专利检索 ap:("Tao Wang" OR "Yasutsugu Ueda" OR "Lawrence G. Hamann" OR "Zhongxing Zhang" OR "Zhiwei Yin" OR "Alicia Regueiro-Ren" OR "David J. Carini" OR "Jacob Swidorski" OR "Zheng Liu" OR "Nicolas A. Meanwell" OR "John F. Kadow" OR "Barry L. Johnson") AND inv:"Lawrence G. Hamann" 第 1 页

1.

发明授权
Diketo substituted pyrrolo[2,3-C]pyridines 有权
标题翻译：二酮取代的吡咯并[2,3-C]吡啶

公开(公告)号：US08124615B2

公开(公告)日：2012-02-28

申请号：US13101591

申请日：2011-05-05

申请人： Tao Wang , Yasutsugu Ueda , Lawrence G. Hamann , Zhongxing Zhang , Zhiwei Yin , Alicia Regueiro-Ren , David J. Carini , Jacob Swidorski , Zheng Liu , Barry L. Johnson , Nicolas A. Meanwell , John F. Kadow

发明人： Tao Wang , Yasutsugu Ueda , Lawrence G. Hamann , Zhongxing Zhang , Zhiwei Yin , Alicia Regueiro-Ren , David J. Carini , Jacob Swidorski , Zheng Liu , Barry L. Johnson , Nicolas A. Meanwell , John F. Kadow

IPC分类号： A61K31/44

CPC分类号： C07D487/04 , C07D471/04 , C07D519/00

摘要： Compounds having drug and bio-affecting properties, their pharmaceutical compositions and methods of use are set forth. In particular, diketo fused azolopiperidine and azolopiperazine derivatives of Formula I: that possess unique antiviral activity are provided. These compounds are useful for the treatment of HIV and AIDS.

摘要翻译： 阐述了具有药物和生物影响特性的化合物，其药物组合物和使用方法。特别地，提供具有独特抗病毒活性的二酮稠合偶氮哌啶和式I的偶氮哌嗪衍生物。这些化合物可用于治疗艾滋病毒和艾滋病。

2.

发明申请
DIKETO FUSED AZOLOPIPERIDINES AND AZOLOPIPERAZINES AS ANTI-HIV AGENTS 有权
标题翻译：作为抗HIV药物的DIKETO FASED AZOLOPIPERIDINES和AZOLOPIPERAZINES

公开(公告)号：US20110212971A1

公开(公告)日：2011-09-01

申请号：US13101591

申请日：2011-05-05

申请人： Tao Wang , Yasutsugu Ueda , Lawrence G. Hamann , Zhongxing Zhang , Zhiwei Yin , Alicia Regueiro-Ren , David J. Carini , Jacob Swidorski , Zheng Liu , Nicolas A. Meanwell , John F. Kadow , Barry L. Johnson

发明人： Tao Wang , Yasutsugu Ueda , Lawrence G. Hamann , Zhongxing Zhang , Zhiwei Yin , Alicia Regueiro-Ren , David J. Carini , Jacob Swidorski , Zheng Liu , Nicolas A. Meanwell , John F. Kadow , Barry L. Johnson

IPC分类号： A61K31/4985 , C07D471/04 , A61K31/506 , A61K31/437 , A61K31/497 , C07D241/04 , A61K31/495 , C07D487/04 , A61P31/18

CPC分类号： C07D487/04 , C07D471/04 , C07D519/00

摘要： Compounds having drug and bio-affecting properties, their pharmaceutical compositions and methods of use are set forth. In particular, diketo fused azolopiperidine and azolopiperazine derivatives that possess unique antiviral activity are provided. These compounds are useful for the treatment of HIV and AIDS.

摘要翻译： 阐述了具有药物和生物影响特性的化合物，其药物组合物和使用方法。特别地，提供具有独特抗病毒活性的二酮稠合偶氮哌啶和偶氮哌嗪衍生物。这些化合物可用于治疗艾滋病毒和艾滋病。

3.

发明申请
Diketo Fused Azolopiperidines and Azolopiperazines as Anti-HIV Agents 有权

公开(公告)号：US20100009993A1

公开(公告)日：2010-01-14

申请号：US12490714

申请日：2009-06-24

申请人： Tao Wang , Yasutsugu Ueda , Lawrence G. Hamann , Zhongxing Zhang , Zhiwei Yin , Alicia Regueiro-Ren , David J. Carini , Jacob Swidorski , Zheng Liu , Nicholas A. Meanwell , John F. Kadow , Barry L. Johnson

发明人： Tao Wang , Yasutsugu Ueda , Lawrence G. Hamann , Zhongxing Zhang , Zhiwei Yin , Alicia Regueiro-Ren , David J. Carini , Jacob Swidorski , Zheng Liu , Nicholas A. Meanwell , John F. Kadow , Barry L. Johnson

IPC分类号： A61K31/495 , A61K31/437 , C07D471/04

CPC分类号： C07D487/04 , C07D471/04 , C07D519/00

摘要： Compounds having drug and bio-affecting properties, their pharmaceutical compositions and methods of use are set forth. In particular, diketo fused azolopiperidine and azolopiperazine derivatives that possess unique antiviral activity are provided. These compounds are useful for the treatment of HIV and AIDS.

摘要翻译： 阐述了具有药物和生物影响特性的化合物，其药物组合物和使用方法。特别地，提供具有独特抗病毒活性的二酮稠合偶氮哌啶和偶氮哌嗪衍生物。这些化合物可用于治疗艾滋病毒和艾滋病。

4.

发明授权
Diketo substituted pyrrolo[2,3-c] pyridines 有权
标题翻译：二酮取代的吡咯并[2,3-c]吡啶

公开(公告)号：US07960406B2

公开(公告)日：2011-06-14

申请号：US12490714

申请日：2009-06-24

申请人： Tao Wang , Yasutsugu Ueda , Lawrence G. Hamann , Zhongxing Zhang , Zhiwei Yin , Alicia Regueiro-Ren , David J. Carini , Jacob Swidorski , Zheng Liu , Barry L. Johnson , Nicholas A. Meanwell , John F. Kadow

发明人： Tao Wang , Yasutsugu Ueda , Lawrence G. Hamann , Zhongxing Zhang , Zhiwei Yin , Alicia Regueiro-Ren , David J. Carini , Jacob Swidorski , Zheng Liu , Barry L. Johnson , Nicholas A. Meanwell , John F. Kadow

IPC分类号： A61K31/44

CPC分类号： C07D487/04 , C07D471/04 , C07D519/00

摘要： Compounds having drug and bio-affecting properties, their pharmaceutical compositions and methods of use are set forth. In particular, diketo fused azolopiperidine and azolopiperazine derivatives of Formula I: that possess unique antiviral activity are provided. These compounds are useful for the treatment of HIV and AIDS.

摘要翻译： 阐述了具有药物和生物影响特性的化合物，其药物组合物和使用方法。特别地，提供具有独特抗病毒活性的二酮稠合偶氮哌啶和式I的偶氮哌嗪衍生物。这些化合物可用于治疗艾滋病毒和艾滋病。

5.

发明授权
Diketo-Piperazine and Piperidine derivatives as antiviral agents 有权
标题翻译： Diketo-Piperazine和哌啶衍生物作为抗病毒剂

公开(公告)号：US07807676B2

公开(公告)日：2010-10-05

申请号：US11877001

申请日：2007-10-23

申请人： Tao Wang , John F. Kadow , Zhongxing Zhang , Zhiwei Yin , Nicholas A. Meanwell , Alicia Regueiro-Ren , Jacob Swidorski , Ying Han , David J. Carini , Lawrence G. Hamann

发明人： Tao Wang , John F. Kadow , Zhongxing Zhang , Zhiwei Yin , Nicholas A. Meanwell , Alicia Regueiro-Ren , Jacob Swidorski , Ying Han , David J. Carini , Lawrence G. Hamann

IPC分类号： A61K31/437 , A61K31/501 , A61K31/506 , C07D471/04

CPC分类号： C07D471/04 , C07D403/12 , C07D417/14

摘要： This disclosure provides compounds having drug and bio-affecting properties, their pharmaceutical compositions and method of use. In particular, the disclosure is concerned with diketo piperazine and piperadine derivatives that possess unique antiviral activity. More particularly, the present disclosure relates to compounds useful for the treatment of HIV and AIDS.

摘要翻译： 本公开提供具有药物和生物影响性质的化合物，其药物组合物和使用方法。特别地，本公开涉及具有独特抗病毒活性的二酮哌嗪和哌嗪衍生物。更具体地，本公开涉及可用于治疗HIV和AIDS的化合物。

6.

发明申请
DIKETO-PIPERAZINE AND PIPERIDINE DERIVATIVES AS ANTIVIRAL AGENTS 有权
标题翻译：作为抗病毒剂的二酮 - 哌嗪和哌啶衍生物

公开(公告)号：US20080139572A1

公开(公告)日：2008-06-12

申请号：US11877001

申请日：2007-10-23

申请人： Tao Wang , John F. Kadow , Zhongxing Zhang , Zhiwei Yin , Nicholas A. Meanwell , Alicia Regueiro-Ren , Jacob Swidorski , Ying Han , David J. Carini , Lawrence G. Hamann

发明人： Tao Wang , John F. Kadow , Zhongxing Zhang , Zhiwei Yin , Nicholas A. Meanwell , Alicia Regueiro-Ren , Jacob Swidorski , Ying Han , David J. Carini , Lawrence G. Hamann

IPC分类号： A61K31/496 , C07D401/14 , A61P31/18

CPC分类号： C07D471/04 , C07D403/12 , C07D417/14

摘要： This disclosure provides compounds having drug and bio-affecting properties, their pharmaceutical compositions and method of use. In particular, the disclosure is concerned with diketo piperazine and piperadine derivatives that possess unique antiviral activity. More particularly, the present disclosure relates to compounds useful for the treatment of HIV and AIDS.

摘要翻译： 本公开提供具有药物和生物影响性质的化合物，其药物组合物和使用方法。特别地，本公开涉及具有独特抗病毒活性的二酮哌嗪和哌嗪衍生物。更具体地，本公开涉及可用于治疗HIV和AIDS的化合物。

7.

发明授权
Diketopiperidine derivatives as HIV attachment inhibitors 有权
标题翻译：二酮哌啶衍生物作为HIV附着抑制剂

公开(公告)号：US08242124B2

公开(公告)日：2012-08-14

申请号：US12490727

申请日：2009-06-24

申请人： Alicia Regueiro-Ren , Jacob Swidorski , Zheng Liu , Tao Wang , Zhongxing Zhang , Lawrence G. Hamann , Nicholas A. Meanwell , David J. Carini , Wenying Li

发明人： Alicia Regueiro-Ren , Jacob Swidorski , Zheng Liu , Tao Wang , Zhongxing Zhang , Lawrence G. Hamann , Nicholas A. Meanwell , David J. Carini , Wenying Li

IPC分类号： A61K31/519 , A61K31/44 , C07D471/04

CPC分类号： C07D471/04 , C07D519/00

摘要： Compounds having drug and bio-affecting properties, their pharmaceutical compositions and methods of use are set forth. In particular, diketopiperidine derivatives that possess unique antiviral activity are provided. These compounds are useful for the treatment of HIV and AIDS.

摘要翻译： 阐述了具有药物和生物影响特性的化合物，其药物组合物和使用方法。特别提供具有独特抗病毒活性的二酮哌啶衍生物。这些化合物可用于治疗艾滋病毒和艾滋病。

8.

发明申请
Diketopiperidine Derivatives as HIV Attachment Inhibitors 有权
标题翻译：二酮哌啶衍生物作为HIV附着抑制剂

公开(公告)号：US20090325985A1

公开(公告)日：2009-12-31

申请号：US12490727

申请日：2009-06-24

申请人： Alicia Regueiro-Ren , Jacob Swidorski , Zheng Liu , Tao Wang , Zhongxing Zhang , Lawrence G. Hamann , Nicholas A. Meanwell , David J. Carini , Wenying Li

发明人： Alicia Regueiro-Ren , Jacob Swidorski , Zheng Liu , Tao Wang , Zhongxing Zhang , Lawrence G. Hamann , Nicholas A. Meanwell , David J. Carini , Wenying Li

IPC分类号： A61K31/519 , A61K31/44 , C07D471/04

CPC分类号： C07D471/04 , C07D519/00

摘要： Compounds having drug and bio-affecting properties, their pharmaceutical compositions and methods of use are set forth. In particular, diketopiperidine derivatives that possess unique antiviral activity are provided. These compounds are useful for the treatment of HIV and AIDS.

摘要翻译： 阐述了具有药物和生物影响特性的化合物，其药物组合物和使用方法。特别提供具有独特抗病毒活性的二酮哌啶衍生物。这些化合物可用于治疗艾滋病毒和艾滋病。

9.

发明申请
THIOAMIDE, AMIDOXIME AND AMIDRAZONE DERIVATIVES AS HIV ATTACHMENT INHIBITORS 有权
标题翻译：作为艾滋病毒治疗抑制剂的噻托咪胺，阿米卡星和阿米卡星衍生物

公开(公告)号：US20130102615A1

公开(公告)日：2013-04-25

申请号：US13444104

申请日：2012-04-11

申请人： Nicholas A. Meanwell , Tao Wang , Zhongxing Zhang , Lawrence G. Hamann , John F. Kadow

发明人： Nicholas A. Meanwell , Tao Wang , Zhongxing Zhang , Lawrence G. Hamann , John F. Kadow

IPC分类号： C07D471/04 , A61K31/496 , A61K45/06 , C07D403/06

CPC分类号： C07D471/04 , A61K31/496 , A61K45/06 , C07D209/12 , C07D209/18 , C07D403/06 , A61K2300/00

摘要： A compound of Formula I, including pharmaceutically acceptable salts thereof: wherein A is selected from the group of:

摘要翻译： 式I的化合物，包括其药学上可接受的盐：其中A选自：

10.

发明授权
Thioamide, amidoxime and amidrazone derivatives as HIV attachment inhibitors 有权
标题翻译：硫酰胺，偕胺肟和氨喋呤衍生物作为HIV附着抑制剂

公开(公告)号：US08685982B2

公开(公告)日：2014-04-01

申请号：US13444104

申请日：2012-04-11

申请人： Nicholas A. Meanwell , Tao Wang , Zhongxing Zhang , Lawrence G. Hamann , John F. Kadow

发明人： Nicholas A. Meanwell , Tao Wang , Zhongxing Zhang , Lawrence G. Hamann , John F. Kadow

IPC分类号： A61K31/497

CPC分类号： C07D471/04 , A61K31/496 , A61K45/06 , C07D209/12 , C07D209/18 , C07D403/06 , A61K2300/00

摘要： A compound of Formula I, including pharmaceutically acceptable salts thereof: wherein A is selected from the group of:

摘要翻译： 式I的化合物，包括其药学上可接受的盐：其中A选自：

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