公开(公告)号：US20020183314A1

公开(公告)日：2002-12-05

申请号：US10080503

申请日：2002-02-22

Applicant: Ligand Pharmaceuticals Incorporated

Inventor： Robert I. Higuchi ,  Lin Zhi ,  Donald S. Karanewsky ,  Anthony W. Thompson ,  Thomas R. Caferro ,  Neelakandha S. Mani ,  Jyun-Hung Chen ,  Marquis L. Cummings ,  James P. Edwards ,  Mark E. Adams ,  Charlotte L.F. Deckhut

IPC: C07D471/02 ,  C07D491/02 ,  C07D498/02

CPC classification number: C07D498/04 ,  C07D498/14 ,  Y02P20/582

Abstract: Novel non-steroidal tricyclic quinolinone and tricyclic quinoline compounds and compositions that are agonists, partial agonists and/or antagonists for androgen receptors (AR), their preparation and their uses are described.

Abstract translation: 描述了新型非甾体三环喹啉酮和三环喹啉化合物以及作为雄激素受体（AR）的激动剂，部分激动剂和/或拮抗剂及其用途的组合物及其用途。