公开(公告)号：US07994094B2

公开(公告)日：2011-08-09

申请号：US12377338

申请日：2007-08-29

申请人： Yasuhiro Endo ,  Go Uenaka ,  Yuichi Shirai

发明人： Yasuhiro Endo ,  Go Uenaka ,  Yuichi Shirai

IPC分类号： A01N43/40 ,  C07D223/00 ,  C07D211/46

CPC分类号： C07D401/14 ,  A01N43/56 ,  A01N43/76 ,  A01N43/78 ,  A01N43/80 ,  A01N43/90 ,  C07D405/14 ,  C07D409/14 ,  C07D413/14 ,  C07D417/14 ,  C07D451/06

摘要： The N-pyridylpiperidine compound of the invention is represented by Formula (1) wherein R1 is a halogen atom, a C1-4 haloalkyl group, a cyano group, a nitro group, or C1-4 alkoxycarbonyl group; R2, R3, R4, R5, R6, R7, R8, and R9 are each independently a hydrogen atom or a C1-4 alkyl group; R10 is a hydrogen atom, etc.; R11 is a halogen atom, etc.; X is an oxygen atom or a sulfur atom, m is an integer of 1 to 4; and n is an integer of 1 or 2. The N-pyridylpiperidine compound of the invention has an excellent miticidal activity against spider mites and rust mites.

摘要翻译： 本发明的N-吡啶基哌啶化合物由式（1）表示，其中R1是卤素原子，C1-4卤代烷基，氰基，硝基或C1-4烷氧基羰基; R2，R3，R4，R5，R6，R7，R8和R9各自独立地为氢原子或C1-4烷基; R10是氢原子等; R11是卤原子等; X是氧原子或硫原子，m是1〜4的整数， n为1或2的整数。本发明的N-吡啶基哌啶化合物对蜘蛛螨和铁锈螨具有优异的杀螨活性。

公开(公告)号：US20100137582A1

公开(公告)日：2010-06-03

申请号：US12377338

申请日：2007-08-29

申请人： Yasuhiro Endo ,  Go Uenaka ,  Yuichi Shirai

发明人： Yasuhiro Endo ,  Go Uenaka ,  Yuichi Shirai

IPC分类号： C07D401/14 ,  C07D223/14 ,  C07D405/14

CPC分类号： C07D401/14 ,  A01N43/56 ,  A01N43/76 ,  A01N43/78 ,  A01N43/80 ,  A01N43/90 ,  C07D405/14 ,  C07D409/14 ,  C07D413/14 ,  C07D417/14 ,  C07D451/06

摘要： The N-pyridylpiperidine compound of the invention is represented by Formula (1) wherein R1 is a halogen atom, a C1-4 haloalkyl group, a cyano group, a nitro group, or C1-4 alkoxycarbonyl group; R2, R3, R4, R5, R6, R7, R8, and R9 are each independently a hydrogen atom or a C1-4 alkyl group; R10 is a hydrogen atom, etc.; R11 is a halogen atom, etc.; X is an oxygen atom or a sulfur atom, m is an integer of 1 to 4; and n is an integer of 1 or 2.The N-pyridylpiperidine compound of the invention has an excellent miticidal activity against spider mites and rust mites.

摘要翻译： 本发明的N-吡啶基哌啶化合物由式（1）表示，其中R1是卤素原子，C1-4卤代烷基，氰基，硝基或C1-4烷氧基羰基; R2，R3，R4，R5，R6，R7，R8和R9各自独立地为氢原子或C1-4烷基; R10是氢原子等; R11是卤原子等; X是氧原子或硫原子，m是1〜4的整数， n为1或2的整数。本发明的N-吡啶基哌啶化合物对蜘蛛螨和铁锈螨具有优异的杀螨活性。

公开(公告)号：US20140148477A1

公开(公告)日：2014-05-29

申请号：US14128807

申请日：2012-07-19

申请人： Yasuhiro Endo ,  Yuichi Shirai

发明人： Yasuhiro Endo ,  Yuichi Shirai

IPC分类号： A61K31/4545 ,  A61K31/439

CPC分类号： A61K31/4545 ,  A61K31/439

摘要： The present invention provides an animal ectoparasite-controlling agent and a method for preventing or treating infection in animals caused by parasites by using the controlling agent. An animal ectoparasite-controlling agent exhibiting excellent insecticidal activity, and a method for preventing or treating infection in animals caused by parasites by using the controlling agent are obtained by using a compound having a pyrazole ring at the 4-position of the piperidine ring as an active ingredient.

摘要翻译： 本发明提供动物外寄生物控制剂和通过使用控制剂预防或治疗由寄生虫引起的动物感染的方法。 通过使用在哌啶环的4位具有吡唑环的化合物作为对象，通过使用控制剂，可以获得表现出优异的杀虫活性的动物外寄生虫控制剂和预防或治疗由寄生虫引起的动物感染的方法 有效成分。