkoxymethylene) derivatives have antiprotozoal and antiparasitic activity. They are particularly useful for controlling cecal and/or intestinal coccidiosis when administered in minor quantities to animals, in particular to poultry, usually in admixture with animal sustenance. The compounds are included in compositions useful for the prevention and treatment of coccidiosis in poultry.
摘要翻译： 5-脱氮甲黄蛋白，其磷酸酯和无毒盐及其新型双（低级烷氧基亚甲基）衍生物具有抗原虫和抗寄生虫活性。 当少量给予动物，特别是通常与动物饲养物混合的家禽时，它们特别有用于控制盲肠和/或肠球虫病。 该化合物包括在用于预防和治疗家禽中的球虫病的组合物中。
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公开(公告)号：US5147868A
公开(公告)日：1992-09-15
申请号：US839725
申请日：1992-02-19
IPC分类号： A61K31/40 , C07D307/16 , C07D477/02
CPC分类号： C07D477/02 , A61K31/40 , C07D307/16
摘要： Novel chemical compounds are provided which selectively inhibit the metabolism of dipeptidase (E.C.3.4.13.11) and therefore are useful in combination with antibacterial products. These chemical compounds are z-2-acylamino-3-monosubstituted propenoates.
摘要翻译： 提供了选择性抑制二肽酶代谢（E.C.3.4.13.11）的新型化合物，因此可与抗菌产品组合使用。 这些化合物是z-2-酰基氨基-3-单取代的丙烯酸酯。
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公开(公告)号：US4091094A
公开(公告)日：1978-05-23
申请号：US716497
申请日：1976-08-23
申请人： Donald W. Graham , Edward F. Rogers
发明人： Donald W. Graham , Edward F. Rogers
IPC分类号： C07D213/74 , C07D471/14 , A61K31/525 , C07H19/22
CPC分类号： C07D213/74 , C07D471/14
摘要： The novel compound 9-azariboflavin is prepared. This compound has anticoccidial, antiprotozoal and antiparasitic activity. It is particularly useful for controlling cecal and/or intestinal coccidiosis when administered in minor quantities to animals, in particular to poultry, usually in admixture with animal sustenance.
摘要翻译： 制备新化合物9-氮杂黄豆素。 该化合物具有抗球虫，抗原虫和抗寄生虫活性。 当以少量施用于动物，特别是通常与动物饲养物混合的家禽时，对于控制盲肠和/或肠球虫病尤其有用。
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公开(公告)号：US5952788A
公开(公告)日：1999-09-14
申请号：US617173
申请日：1996-03-18
IPC分类号： H05B37/02
CPC分类号： G09G3/22 , G09G2320/0209 , G09G2330/021 , G09G2330/028
摘要： A drive circuit for controlling a vacuum fluorescent display is provided. A charge storage device is connected between signal ground or a voltage supply and a display element. One multiway switch or two single-position switches are connected to the display element opposite the charge storage device. In either configuration, the switch or switches are controlled by an oscillator which, by toggling the switch or switches, alternates the configuration of the circuit to charge or discharge the charge storage device through the display element. The charge storage device and the display element may be connected to a regulated voltage which is maintained at a potential above the grid voltage to reduce cross-talk in the display. The switching operation is break before make and produces an AC voltage across the display element.
摘要翻译： 提供一种用于控制真空荧光显示器的驱动电路。 电荷存储装置连接在信号地或电压源与显示元件之间。 一个多路开关或两个单位开关连接到与电荷存储装置相对的显示元件。 在任一配置中，开关或开关由振荡器控制，振荡器通过切换开关或开关来交替电路的配置以通过显示元件对电荷存储装置进行充电或放电。 电荷存储装置和显示元件可以连接到保持在电网电压以上的电压的调节电压，以减少显示器中的串扰。 切换操作在make之前断开，并在显示元件上产生交流电压。
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8.发明授权16-substituted-6-aza-androsten-4-ene-3-ones as 5-.alpha.-reductase inhibitors 失效16-取代-6-氮杂 - 雄-4-烯-3-酮作为5-α-还原酶抑制剂
公开(公告)号：US5741795A
公开(公告)日：1998-04-21
申请号：US732953
申请日：1996-10-17
IPC分类号： A61K31/58 , A61K31/00 , A61P5/28 , C07D221/18 , C07J31/00 , C07J73/00 , A61K31/715
CPC分类号： A61K31/58 , C07D221/18 , C07J31/006 , C07J73/005
摘要： Compounds of the formula I ##STR1## are inhibitors of 5.alpha.-reductase, and are useful for the treatment of hyperandrogenic disorders such as acne vulgaris, seborrhea, female hirsutism, male pattern baldness, prostatic carcinoma, prostatitis and benign prostatic hyperplasia.
摘要翻译： 式I的化合物是5α-还原酶的抑制剂，可用于治疗高雄激素性疾病，如寻常痤疮，皮脂溢，女性多毛症，男性型秃发，前列腺癌，前列腺炎和良性前列腺增生。
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9.发明授权Substituted 3-phenanthridinone derivatives as 5-alpha-reductase inhibitors 失效取代的3-菲啶酮衍生物作为5-α-还原酶抑制剂
公开(公告)号：US5621104A
公开(公告)日：1997-04-15
申请号：US522350
申请日：1995-09-15
IPC分类号： C07D221/12 , C07D401/12
CPC分类号： C07D221/12
摘要： The present invention provides for the preparation of compounds,namely, 3-phenanthridinones and their derivatives and their unique ability to inhibit 5-alpha-reductase or their isozymes thereof in mammals enabling said compounds for treating hyperandrogenic conditions of acne, androgenic alopecia, male pattern baldness,female hirsutism,benign prostatic hyperplasia, prostatitis and prostatic cancer.
摘要翻译： PCT No.PCT / US94 / 03080 Sec。 371 1995年9月15日第 102（e）日期1995年9月15日PCT 1994年3月22日PCT公布。 公开号WO94 / 21614 日期1994年9月29日本发明提供化合物的制备，即3-菲啶酮及其衍生物及其在哺乳动物中抑制5-α-还原酶或其同功酶的独特能力，使所述化合物能治疗痤疮的雄激素过多症状， 雄激素性脱发，男性型秃发，女性多毛症，良性前列腺增生，前列腺炎和前列腺癌。
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公开(公告)号：US4094976A
公开(公告)日：1978-06-13
申请号：US755366
申请日：1976-12-29
IPC分类号： A61K31/63 , A61K31/635 , A61K31/40 , A61K31/65
CPC分类号： A61K31/63 , A61K31/635
摘要： Novel anticoccidial poultry compositions comprising an anticoccidially effective amount of a compound of the formula: ##STR1## wherein n is 3, 4 or 5 and R is hydrogen or an acyl radical derived from a non-toxic carboxylic acid or a non-toxic acid addition salt thereof methods of combatting poultry coccidiosis, novel compounds and methods of preparing these novel compounds.
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