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公开(公告)号:US20190233426A1
公开(公告)日:2019-08-01
申请号:US16311575
申请日:2017-06-09
Applicant: Novartis AG
Inventor: Ho Man CHAN , Xingnian Fu , Xiang-Ju Justin Gu , Ying HUANG , Ling LI , Yuan MI , Wei QI , Martin SENDZIK , Yongfeng SUN , Long WANG , Zhengtian YU , Hailong ZHANG , Ji Yue ZHANG , Man ZHANG , Qiong ZHANG , Kehao ZHAO
IPC: C07D487/04 , A61P35/00
Abstract: A compound of Formula (IA), or a pharmaceutically acceptable salt thereof, is provided that has been shown to be useful for treating a PRC2-mediated disease or disorder: wherein A, R3, R4, R6, and R7 are as defined herein.
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公开(公告)号:US20240216378A1
公开(公告)日:2024-07-04
申请号:US18423776
申请日:2024-01-26
Applicant: NOVARTIS AG
Inventor: Ho Man CHAN , Xiang-Ju Justin GU , Ying HUANG , Ling LI , Yuan MI , Wei QI , Martin SENDZIK , Yongfeng SUN , Long WANG , Zhengtian YU , Hailong ZHANG , Ji Yue (Jeff) ZHANG , Man ZHANG , Qiong ZHANG , Kehao ZHAO
IPC: A61K31/519 , A61K31/5377 , A61K31/541 , A61K31/551 , A61K45/06 , C07D487/04
CPC classification number: A61K31/519 , A61K31/5377 , A61K31/541 , A61K31/551 , A61K45/06 , C07D487/04
Abstract: A compound of Formula (I), or a pharmaceutically acceptable salt thereof, is provided that has been shown to be useful for treating a PRC2-mediated disease or disorder:
wherein R1, R2, R3, R4, R5, and n are as defined herein.-
公开(公告)号:US20190202828A1
公开(公告)日:2019-07-04
申请号:US16311621
申请日:2017-06-06
Applicant: Novartis AG
Inventor: Ho Man CHAN , Xingnian Fu , Xiang-Ju Justin Gu , Ying HUANG , Ling LI , Yuan MI , Wei QI , Martin SENDZIK , Yongfeng SUN , Long WANG , Zhengtian YU , Hailong ZHANG , Ji Yue ZHANG , Man ZHANG , Qiong ZHANG , Kehao ZHAO
IPC: C07D471/04 , A61P35/00
Abstract: A compound of Formula (IA), or a pharmaceutically acceptable salt thereof, is provided that has been shown to be useful for treating a PRC2-mediated disease or disorder: wherein A, R6, R7 and R8 are as defined herein.
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公开(公告)号:US20190142837A1
公开(公告)日:2019-05-16
申请号:US16246380
申请日:2019-01-11
Applicant: Novartis AG
Inventor: Ho Man CHAN , Xiang-Ju Justin GU , Ying HUANG , Ling LI , Yuan MI , Wei QI , Martin SENDZIK , Yongfeng SUN , Long WANG , Zhengtian YU , Hailong ZHANG , Ji Yue (Jeff) ZHANG , Man ZHANG , Qiong ZHANG , Kehao ZHAO
IPC: A61K31/519 , A61K45/06 , A61K31/551 , C07D487/04 , A61K31/5377 , A61K31/541
Abstract: A compound of Formula (I), or a pharmaceutically acceptable salt thereof, is provided that has been shown to be useful for treating a PRC2-mediated disease or disorder: wherein R1, R2, R3, R4, R5, and n are as defined herein.
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公开(公告)号:US20230033320A1
公开(公告)日:2023-02-02
申请号:US17505271
申请日:2021-10-19
Applicant: Novartis AG
Inventor: Ho Man CHAN , Xiang-Ju Justin GU , Ying HUANG , Ling LI , Yuan MI , Wei QI , Martin SENDZIK , Yongfeng SUN , Long WANG , Zhengtian YU , Hailong ZHANG , Ji Yue (Jeff) ZHANG , Man ZHANG , Qiong ZHANG , Kehao ZHAO
IPC: A61K31/519 , C07D487/04 , A61K45/06 , A61K31/5377 , A61K31/541 , A61K31/551
Abstract: A compound of Formula (I), or a pharmaceutically acceptable salt thereof, is provided that has been shown to be useful for treating a PRC2-mediated disease or disorder: wherein R1, R2, R3, R4, R5, and n are as defined herein.
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公开(公告)号:US20200323859A1
公开(公告)日:2020-10-15
申请号:US16863631
申请日:2020-04-30
Applicant: Novartis AG
Inventor: Ho Man CHAN , Xiang-Ju Justin GU , Ying HUANG , Ling LI , Yuan MI , Wei QI , Martin SENDZIK , Yongfeng SUN , Long WANG , Zhengtian YU , Hailong ZHANG , Ji Yue (Jeff) ZHANG , Man ZHANG , Qiong ZHANG , Kehao ZHAO
IPC: A61K31/519 , C07D487/04 , A61K45/06 , A61K31/5377 , A61K31/541 , A61K31/551
Abstract: A compound of Formula (I), or a pharmaceutically acceptable salt thereof, is provided that has been shown to be useful for treating a PRC2-mediated disease or disorder: wherein R1, R2, R3, R4, R5, and n are as defined herein.
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