公开(公告)号：US4472395A

公开(公告)日：1984-09-18

申请号：US343054

申请日：1982-01-27

申请人： Wolfgang Kramer ,  Karl H. Buchel ,  Hans-Ludwig Elbe ,  Udo Kraatz ,  Wolf Reiser ,  Andreas Schulze ,  Erik Regel ,  Wilhelm Brandes ,  Paul-Ernest Frohberger

发明人： Wolfgang Kramer ,  Karl H. Buchel ,  Hans-Ludwig Elbe ,  Udo Kraatz ,  Wolf Reiser ,  Andreas Schulze ,  Erik Regel ,  Wilhelm Brandes ,  Paul-Ernest Frohberger

IPC分类号： C07D405/06 ,  A61K31/41 ,  A61P31/04 ,  C07D521/00 ,  A01N43/50 ,  A01N43/64 ,  C07D405/14

CPC分类号： C07D231/12 ,  C07D233/56 ,  C07D249/08

摘要： A 2-azolylmethyl-1,3-dioxolane or -dioxane derivative of the formula ##STR1## in which Az is imidazol-1-yl or 1,2,4-triazol-1-yl,R.sup.1, R.sup.2, R.sup.3 and R.sup.5 each independently is hydrogen or alkyl, orR.sup.1 and R.sup.3 together are an optionally substituted multi-membered methylene bridge,R.sup.4 is hydrogen, optionally substituted alkyl, optionally substituted aryl or optionally substituted aralykyl,m is 0 or 1,R.sup.6 is hydrogen, halogen, cyano, alkyl, optionally substituted aryl, --X--R.sup.7, --COOR.sup.8 or --CONHR.sup.9,X is oxygen, sulphur, SO, or SO.sub.2,R.sup.7 is alkyl, halogenoalkyl, cyano, optionally substituted aralkyl or optionally substituted aryl,R.sup.8 is alkyl,R.sup.9 is alkyl or optionally substituted aryl, andn is 0 or 1, or a plant-tolerated acid addition salt or metal salt complex thereof which possesses fungicidal activity.

摘要翻译： 其中Az为咪唑-1-基或1,2,4-三唑-1-基的式（Ⅰ）的2-吡唑基甲基-1,3-二氧戊环或二恶烷衍生物，R1，R2，R3 R 5和R 5各自独立地为氢或烷基，或者R 1和R 3一起为任选取代的多元亚甲基桥，R 4为氢，任选取代的烷基，任选取代的芳基或任选取代的芳烷基，m为0或1，R 6为氢， 卤素，氰基，烷基，任选取代的芳基，-X-R7，-COOR8或-CONHR9，X是氧，硫，SO或SO2，R7是烷基，卤代烷基，氰基，任选取代的芳烷基或任选取代的芳基， 烷基，R9为烷基或任选取代的芳基，n为0或1，或其具有杀真菌活性的植物耐受酸加成盐或金属盐络合物。