专利检索 ipc:"A06K31/443" 第 1 页

1.

发明授权
Piperidinyl indole and tetrohydropyridinyl indole derivatives and method of their use 失效
标题翻译：哌啶基吲哚和四氢吡啶基吲哚衍生物及其使用方法

公开(公告)号：US07235569B2

公开(公告)日：2007-06-26

申请号：US10835998

申请日：2004-04-30

申请人： Aranapakam Mudumbai Venkatesan , Osvaldo Dos Santos , Yansong Gu

发明人： Aranapakam Mudumbai Venkatesan , Osvaldo Dos Santos , Yansong Gu

IPC分类号： A61K31/4439 , A06K31/443 , C07D401/14

CPC分类号： C07D405/14 , C07D409/14 , C07D471/04

摘要： 3-Piperidin-4-yl-1H-indole and 3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole derivatives are disclosed. Methods of using the derivatives and compositions containing the derivatives in the prevention and/or treatment of serotonin disorders, such as depression and anxiety, are also disclosed. Additionally, processes for the preparation of 3-piperidin-4-yl-1H-indole and 3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole derivatives are disclosed.

摘要翻译： 3-哌啶-4-基-1H-吲哚和3-（1,2,3,6-四氢 - 吡啶-4-基）-1H-吲哚衍生物。还公开了使用含有衍生物的衍生物和组合物在预防和/或治疗5-羟色胺病症例如抑郁和焦虑中的方法。另外，公开了制备3-哌啶-4-基-1H-吲哚和3-（1,2,3,6-四氢 - 吡啶-4-基）-1H-吲哚衍生物的方法。