公开(公告)号：US5571830A

公开(公告)日：1996-11-05

申请号：US586119

申请日：1996-01-16

申请人： Winfried Lunkenheimer ,  Heinz-Wilheim Dehne ,  Ulrike Wachendorff-Neumann

发明人： Winfried Lunkenheimer ,  Heinz-Wilheim Dehne ,  Ulrike Wachendorff-Neumann

IPC分类号： A01N43/90 ,  C07D491/04 ,  C07D491/056 ,  C07D491/113 ,  C07D235/02

CPC分类号： C07D491/04 ,  A01N43/90

摘要： New 2-cyanobenzimidazoles of the formula (I) ##STR1## in which R.sup.1, R.sup.2 and A have the meaning given in the description, a preparation process, their use in agriculture, for example against fungi, insects etc., and new intermediates.Formula (I) provides a definition of the compounds; for example they are obtained from suitable 2-cyanobenzimidazoles which are unsubstituted in the 1-position with N,N-dimethylsulphamoyl halide. The 2-cyanobenzimidazoles which are unsubstituted in the 1-position are equally new and can be reacted from suitable phenylenediamines of the formula (IV) with methyl 2,2,2-trichloroacetimidate of the formula (V) to give the 2-trichloromethylbenzimidazoles of the formula (VI), which are equally new and from which the compounds of the formula (II) can subsequently be obtained with ammonia.

摘要翻译： 式（I）的新的2-氰基苯并咪唑其中R1，R2和A具有说明书中给出的含义，制备方法，它们在农业中的用途，例如抗真菌，昆虫等，以及 新中间体 式（I）提供化合物的定义; 例如，它们可由合适的2-氰基苯并咪唑得到，其中N，N-二甲基氨磺酰卤在1位未被取代。 在1-位未被取代的2-氰基苯并咪唑是同等新的，并且可以由适当的式（Ⅳ）亚苯基二胺与式（Ⅴ）的2,2,2-三氯乙酰亚氨酸甲酯反应得到2-（三氟甲基）苯并咪唑 式（VI）同样新，随后可以用氨获得式（II）化合物。