-
1.1-substituted 4-arylpiperazine as kappa opioid receptor antagonists 有权
Title translation: 1-取代的4-芳基哌嗪作为κ阿片受体拮抗剂公开(公告)号:US09512105B2
公开(公告)日:2016-12-06
申请号:US14364003
申请日:2012-12-10
Applicant: RESEARCH TRIANGLE INSTITUTE
Inventor: Frank I. Carroll , James B. Thomas , Hernan A. Navarro , S. Wayne Mascarella , Scott P. Runyon , Chunyang Jin , Chad M. Kormos
IPC: C07D241/04 , C07D401/12 , C07D295/13
CPC classification number: C07D401/12 , C07D241/04 , C07D295/13
Abstract: Provided are compounds represented by the formula: where R, Y3, R1, R2, R3, R4, R6, G, R7, E1, E2, A, B, W, X, Y and Z are as defined herein.
-
2.1-SUBSTITUTED 4-ARYLPIPERAZINE AS KAPPA OPIOID RECEPTOR ANTAGONISTS 有权
Title translation: 1-取代的4-ARYLPIPERAZINE作为KAPPA阿片受体拮抗剂公开(公告)号:US20150005315A1
公开(公告)日:2015-01-01
申请号:US14364003
申请日:2012-12-10
Applicant: RESEARCH TRIANGLE INSTITUTE
Inventor: Frank I. Carroll , James B. Thomas , Hernan A. Navarro , S. Wayne Mascarella , Scott P. Runyon , Chunyang Jin , Chad M. Kormos
IPC: C07D401/12 , C07D241/04
CPC classification number: C07D401/12 , C07D241/04 , C07D295/13
Abstract: Provided are compounds represented by the formula: where R, Y3, R1, R2, R3, R4, R6, G, R7, E1, E2, A, B, W, X, Y and Z are as defined herein.
Abstract translation: 提供了由下式表示的化合物:其中R,Y3,R1,R2,R3,R4,R6,G,R7,E1,E2,A,B,W,X,Y和Z如本文所定义。
-