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1.METHOD AND INTERMEDIATES FOR THE PREPARATION OF DERIVATIVES OF N (1-BENZHYDRYLAZETIDIN-3-YL)-N-PHENYLMETHYLSULFONAMIDE 有权
标题翻译: 制备N(1-苯甲酰基-3-氨基)-N-苯基甲基磺酰胺衍生物的方法和中间体公开(公告)号:US20100087414A1
公开(公告)日:2010-04-08
申请号:US12635965
申请日:2009-12-11
申请人: Philippe BOFFELLI , Michel DELTHIL , Luc GRONDARD , Maxime LAMPILAS , Joel MALPART , Stephane MUTTI , Lahlou NAIT-BOUDA , Joerg RIEKE-ZAPP
发明人: Philippe BOFFELLI , Michel DELTHIL , Luc GRONDARD , Maxime LAMPILAS , Joel MALPART , Stephane MUTTI , Lahlou NAIT-BOUDA , Joerg RIEKE-ZAPP
IPC分类号: A61K31/397 , C07C211/01 , C07C231/06 , C07D205/04 , A61P3/00
CPC分类号: C07D205/04
摘要: The invention relates to a novel method for the synthesis of N-{1-[bis(4-chlorophenyl)methyl]azetidin-3-yl}-N-(3,5 -difluorophenyl)methylsulfonamide.
摘要翻译: 本发明涉及一种合成N- {1- [双(4-氯苯基)甲基]吖丁啶-3-基} -N-(3,5-二氟苯基)甲基磺酰胺的新方法。
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2.METHOD AND INTERMEDIATES FOR THE PREPARATION OF DERIVATIVES OF N (1-BENZHYDRYLAZETIDIN-3-YL)-N-PHENYLMETHYLSULFONAMIDE 有权
标题翻译: 用于制备N-(1-苯甲酰氨基-3-基)-N-苯基甲基磺酰胺衍生物的方法和中间体公开(公告)号:US20080312205A1
公开(公告)日:2008-12-18
申请号:US12194644
申请日:2008-08-20
申请人: Philippe BOFFELLI , Michel DELTHIL , Luc GRONDARD , Maxime LAMPILAS , Joel MALPART , Stephane MUTTI , Lahlou NAIT-BOUDA , Joerg RIEKE-ZAPP
发明人: Philippe BOFFELLI , Michel DELTHIL , Luc GRONDARD , Maxime LAMPILAS , Joel MALPART , Stephane MUTTI , Lahlou NAIT-BOUDA , Joerg RIEKE-ZAPP
IPC分类号: A61K31/397 , C07D205/04 , C07C231/06 , A61P3/00
CPC分类号: C07D205/04
摘要: The invention relates to a novel method for the synthesis of N-{1-[bis(4-chlorophenyl)methyl]azetidin-3-yl}-N-(3,5-difluorophenyl)methylsulfonamide.
摘要翻译: 本发明涉及一种合成N- {1- [双(4-氯苯基)甲基]吖丁啶-3-基} -N-(3,5-二氟苯基)甲基磺酰胺的新方法。
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