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公开(公告)号:US20120015929A1
公开(公告)日:2012-01-19
申请号:US13245187
申请日:2011-09-26
申请人: Teodozyj Kolasa , Jennifer M. Frost , Meena V. Patel , Steven P. Latshaw , Arturo Perez Medrano , Xueqing Wang , Karin Rose Marie Tietje , Sridhar Peddi , William A. Carroll
发明人: Teodozyj Kolasa , Jennifer M. Frost , Meena V. Patel , Steven P. Latshaw , Arturo Perez Medrano , Xueqing Wang , Karin Rose Marie Tietje , Sridhar Peddi , William A. Carroll
IPC分类号: A61K31/427 , C07D277/46 , C07D417/14 , A61K31/433 , A61P9/00 , A61K31/4439 , A61K31/454 , A61P29/00 , A61P25/00 , A61P11/00 , C07D417/06 , A61K31/426
CPC分类号: C07D417/06
摘要: Disclosed herein are compounds of formula (I) wherein R1, R2, R3, R25a, R26a, X, and n are as defined in the specification. Pharmaceutical compositions comprising such compounds, and methods of treating conditions and disorders using such compounds and pharmaceutical compositions are also described.
摘要翻译: 本文公开了式(I)的化合物,其中R 1,R 2,R 3,R 25a,R 26a,X和n如说明书中所定义。 还描述了包含这些化合物的药物组合物,以及使用这些化合物和药物组合物治疗病症和病症的方法。
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公开(公告)号:US08058293B2
公开(公告)日:2011-11-15
申请号:US12401788
申请日:2009-03-11
申请人: Teodozyj Kolasa , Jennifer M. Frost , Meena V. Patel , Steven P. Latshaw , Arturo Perez Medrano , Xueqing Wang , Karin Rose Marie Tietje , Sridhar Peddi , William A. Carroll
发明人: Teodozyj Kolasa , Jennifer M. Frost , Meena V. Patel , Steven P. Latshaw , Arturo Perez Medrano , Xueqing Wang , Karin Rose Marie Tietje , Sridhar Peddi , William A. Carroll
IPC分类号: A61K31/433 , A61K31/4025 , C07D205/08 , C07D207/12 , C07D285/135
CPC分类号: C07D417/06
摘要: Disclosed herein are compounds of formula (I) wherein R1, R2, R3, R25a, R26a, X, and n are as defined in the specification. Pharmaceutical compositions comprising such compounds, and methods of treating conditions and disorders using such compounds and pharmaceutical compositions are also described.
摘要翻译: 本文公开了式(I)的化合物,其中R 1,R 2,R 3,R 25a,R 26a,X和n如说明书中所定义。 还描述了包含这些化合物的药物组合物,以及使用这些化合物和药物组合物治疗病症和病症的方法。
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公开(公告)号:US20090247500A1
公开(公告)日:2009-10-01
申请号:US12401788
申请日:2009-03-11
申请人: Teodozyj Kolasa , Jennifer M. Frost , Meena V. Patel , Steven P. Latshaw , Arturo Perez Medrano , Xueqing Wang , Karin Rosemarie Tietje , Sridhar Peddi , William A. Carroll
发明人: Teodozyj Kolasa , Jennifer M. Frost , Meena V. Patel , Steven P. Latshaw , Arturo Perez Medrano , Xueqing Wang , Karin Rosemarie Tietje , Sridhar Peddi , William A. Carroll
IPC分类号: A61K31/427 , C07D417/02 , C07D417/14 , A61P25/00 , A61P11/00 , A61P9/00 , A61K31/4439 , A61K31/454
CPC分类号: C07D417/06
摘要: Disclosed herein are compounds of formula (I) wherein R1, R2, R3, R25a, R26a, X, and n are as defined in the specification. Pharmaceutical compositions comprising such compounds, and methods of treating conditions and disorders using such compounds and pharmaceutical compositions are also described.
摘要翻译: 本文公开了式(I)的化合物,其中R 1,R 2,R 3,R 25a,R 26a,X和n如说明书中所定义。 还描述了包含这些化合物的药物组合物,以及使用这些化合物和药物组合物治疗病症和病症的方法。
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公开(公告)号:US06495576B2
公开(公告)日:2002-12-17
申请号:US10046465
申请日:2002-01-14
申请人: Michael E. Kort , Robert J. Gregg , William A. Carroll , Arturo Perez Medrano , Jürgen Dinges , Fatima Z. Basha
发明人: Michael E. Kort , Robert J. Gregg , William A. Carroll , Arturo Perez Medrano , Jürgen Dinges , Fatima Z. Basha
IPC分类号: A61K3144
CPC分类号: C07D213/74 , C07C233/78 , C07C2601/04 , C07D213/75 , C07D213/76 , C07D213/81 , C07D213/82 , C07D241/20 , C07D405/12 , C07D409/12
摘要: Compounds of formula (I) may be useful in treating diseases prevented by or ameliorated with potassium channel openers. Also disclosed are potassium channel opening compositions and a method of opening potassium channels in a mammal
摘要翻译: 式(I)化合物可用于治疗用钾通道开放剂预防或改善的疾病。 还公开了钾通道开放组合物和在哺乳动物中开放钾通道的方法
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