公开(公告)号：US07371768B2

公开(公告)日：2008-05-13

申请号：US10355182

申请日：2003-01-31

申请人： Shuko Okui ,  Nobuo Kyomura ,  Toshiki Fukuchi ,  Kazuya Okano ,  Liangyou He ,  Akiko Miyauchi

发明人： Shuko Okui ,  Nobuo Kyomura ,  Toshiki Fukuchi ,  Kazuya Okano ,  Liangyou He ,  Akiko Miyauchi

IPC分类号： A01N43/56

CPC分类号： C07D401/12 ,  A01N43/56

摘要： The present invention relates to pest control agent having systemic activity and a high safety along with a wide insecticidal spectrum and excellent insecticidal activity, which are 1-aryl-3-cyano-5-pyridylalkylaminopyrazole derivatives represented by formula (1): wherein X represents an N or C-halogen atom; R1 represents a haloalkyl group, excluding a perhaloalkyl group; R2 represents a hydrogen atom or an alkyl group, R3 represents a hydrogen atom, an alkyl group, or an acyl group; and R4 represents a hydrogen atom, a hydroxyl group, an alkyl group, a haloalkyl group, an alkoxy group, a haloalkoxy group, an alkylthio group, an alkylsulfinyl group, an alkylsulfonyl group, a halogen atom, a nitro group, or a cyano group.

摘要翻译： 本发明涉及具有全身活性和高安全性以及广泛的杀虫谱和优异的杀虫活性的害虫防治剂，它是由式（1）表示的1-芳基-3-氰基-5-吡啶基烷基氨基吡唑衍生物：其中X表示 N或C-卤素原子; R 1表示不包括全卤代烷基的卤代烷基; R 2表示氢原子或烷基，R 3表示氢原子，烷基或酰基; R 4表示氢原子，羟基，烷基，卤代烷基，烷氧基，卤代烷氧基，烷硫基，烷基亚磺酰基，烷基磺酰基，卤素原子 ，硝基或氰基。

公开(公告)号：US06849633B2

公开(公告)日：2005-02-01

申请号：US10028786

申请日：2001-12-28

申请人： Shuko Okui ,  Nobuo Kyomura ,  Toshiki Fukuchi ,  Ken Tanaka ,  Manabu Katsurada ,  Kazuya Okano ,  Naoko Sumitani ,  Akiko Miyauchi ,  Akiko Yabe

发明人： Shuko Okui ,  Nobuo Kyomura ,  Toshiki Fukuchi ,  Ken Tanaka ,  Manabu Katsurada ,  Kazuya Okano ,  Naoko Sumitani ,  Akiko Miyauchi ,  Akiko Yabe

IPC分类号： A01N43/56 ,  A01N43/58 ,  A01N43/60 ,  A01N47/02 ,  C07D401/12 ,  C07D403/12 ,  C07D401/14

CPC分类号： C07D401/12 ,  A01N43/56 ,  A01N43/58 ,  A01N43/60 ,  A01N47/02 ,  C07D403/12

摘要： The invention provides a novel pest control agent having a high systemic activity and a high safety with reduced adverse influences on the environment neighboring the place to which the agent is applied, and a process for producing the same.Namely, the present invention relates to a novel 1-aryl-3-cyano-5-heteroarylalkylaminopyrazole derivative represented by the following general formula (1) and a process for producing the same, and a pest control agent containing the same as an active ingredient. (wherein X represents N or C-halogen, R1 represents an alkyl group, an alkenyl group, an alkynyl group, or a haloalkyl group, R2 represents hydrogen atom, an alkyl group, or an acyl group, R3 represents hydrogen atom or an alkyl group, A represents any one of the groups represented by A-1 to A-4, R4 represents hydrogen atom, an alkyl group, a halogen atom, and n represents 0, 1, or 2, provided that R1 is a haloalkyl group except a perhaloalkyl group when A is A-1 and n is 0, and that n is not 0 when A is A-4.).

摘要翻译： 本发明提供了一种具有高体系活性和高安全性的新型有害生物防治剂及其对施用该药剂的地方附近的环境的不良影响，以及其制备方法。本发明涉及一种 由以下通式（1）表示的新颖的1-芳基-3-氰基-5-杂芳基烷基氨基吡唑衍生物及其制备方法和含有该有效成分的害虫控制剂（其中X表示N或C - 卤素，R 1表示烷基，烯基，炔基或卤代烷基，R 2表示氢原子，烷基或酰基，R 3表示氢原子或 烷基，A表示由A-1〜A-4表示的基团中的任一个，R 4表示氢原子，烷基，卤素原子，n表示0,1或2，条件是R 当A是A-1且n是0时，除了全卤代烷基之外的卤代烷基，和tha 当A为A-4时，t n不为0。