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1.
公开(公告)号:US08846672B2
公开(公告)日:2014-09-30
申请号:US13993692
申请日:2011-12-16
申请人: Ludwig Paul Cooymans , Lili Hu , Tim Hugo Maria Jonckers , Pierre Jean-Marie Bernard Raboisson , Abdellah Tahri , Steven Maurice Paula Van Hoof , Sandrine Marie Helene Vendeville
发明人: Ludwig Paul Cooymans , Lili Hu , Tim Hugo Maria Jonckers , Pierre Jean-Marie Bernard Raboisson , Abdellah Tahri , Steven Maurice Paula Van Hoof , Sandrine Marie Helene Vendeville
IPC分类号: A61K31/5377 , A61K31/496 , A61K31/495 , A61K31/4427 , C07D413/14 , C07D417/04 , C07D487/04 , C07D471/04
CPC分类号: C07D487/04 , C07D471/04
摘要: A compound satisfying formula I, a prodrug, N-oxide, addition salt, quaternary amine, metal complex, or a stereochemically isomeric form thereof; compositions contain these compounds as active ingredient and processes for preparing these compounds and compositions.
摘要翻译: 满足式I的化合物,前药,N-氧化物,加成盐,季胺,金属络合物或其立体化学异构形式; 组合物含有这些化合物作为活性成分和制备这些化合物和组合物的方法。
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公开(公告)号:US20130324527A1
公开(公告)日:2013-12-05
申请号:US13993692
申请日:2011-12-16
申请人: Ludwig Paul Cooymans , Lili Hu , Tim Hugo Maria Jonckers , Pierre Jean-Marie Bernard Raboisson , Abdella Tahri , Steven Maurice Paula Van Hoof , Sandrine Marie Helene Vendeville
发明人: Ludwig Paul Cooymans , Lili Hu , Tim Hugo Maria Jonckers , Pierre Jean-Marie Bernard Raboisson , Abdella Tahri , Steven Maurice Paula Van Hoof , Sandrine Marie Helene Vendeville
IPC分类号: C07D487/04 , C07D471/04
CPC分类号: C07D487/04 , C07D471/04
摘要: A compound satisfying formula I, a prodrug, N-oxide, addition salt, quaternary amine, metal complex, or a stereochemically isomeric form thereof: compositions contain these compounds as active ingredient and processes for preparing these compounds and compositions.
摘要翻译: 满足式I的化合物,前药,N-氧化物,加成盐,季胺,金属络合物或其立体化学异构形式:含有这些化合物作为活性成分的组合物和制备这些化合物和组合物的方法。
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公开(公告)号:US20130267555A1
公开(公告)日:2013-10-10
申请号:US13993200
申请日:2011-12-16
申请人: Ludwig Paul Cooymans , Samuël Dominique Demin , Lili Hu , Tim Hugo Maria Jonckers , Pierre Jean-Marie Bernard Raboisson , Abdellah Tahri , Sandrine Marie Helene Vendeville
发明人: Ludwig Paul Cooymans , Samuël Dominique Demin , Lili Hu , Tim Hugo Maria Jonckers , Pierre Jean-Marie Bernard Raboisson , Abdellah Tahri , Sandrine Marie Helene Vendeville
IPC分类号: C07D471/04
CPC分类号: C07D471/04 , C07D209/10 , C07D209/12 , C07D235/26 , C07D403/06
摘要: Indoles having inhibitory activity on RSV replication and having the formula I the prodrugs, N-oxides, addition salts, quaternary amines, metal complexes and stereochemically isomeric forms thereof; compositions containing these compounds as active ingredient and processes for preparing these compounds and compositions.
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公开(公告)号:US20130267556A1
公开(公告)日:2013-10-10
申请号:US13993543
申请日:2011-12-16
申请人: Ludwig Paul Cooymans , Samuël Dominique Demin , Lili Hu , Tim Hugo Maria Jonckers , Pierre Jean-Marie Bernard Raboisson , Abdellah Tahri , Sandrine Marie Helene Vendeville
发明人: Ludwig Paul Cooymans , Samuël Dominique Demin , Lili Hu , Tim Hugo Maria Jonckers , Pierre Jean-Marie Bernard Raboisson , Abdellah Tahri , Sandrine Marie Helene Vendeville
IPC分类号: C07D471/04
CPC分类号: C07D519/00 , A61K31/437 , C07D471/04
摘要: Azaindoles having inhibitory activity on RSV replication and having the formula I compositions containing these compounds as active ingredient and processes for preparing these compounds and compositions.
摘要翻译: 对RSV复制具有抑制活性的Azaindoles和具有含有这些化合物作为活性成分的式I组合物和制备这些化合物和组合物的方法。
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公开(公告)号:US20130261151A1
公开(公告)日:2013-10-03
申请号:US13993141
申请日:2011-12-16
申请人: Ludwig Paul Cooymans , Samuël Dominique Demin , Lili Hu , Tim Hugo Maria Jonckers , Pierre Jean-Marie Bernard Raboisson , Abdellah Tahri , Sandrine Marie Helene Vendeville
发明人: Ludwig Paul Cooymans , Samuël Dominique Demin , Lili Hu , Tim Hugo Maria Jonckers , Pierre Jean-Marie Bernard Raboisson , Abdellah Tahri , Sandrine Marie Helene Vendeville
IPC分类号: C07D471/04
CPC分类号: C07D519/00 , C07D471/04 , C07F5/025
摘要: A compound satisfying formula I, a prodrug, N-oxide, addition salt, quaternary amine, metal complex, or a stereochemically isomeric form thereof; compositions contain these compounds as active ingredient and processes for preparing these compounds and compositions
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公开(公告)号:US09051317B2
公开(公告)日:2015-06-09
申请号:US13993543
申请日:2011-12-16
申请人: Ludwig Paul Cooymans , Samuël Dominique Demin , Lili Hu , Tim Hugo Maria Jonckers , Pierre Jean-Marie Bernard Raboisson , Abdellah Tahri , Sandrine Marie Helene Vendeville
发明人: Ludwig Paul Cooymans , Samuël Dominique Demin , Lili Hu , Tim Hugo Maria Jonckers , Pierre Jean-Marie Bernard Raboisson , Abdellah Tahri , Sandrine Marie Helene Vendeville
IPC分类号: C07D471/04 , C07D403/06 , C07D513/02 , C07D515/02 , A61K31/437 , A61P31/12
CPC分类号: C07D519/00 , A61K31/437 , C07D471/04
摘要: Azaindoles having inhibitory activity on RSV replication and having the formula I compositions containing these compounds as active ingredient and processes for preparing these compounds and compositions.
摘要翻译: 对RSV复制具有抑制活性的Azaindoles和具有含有这些化合物作为活性成分的式I组合物和制备这些化合物和组合物的方法。
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公开(公告)号:US08865705B2
公开(公告)日:2014-10-21
申请号:US13993107
申请日:2011-12-16
申请人: Ludwig Paul Cooymans , Samuël Dominique Demin , Lili Hu , Tim Hugo Maria Jonckers , Pierre Jean-Marie Bernard Raboisson , Abdellah Tahri , Sandrine Marie Helene Vendeville
发明人: Ludwig Paul Cooymans , Samuël Dominique Demin , Lili Hu , Tim Hugo Maria Jonckers , Pierre Jean-Marie Bernard Raboisson , Abdellah Tahri , Sandrine Marie Helene Vendeville
IPC分类号: C07D471/04
CPC分类号: C07D471/04 , C07D235/26
摘要: Benzimidazoles having inhibitory activity on RSV replication and having the formula the prodrugs, N-oxides, addition salts, quaternary amines, metal complexes and stereochemically isomeric forms thereof, compositions containing these compounds as active ingredient and processes for preparing these compounds and compositions.
摘要翻译: 对RSV复制具有抑制活性的苯并咪唑,其具有前药,N-氧化物,加成盐,季胺,金属络合物及其立体化学异构形式的组合物,含有这些化合物作为活性成分的组合物和制备这些化合物和组合物的方法。
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8.
公开(公告)号:US08927720B2
公开(公告)日:2015-01-06
申请号:US13993141
申请日:2011-12-16
申请人: Ludwig Paul Cooymans , Samuël Dominique Demin , Lili Hu , Tim Hugo Maria Jonckers , Pierre Jean-Marie Bernard Raboisson , Abdellah Tahri , Sandrine Marie Helene Vendeville
发明人: Ludwig Paul Cooymans , Samuël Dominique Demin , Lili Hu , Tim Hugo Maria Jonckers , Pierre Jean-Marie Bernard Raboisson , Abdellah Tahri , Sandrine Marie Helene Vendeville
IPC分类号: C07D471/04 , A61K31/437 , A61P31/12
CPC分类号: C07D519/00 , C07D471/04 , C07F5/025
摘要: A compound satisfying formula I, a prodrug, N-oxide, addition salt, quaternary amine, metal complex, or a stereochemically isomeric form thereof; compositions contain these compounds as active ingredient and processes for preparing these compounds and compositions.
摘要翻译: 满足式I的化合物,前药,N-氧化物,加成盐,季胺,金属络合物或其立体化学异构形式; 组合物含有这些化合物作为活性成分和制备这些化合物和组合物的方法。
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公开(公告)号:US08921560B2
公开(公告)日:2014-12-30
申请号:US13993200
申请日:2011-12-16
申请人: Ludwig Paul Cooymans , Samuël Dominique Demin , Lili Hu , Tim Hugo Maria Jonckers , Pierre Jean-Marie Bernard Raboisson , Abdellah Tahri , Sandrine Marie Helene Vendeville
发明人: Ludwig Paul Cooymans , Samuël Dominique Demin , Lili Hu , Tim Hugo Maria Jonckers , Pierre Jean-Marie Bernard Raboisson , Abdellah Tahri , Sandrine Marie Helene Vendeville
IPC分类号: C07D471/04 , C07D403/06 , C07D513/02 , C07D515/02 , A61K31/437 , A61P31/12
CPC分类号: C07D471/04 , C07D209/10 , C07D209/12 , C07D235/26 , C07D403/06
摘要: Indoles having inhibitory activity on RSV replication and having the formula I the prodrugs, N-oxides, addition salts, quaternary amines, metal complexes and stereochemically isomeric forms thereof; compositions containing these compounds as active ingredient and processes for preparing these compounds and compositions.
摘要翻译: 吲哚对RSV复制具有抑制活性,并具有式I的前药,N-氧化物,加成盐,季胺,金属络合物及其立体化学异构形式; 含有这些化合物作为活性成分的组合物和制备这些化合物和组合物的方法。
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公开(公告)号:US20130267508A1
公开(公告)日:2013-10-10
申请号:US13993107
申请日:2011-12-16
申请人: Ludwig Paul Cooymans , Lili Wu , Tim Hugo Maria Jonckers , Pierre Jean-Marie Bernard Raboisson , Abdellah Tahri , Sandrine Marie Helene Vendeville
发明人: Ludwig Paul Cooymans , Samuël Dominique Demin , Lili Wu , Tim Hugo Maria Jonckers , Pierre Jean-Marie Bernard Raboisson , Abdellah Tahri , Sandrine Marie Helene Vendeville
IPC分类号: C07D471/04
CPC分类号: C07D471/04 , C07D235/26
摘要: Benzimidazoles having inhibitory activity on RSV replication and having the formula the prodrugs, N-oxides, addition salts, quaternary amines, metal complexes and stereochemically isomeric forms thereof, compositions containing these compounds as active ingredient and processes for preparing these compounds and compositions.
摘要翻译: 对RSV复制具有抑制活性的苯并咪唑,其具有前药,N-氧化物,加成盐,季胺,金属络合物及其立体化学异构形式的组合物,含有这些化合物作为活性成分的组合物和制备这些化合物和组合物的方法。
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